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Hispidulin attenuates the social withdrawal in isolated disrupted‐in‐schizophrenia‐1 mutant and chronic phencyclidine‐treated mice
Mouri, Akihiro, Lee, Hsin‐Jung, Mamiya, Takayoshi, Aoyama, Yuki, Matsumoto, Yurie, Kubota, Hisayoshi, Huang, Wei‐Jan, Chiou, Lih‐Chu, Nabeshima, Toshitaka
Published in British journal of pharmacology (01.07.2020)
Published in British journal of pharmacology (01.07.2020)
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An ensemble machine learning model generates a focused screening library for the identification of CDK8 inhibitors
Lin, Tony Eight, Yen, Dyan, HuangFu, Wei‐Chun, Wu, Yi‐Wen, Hsu, Jui‐Yi, Yen, Shih‐Chung, Sung, Tzu‐Ying, Hsieh, Jui‐Hua, Pan, Shiow‐Lin, Yang, Chia‐Ron, Huang, Wei‐Jan, Hsu, Kai‐Cheng
Published in Protein science (01.06.2024)
Published in Protein science (01.06.2024)
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Novel Class IIa-Selective Histone Deacetylase Inhibitors Discovered Using an in Silico Virtual Screening Approach
Hsu, Kai-Cheng, Liu, Chang-Yi, Lin, Tony Eight, Hsieh, Jui-Hua, Sung, Tzu-Ying, Tseng, Hui-Ju, Yang, Jinn-Moon, Huang, Wei-Jan
Published in Scientific reports (12.06.2017)
Published in Scientific reports (12.06.2017)
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HDAC8 Inhibition Specifically Targets Inv(16) Acute Myeloid Leukemic Stem Cells by Restoring p53 Acetylation
Qi, Jing, Singh, Sandeep, Hua, Wei-Kai, Cai, Qi, Chao, Shi-Wei, Li, Ling, Liu, Hongjun, Ho, Yinwei, McDonald, Tinisha, Lin, Allen, Marcucci, Guido, Bhatia, Ravi, Huang, Wei-Jan, Chang, Chung-I, Kuo, Ya-Huei
Published in Cell stem cell (05.11.2015)
Published in Cell stem cell (05.11.2015)
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Suberoylanilide Hydroxamic Acid, an Inhibitor of Histone Deacetylase, Enhances Radiosensitivity and Suppresses Lung Metastasis in Breast Cancer In Vitro and In Vivo
Chiu, Hui-Wen, Yeh, Ya-Ling, Wang, Yi-Ching, Huang, Wei-Jan, Chen, Yi-An, Chiou, Yi-Shiou, Ho, Sheng-Yow, Lin, Pinpin, Wang, Ying-Jan
Published in PloS one (10.10.2013)
Published in PloS one (10.10.2013)
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Pan-Inhibition of Protein Disulfide Isomerase Caused Cell Death through Disrupting Cellular Proteostasis in Pancreatic Ductal Adenocarcinoma Cells
Hung, Ching-Sheng, Lee, Kun-Lin, Huang, Wei-Jan, Su, Fang-He, Liang, Yu-Chih
Published in International journal of molecular sciences (01.11.2023)
Published in International journal of molecular sciences (01.11.2023)
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Synthesis and biological evaluation of ortho-phenyl phenylhydroxamic acids containing phenothiazine with improved selectivity for class IIa histone deacetylases
Hsu, Kai-Cheng, Huang, Yun-Yi, Chu, Jung-Chun, Huang, Yu-Wen, Hu, Jing-Lan, Lin, Tony Eight, Yen, Shih-Chung, Weng, Jing-Ru, Huang, Wei-Jan
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2024)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2024)
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The hydroxamate based HDAC inhibitor WMJ-J-09 induces colorectal cancer cell death by targeting tubulin and downregulating survivin
Huang, Yu-Han, Huang, Yu-Min, Huang, Wei-Jan, Yu, Meng-Chieh, Chuang, Chin-Hui, Hsu, Ya-Fen, Chen, Hsiu-Chen, Chen, Liang-Chieh, Huang, Shiu-Wen, Hsu, Ming-Jen
Published in Scientific reports (04.06.2025)
Published in Scientific reports (04.06.2025)
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Synthesis and biological evaluation of C-4 substituted phenoxazine-bearing hydroxamic acids with potent class II histone deacetylase inhibitory activities
