Histone deacetylase inhibitors in clinical studies as templates for new anticancer agents
Mottamal, Madhusoodanan, Zheng, Shilong, Huang, Tien L, Wang, Guangdi
Published in Molecules (02.03.2015)
Published in Molecules (02.03.2015)
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Journal Article
Book Review
Alkanediamide-Linked Bisbenzamidines Are Promising Antiparasitic Agents
Vanden Eynde, Jean J, Mayence, Annie, Mottamal, Madhusoodanan, Bacchi, Cyrus J, Yarlett, Nigel, Kaiser, Marcel, Brun, Reto, Huang, Tien L
Published in Pharmaceuticals (Basel, Switzerland) (19.04.2016)
Published in Pharmaceuticals (Basel, Switzerland) (19.04.2016)
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Journal Article
In Vitro Selection and In Vivo Efficacy of Piperazine- and Alkanediamide-Linked Bisbenzamidines against Pneumocystis Pneumonia in Mice
Cushion, Melanie T, Walzer, Peter D, Ashbaugh, Alan, Rebholz, Sandra, Brubaker, Ronald, Vanden Eynde, Jean Jacques, Mayence, Annie, Huang, Tien L
Published in Antimicrobial Agents and Chemotherapy (01.07.2006)
Published in Antimicrobial Agents and Chemotherapy (01.07.2006)
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Journal Article
Bisbenzamidines as antifungal agents. are both amidine functions required to observe an anti-Pneumocystis carinii activity?
Laurent, Julien, Stanicki, Dimitri, Huang, Tien L, Dei-Cas, Eduardo, Pottier, Muriel, Aliouat, El Mouktar, Vanden Eynde, Jean Jacques
Published in Molecules (Basel, Switzerland) (11.06.2010)
Published in Molecules (Basel, Switzerland) (11.06.2010)
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Journal Article
Some non-conventional biomolecular targets for diamidines. A short survey
Huang, Tien L., Mayence, Annie, Vanden Eynde, Jean Jacques
Published in Bioorganic & medicinal chemistry (01.04.2014)
Published in Bioorganic & medicinal chemistry (01.04.2014)
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Journal Article
Small-molecule inhibitors of Wnt signaling pathway: towards novel anticancer therapeutics
Zheng, Shilong, Liu, Jiawang, Wu, Yanyuan, Huang, Tien L, Wang, Guangdi
Published in Future medicinal chemistry (01.12.2015)
Published in Future medicinal chemistry (01.12.2015)
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Journal Article
Potential of bisbenzimidazole‐analogs toward metronidazole‐resistant Trichomonas vaginalis isolates
Korosh, Travis, Bujans, Emmanuel, Morada, Mary, Karaalioglu, Canan, Vanden Eynde, Jean Jacques, Mayence, Annie, Huang, Tien L., Yarlett, Nigel
Published in Chemical biology & drug design (01.10.2017)
Published in Chemical biology & drug design (01.10.2017)
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Journal Article
Pentamidine analogs as inhibitors of [3H]MK-801 and [3H]ifenprodil binding to rat brain NMDA receptors
Berger, Michael L., Maciejewska, Dorota, Vanden Eynde, Jean Jacques, Mottamal, Madhusoodanan, Żabiński, Jerzy, Kaźmierczak, Paweł, Rezler, Mateusz, Jarak, Ivana, Piantanida, Ivo, Karminski-Zamola, Grace, Mayence, Annie, Rebernik, Patrick, Kumar, Arvind, Ismail, Mohamed A., Boykin, David W., Huang, Tien L.
Published in Bioorganic & medicinal chemistry (01.08.2015)
Published in Bioorganic & medicinal chemistry (01.08.2015)
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Journal Article
Fragment-Based Design of Symmetrical Bis-benzimidazoles as Selective Inhibitors of the Trimethoprim-Resistant, Type II R67 Dihydrofolate Reductase
Bastien, Dominic, Ebert, Maximilian C. C. J. C, Forge, Delphine, Toulouse, Jacynthe, Kadnikova, Natalia, Perron, Florent, Mayence, Annie, Huang, Tien L, Vanden Eynde, Jean Jacques, Pelletier, Joelle N
Published in Journal of medicinal chemistry (12.04.2012)
Published in Journal of medicinal chemistry (12.04.2012)
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Journal Article
Synthesis and SAR of alkanediamide-linked bisbenzamidines with anti-trypanosomal and anti-pneumocystis activity
Huang, Tien L., Eynde, Jean Jacques Vanden, Mayence, Annie, Collins, Margaret S., Cushion, Melanie T., Rattendi, Donna, Londono, Indira, Mazumder, Lakshman, Bacchi, Cyrus J., Yarlett, Nigel
Published in Bioorganic & medicinal chemistry letters (15.10.2009)
Published in Bioorganic & medicinal chemistry letters (15.10.2009)
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Journal Article
Trypanocidal Activity of Conformationally Restricted Pentamidine Congeners
Donkor, Isaac O, Huang, Tien L, Tao, Bin, Rattendi, Donna, Lane, Schennella, Vargas, Marc, Goldberg, Burt, Bacchi, Cyrus
Published in Journal of medicinal chemistry (13.03.2003)
Published in Journal of medicinal chemistry (13.03.2003)
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Journal Article
Trypanocidal activity of piperazine-linked bisbenzamidines and bisbenzamidoxime, an orally active prodrug
Huang, Tien L, Bacchi, Cyrus J, Kode, Nageswara R, Zhang, Qiang, Wang, Guangdi, Yartlet, Nigel, Rattendi, Donna, Londono, Indira, Mazumder, Lakshman, Vanden Eynde, Jean Jacques, Mayence, Annie, Donkor, Isaac O
Published in International journal of antimicrobial agents (01.12.2007)
Published in International journal of antimicrobial agents (01.12.2007)
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Journal Article
Parallel Solution-Phase Synthesis of Conformationally Restricted Congeners of Pentamidine and Evaluation of Their Antiplasmodial Activities
Mayence, Annie, Vanden Eynde, Jean Jacques, Krogstad, Fran M, Krogstad, Donald J, Cushion, Melanie T, Huang, Tien L
Published in Journal of medicinal chemistry (06.05.2004)
Published in Journal of medicinal chemistry (06.05.2004)
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Journal Article
Anti-plasmodial and anti-leishmanial activity of conformationally restricted pentamidine congeners
Huang, Tien L, Vanden Eynde, Jean Jacques, Mayence, Annie, Donkor, Isaac O, Khan, Shabana I, Tekwani, Babu L
Published in Journal of pharmacy and pharmacology (01.08.2006)
Published in Journal of pharmacy and pharmacology (01.08.2006)
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Journal Article
Peptidyl aldehyde inhibitors of calpain incorporating P2-Proline mimetics
DONKOR, Isaac O, KORUKONDA, Rajani, HUANG, Tien L, LECOUR, Louis JR
Published in Bioorganic & medicinal chemistry letters (10.03.2003)
Published in Bioorganic & medicinal chemistry letters (10.03.2003)
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