Discovery of a novel indole series of EP1 receptor antagonists by scaffold hopping
HALL, Adrian, BILLINTON, Andy, THEOBALD, Pamela J, BROWN, Susan H, CHOWDHURY, Anita, GIBLIN, Gerard M. P, GOLDSMITH, Paul, HURST, David N, NAYLOR, Alan, PATEL, Sadhana, SCOCCITTI, Tiziana
Published in Bioorganic & medicinal chemistry letters (15.04.2008)
Published in Bioorganic & medicinal chemistry letters (15.04.2008)
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Discovery of novel biaryl heterocyclic EP1 receptor antagonists
Hall, Adrian, Bit, Rino A., Brown, Susan H., Chaignot, Helene M., Chessell, Iain P., Coleman, Tanya, Giblin, Gerard M.P., Hurst, David N., Kilford, Ian R., Lewell, Xiao Q., Michel, Anton D., Mohamed, Shiyam, Naylor, Alan, Novelli, Riccardo, Skinner, Lee, Spalding, David J., Tang, Sac P., Wilson, Richard J.
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
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The identification of α-ketoamides as potent inhibitors of hepatitis C virus NS3-4A proteinase
BENNETT, J. M, CAMPBELL, A. D, KAY, P. B, O'BRIEN, M. A, KING-UNDERWOOD, J, RAYNHAM, T. M, WILKINSON, C. S, WILKINSON, T. C. I, WILSON, F. X, CAMPBELL, A. J, CARR, M. G, DUNSDON, R. M, GREENING, J. R, HURST, D. N, JENNINGS, N. S, JONES, P. S, JORDAN, S
Published in Bioorganic & medicinal chemistry letters (12.02.2001)
Published in Bioorganic & medicinal chemistry letters (12.02.2001)
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The Design and Synthesis of Potent Inhibitors of Hepatitis C Virus NS3–4A Proteinase
Attwood, MR, Bennett, JM, Campbell, AD, Canning, GGM, Carr, MG, Conway, E, Dunsdon, RM, Greening, JR, Jones, PS, Kay, PB, Handa, BK, Hurst, DN, Jennings, NS, Jordan, S, Keech, E, O'Brien, MA, Overton, HA, King-Underwood, J, Raynham, TM, Stenson, KP, Wilkinson, CS, Wilkinson, TCI, Wilson, FX
Published in Antiviral chemistry & chemotherapy (01.09.1999)
Published in Antiviral chemistry & chemotherapy (01.09.1999)
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Synthesis of homochiral potassium channel openers: role of the benzopyranyl 3-hydroxyl group in cromakalim and pyridine N-oxides in determining the biological activities of enantiomers
Attwood, Michael R., Brown, Barbara S., Dunsdon, Rachel M., Hurst, David N., Jones, Philip S., Kay, Paul B.
Published in Bioorganic & medicinal chemistry letters (1992)
Published in Bioorganic & medicinal chemistry letters (1992)
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beta.-Adrenoceptor activity of the stereoisomers of the bufuralol alcohol and ketone metabolites
Machin, Peter J, Hurst, David N, Osbond, John M
Published in Journal of medicinal chemistry (01.11.1985)
Published in Journal of medicinal chemistry (01.11.1985)
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Beta 1-selective adrenoceptor antagonists. 3. 4-Azolyl-linked phenoxypropanolamines
Machin, P J, Hurst, D N, Bradshaw, R M, Blaber, L C, Burden, D T, Melarange, R A
Published in Journal of medicinal chemistry (01.04.1984)
Published in Journal of medicinal chemistry (01.04.1984)
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beta 1-selective adrenoceptor antagonists. 2. 4-ether-linked phenoxypropanolamines
Machin, P J, Hurst, D N, Bradshaw, R M, Blaber, L C, Burden, D T, Fryer, A D, Melarange, R A, Shivdasani, C
Published in Journal of medicinal chemistry (01.11.1983)
Published in Journal of medicinal chemistry (01.11.1983)
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