Ligand-induced changes in hepatitis C virus NS5B polymerase structure
Rigat, Karen, Wang, Yi, Hudyma, Thomas W., Ding, Min, Zheng, Xiaofan, Gentles, Robert G., Beno, Brett R., Gao, Min, Roberts, Susan B.
Published in Antiviral research (01.11.2010)
Published in Antiviral research (01.11.2010)
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Syntheses and initial evaluation of a series of indolo-fused heterocyclic inhibitors of the polymerase enzyme (NS5B) of the hepatitis C virus
Zheng, Xiaofan, Hudyma, Thomas W., Martin, Scott W., Bergstrom, Carl, Ding, Min, He, Feng, Romine, Jeffrey, Poss, Michael A., Kadow, John F., Chang, Chong-Hwan, Wan, John, Witmer, Mark R., Morin, Paul, Camac, Daniel M., Sheriff, Steven, Beno, Brett R., Rigat, Karen L., Wang, Ying-Kai, Fridell, Robert, Lemm, Julie, Qiu, Dike, Liu, Mengping, Voss, Stacey, Pelosi, Lenore, Roberts, Susan B., Gao, Min, Knipe, Jay, Gentles, Robert G.
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Synthesis and SAR studies of novel heteroaryl fused tetracyclic indole-diamide compounds: Potent allosteric inhibitors of the hepatitis C virus NS5B polymerase
Ding, Min, He, Feng, Hudyma, Thomas W., Zheng, Xiaofan, Poss, Michael A., Kadow, John F., Beno, Brett R., Rigat, Karen L., Wang, Ying-Kai, Fridell, Robert A., Lemm, Julie A., Qiu, Dike, Liu, Mengping, Voss, Stacey, Pelosi, Lenore A., Roberts, Susan B., Gao, Min, Knipe, Jay, Gentles, Robert G.
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
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Phosphonooxymethyl prodrugs of the broad spectrum antifungal azole, ravuconazole: Synthesis and biological properties
UEDA, Yasutsugu, MATISKELLA, John D, VARIA, Sailesh, KNIPE, Jay, MING ZHENG, MATHEW, Marina, MOSURE, Kathy, CLARK, Junius, LAMB, Lucinda, MEDIN, Ivette, QI GAO, HUANG, Stella, GOLIK, Jerzy, CHEN, Chung-Pin, BRONSON, Joanne J, CONNOLLY, Timothy P, HUDYMA, Thomas W, VENKATESH, Srini, DALI, Mandar, KANG, Shin-Hong, BARBOUR, Nancy, TEJWANI, Ravi
Published in Bioorganic & medicinal chemistry letters (03.11.2003)
Published in Bioorganic & medicinal chemistry letters (03.11.2003)
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Novel semi-synthetic nocathiacin antibiotics: synthesis and antibacterial activity of bis- and mono- O-alkylated derivatives
Regueiro-Ren, Alicia, Naidu, B.Narasimhulu, Zheng, Xiaofan, Hudyma, Thomas W., Connolly, Timothy P., Matiskella, John D., Zhang, Yunhui, Kim, Oak K., Sorenson, Margaret E., Pucci, Michael, Clark, Junius, Bronson, Joanne J., Ueda, Yasutsugu
Published in Bioorganic & medicinal chemistry letters (05.01.2004)
Published in Bioorganic & medicinal chemistry letters (05.01.2004)
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Discovery and Preclinical Characterization of the Cyclopropylindolobenzazepine BMS-791325, A Potent Allosteric Inhibitor of the Hepatitis C Virus NS5B Polymerase
Gentles, Robert G., Ding, Min, Bender, John A., Bergstrom, Carl P., Grant-Young, Katharine, Hewawasam, Piyasena, Hudyma, Thomas, Martin, Scott, Nickel, Andrew, Regueiro-Ren, Alicia, Tu, Yong, Yang, Zhong, Yeung, Kap-Sun, Zheng, Xiaofan, Chao, Sam, Sun, Jung-Hui, Beno, Brett R., Camac, Daniel M., Chang, Chong-Hwan, Gao, Mian, Morin, Paul E., Sheriff, Steven, Tredup, Jeff, Wan, John, Witmer, Mark R., Xie, Dianlin, Hanumegowda, Umesh, Knipe, Jay, Mosure, Kathy, Santone, Kenneth S., Parker, Dawn D., Zhuo, Xiaoliang, Lemm, Julie, Liu, Mengping, Pelosi, Lenore, Rigat, Karen, Voss, Stacey, Wang, Yi, Wang, Ying-Kai, Colonno, Richard J., Gao, Min, Roberts, Susan B., Gao, Qi, Ng, Alicia, Meanwell, Nicholas A, Kadow, John F.