Chu, Jung-Chun, Tseng, Hui-Ju, Lee, Sung-Bau, Hsu, Kai-Cheng, Hsin, Ling-Wei, Liang, Ru-Hao, Lin, Tony Eight, Gao, Nain-Chu, Chen, Liang-Chieh, Lu, Wan-Hsun, Wang, Andrew H.-J, Huang, Wei-Jan
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
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Acacetin Inhibits Glutamate Release and Prevents Kainic Acid-Induced Neurotoxicity in Rats
Lin, Tzu-Yu, Huang, Wei-Jan, Wu, Chia-Chan, Lu, Cheng-Wei, Wang, Su-Jane
Published in PloS one (10.02.2014)
Published in PloS one (10.02.2014)
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CircRNA hsa_circ_0004781 promoted cell proliferation by acting as a sponge for miR-9-5p and miR-338-3p and upregulating KLF5 and ADAM17 expression in pancreatic ductal adenocarcinoma
Lee, Kun-Lin, Liu, Jun-Jen, Huang, Wei-Jan, Hung, Ching-Sheng, Liang, Yu-Chih
Published in Cancer cell international (19.02.2025)
Published in Cancer cell international (19.02.2025)
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Exploring the Synergistic Effects of Erinacines on Microglial Regulation and Alzheimer's Pathology Under Metabolic Stress
Bui, Van Thanh, Wu, Kuan‐Wei, Chen, Chin‐Chu, Nguyen, Anh Thuc, Huang, Wei‐Jan, Lee, Li‐Ya, Chen, Wan‐Ping, Huang, Chi‐Ying, Shiao, Young‐Ji
Published in CNS neuroscience & therapeutics (01.12.2024)
Published in CNS neuroscience & therapeutics (01.12.2024)
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A novel histone deacetylase inhibitor TMU-35435 enhances etoposide cytotoxicity through the proteasomal degradation of DNA-PKcs in triple-negative breast cancer
Wu, Yuan-Hua, Hong, Chi-Wei, Wang, Yi-Ching, Huang, Wei-Jan, Yeh, Ya-Ling, Wang, Bour-Jr, Wang, Ying-Jan, Chiu, Hui-Wen
Published in Cancer letters (01.08.2017)
Published in Cancer letters (01.08.2017)
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HDAC8 Inhibitor WK2-16 Therapeutically Targets Lipopolysaccharide-Induced Mouse Model of Neuroinflammation and Microglial Activation
Lin, Fan-Li, Yen, Jing-Lun, Kuo, Yu-Cheng, Kang, Jaw-Jou, Cheng, Yu-Wen, Huang, Wei-Jan, Hsiao, George
Published in International journal of molecular sciences (18.01.2019)
Published in International journal of molecular sciences (18.01.2019)
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Cerebellar α6‐subunit‐containing GABAA receptors: a novel therapeutic target for disrupted prepulse inhibition in neuropsychiatric disorders
Chiou, Lih‐Chu, Lee, Hsin‐Jung, Ernst, Margot, Huang, Wei‐Jan, Chou, Jui‐Feng, Chen, Hon‐Lie, Mouri, Akihiro, Chen, Liang‐Chieh, Treven, Marco, Mamiya, Takayoshi, Fan, Pi‐Chuan, Knutson, Daniel E, Witzigmann, Chris, Cook, James, Sieghart, Werner, Nabeshima, Toshitaka
Published in British journal of pharmacology (01.06.2018)
Published in British journal of pharmacology (01.06.2018)
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A histone deacetylase inhibitor enhances expression of genes inhibiting Wnt pathway and augments activity of DNA demethylation reagent against nonsmall‐cell lung cancer
Shieh, Jiunn‐Min, Tang, Yen‐An, Hu, Fu‐Han, Huang, Wei‐Jan, Wang, Ying‐Jan, Jen, Jayu, Liao, Sheng‐You, Lu, Ying‐Hung, Yeh, Ya‐Ling, Wang, Tseng‐Wei, Lin, Pinpin, Wang, Yi‐Ching
Published in International journal of cancer (15.05.2017)
Published in International journal of cancer (15.05.2017)
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WMJ‐8‐B, a novel hydroxamate derivative, induces MDA‐MB‐231 breast cancer cell death via the SHP‐1‐STAT3‐survivin cascade
Chuang, Yu‐Fan, Huang, Shiu‐Wen, Hsu, Ya‐Fen, Yu, Meng‐Chieh, Ou, George, Huang, Wei‐Jan, Hsu, Ming‐Jen
Published in British journal of pharmacology (01.09.2017)
Published in British journal of pharmacology (01.09.2017)
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