Published in Journal of medicinal chemistry (13.03.2014)
Published in Journal of medicinal chemistry (13.03.2014)
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A practical and efficient synthesis of 6-carboalkoxy-13-cycloalkyl-5H-indolo[2,1-a][2]benzazepine-10-carboxylic acid derivatives
Hewawasam, Piyasena, Tu, Yong, Hudyma, Thomas W., Zhang, Xiaofan, Gentles, Robert G., Kadow, John F., Meanwell, Nicholas A.
Published in Tetrahedron letters (05.02.2014)
Published in Tetrahedron letters (05.02.2014)
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A practical and efficient synthesis of 6-carboalkoxy-13-cycloalkyl-5H-indolo[2,1-a][2]benzazepine-10-carb o xylic acid derivatives
Hewawasam, Piyasena, Tu, Yong, Hudyma, Thomas, Zhang, Xiaofan, Gentles, Robert, Kadow, John, Meanwell, Nicholas
Published in Tetrahedron letters (01.01.2014)
Published in Tetrahedron letters (01.01.2014)
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ChemInform Abstract: A Practical and Efficient Synthesis of 6-Carboalkoxy-13-cycloalkyl-5H-indolo[2,1-a] [2]benzazepine-10-carboxylic Acid Derivatives
Hewawasam, Piyasena, Tu, Yong, Hudyma, Thomas W., Zhang, Xiaofan, Gentles, Robert G., Kadow, John F., Meanwell, Nicholas A.
Published in ChemInform (15.07.2014)
Published in ChemInform (15.07.2014)
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Trypsin Digestion of Hepatitis C Virus NS5B Polymerase Exposes a Hinge at the Active Site
Rigat, Karen, Wang, Yi, Hudyma, Thomas W., Ding, Min, Zheng, Xiaofan, Gentles, Robert G., Beno, Brett R., Gao, Min, Roberts, Susan B.
Published in Antiviral research (01.04.2010)
Published in Antiviral research (01.04.2010)
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Antiallergy agents. 2. 2-Phenyl-5-(1H-tetrazol-5-yl)pyrimidin-4(3H)-ones
Juby, Peter F, Hudyma, Thomas W, Brown, Myron, Essery, John M, Partyka, Richard A
Published in Journal of medicinal chemistry (01.10.1982)
Published in Journal of medicinal chemistry (01.10.1982)
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Antiallergy agents. 1. 1,6-Dihydro-6-oxo-2-phenylpyrimidine-5-carboxylic acids and esters
Juby, Peter F, Hudyma, Thomas W, Brown, Myron, Essery, John M, Partyka, Richard A
Published in Journal of medicinal chemistry (01.03.1979)
Published in Journal of medicinal chemistry (01.03.1979)
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Synthesis and antibacterial activity of O-substituted nocathiacin I derivatives
NARASIMHULU NAIDU, B, SORENSON, Margaret E, HUDYMA, Thomas, XIAOFAN ZHENG, YUNHUI ZHANG, BRONSON, Joanne J, PUCCI, Michael J, CLARK, Junius M, UEDA, Yasutsugu
Published in Bioorganic & medicinal chemistry letters (16.07.2004)
Published in Bioorganic & medicinal chemistry letters (16.07.2004)
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CEPHALOSPORIN SALTS
LIPPER, ROBERT A, SHIH, KUN M, BOETTGER, SUSAN D, KAPLAN, MURRAY A, HUDYMA, THOMAS W
Year of Publication 17.04.1995
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Year of Publication 17.04.1995
Patent
Synthesis and anti-MRSA Activity of Novel Cephalosporin Derivatives
D'Andrea, Stan V., Bonner, Daniel, Bronson, Joanne J., Clark, Junius, Denbleyker, Ken, Fung-Tomc, Joan, Hoeft, Shelley E., Hudyma, Thomas W., Matiskella, John D., Miller, Raymond F., Misco, Peter F., Pucci, Michael, Sterzycki, Roman, Tsai, Yuan, Ueda, Yasutsuga, Wichtowski, John A., Singh, Janak, Kissick, Thomas P., North, Jeffery T., Pullockaran, Annie, Humora, Michael, Boyhan, Brenda, Vu, Truc, Fritz, Alan, Heikes, J., Fox, Rita, Godfrey, Jollie D., Perrone, Robert, Kaplan, Murray, Kronenthal, David, Mueller, Richard H.
Published in Tetrahedron (28.07.2000)
Published in Tetrahedron (28.07.2000)
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Synthesis and structure-activity relationship of C-3 quaternary ammonium cephalosporins exhibiting anti-MRSA activities
Kim, Oak K., Hudyma, Thomas W., Matiskella, John D., Ueda, Yasutsugu, Bronson, Joanne J., Mansuri, Muzammil M.
Published in Bioorganic & medicinal chemistry letters (04.11.1997)
Published in Bioorganic & medicinal chemistry letters (04.11.1997)
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