BMI1–RING1B is an autoinhibited RING E3 ubiquitin ligase
Taherbhoy, Asad M., Huang, Oscar W., Cochran, Andrea G.
Published in Nature communications (07.07.2015)
Published in Nature communications (07.07.2015)
Get full text
Journal Article
Wnt Antagonists Bind through a Short Peptide to the First β-Propeller Domain of LRP5/6
Bourhis, Eric, Wang, Weiru, Tam, Christine, Hwang, Jiyoung, Zhang, Yingnan, Spittler, Didier, Huang, Oscar W., Gong, Yan, Estevez, Alberto, Zilberleyb, Inna, Rouge, Lionel, Chiu, Cecilia, Wu, Yan, Costa, Mike, Hannoush, Rami N., Franke, Yvonne, Cochran, Andrea G.
Published in Structure (London) (12.10.2011)
Published in Structure (London) (12.10.2011)
Get full text
Journal Article
Preparation of Distinct Ubiquitin Chain Reagents of High Purity and Yield
Dong, Ken C., Helgason, Elizabeth, Yu, Christine, Phu, Lilian, Arnott, David P., Bosanac, Ivan, Compaan, Deanne M., Huang, Oscar W., Fedorova, Anna V., Kirkpatrick, Donald S., Hymowitz, Sarah G., Dueber, Erin C.
Published in Structure (London) (10.08.2011)
Published in Structure (London) (10.08.2011)
Get full text
Journal Article
Exploiting the Cullin E3 Ligase Adaptor Protein SKP1 for Targeted Protein Degradation
Hong, Seong Ho, Divakaran, Anand, Osa, Akane, Huang, Oscar W., Wertz, Ingrid E., Nomura, Daniel K.
Published in ACS chemical biology (16.02.2024)
Published in ACS chemical biology (16.02.2024)
Get full text
Journal Article
Covalent Degrader of the Oncogenic Transcription Factor β‑Catenin
Gowans, Flor A., Forte, Nafsika, Hatcher, Justin, Huang, Oscar W., Wang, Yangzhi, Altamirano Poblano, Belen E., Wertz, Ingrid E., Nomura, Daniel K.
Published in Journal of the American Chemical Society (06.06.2024)
Published in Journal of the American Chemical Society (06.06.2024)
Get full text
Journal Article
Deubiquitinase DUBA is a post-translational brake on interleukin-17 production in T cells
Rutz, Sascha, Kayagaki, Nobuhiko, Phung, Qui T., Eidenschenk, Celine, Noubade, Rajkumar, Wang, Xiaoting, Lesch, Justin, Lu, Rongze, Newton, Kim, Huang, Oscar W., Cochran, Andrea G., Vasser, Mark, Fauber, Benjamin P., DeVoss, Jason, Webster, Joshua, Diehl, Lauri, Modrusan, Zora, Kirkpatrick, Donald S., Lill, Jennie R., Ouyang, Wenjun, Dixit, Vishva M.
Published in Nature (London) (19.02.2015)
Published in Nature (London) (19.02.2015)
Get full text
Journal Article
Phosphorylation-dependent activity of the deubiquitinase DUBA
Huang, Oscar W, Ma, Xiaolei, Yin, JianPing, Flinders, Jeremy, Maurer, Till, Kayagaki, Nobuhiko, Phung, Qui, Bosanac, Ivan, Arnott, David, Dixit, Vishva M, Hymowitz, Sarah G, Starovasnik, Melissa A, Cochran, Andrea G
Published in Nature structural & molecular biology (01.02.2012)
Published in Nature structural & molecular biology (01.02.2012)
Get full text
Journal Article
A Class of 2,4-Bisanilinopyrimidine Aurora A Inhibitors with Unusually High Selectivity against Aurora B
Aliagas-Martin, Ignacio, Burdick, Dan, Corson, Laura, Dotson, Jennafer, Drummond, Jason, Fields, Carter, Huang, Oscar W, Hunsaker, Thomas, Kleinheinz, Tracy, Krueger, Elaine, Liang, Jun, Moffat, John, Phillips, Gail, Pulk, Rebecca, Rawson, Thomas E, Ultsch, Mark, Walker, Leslie, Wiesmann, Christian, Zhang, Birong, Zhu, Bing-Yan, Cochran, Andrea G
Published in Journal of medicinal chemistry (28.05.2009)
Published in Journal of medicinal chemistry (28.05.2009)
Get full text
Journal Article
Fragment-Based Discovery of a Selective and Cell-Active Benzodiazepinone CBP/EP300 Bromodomain Inhibitor (CPI-637)
Taylor, Alexander M, Côté, Alexandre, Hewitt, Michael C, Pastor, Richard, Leblanc, Yves, Nasveschuk, Christopher G, Romero, F. Anthony, Crawford, Terry D, Cantone, Nico, Jayaram, Hariharan, Setser, Jeremy, Murray, Jeremy, Beresini, Maureen H, de Leon Boenig, Gladys, Chen, Zhongguo, Conery, Andrew R, Cummings, Richard T, Dakin, Leslie A, Flynn, E. Megan, Huang, Oscar W, Kaufman, Susan, Keller, Patricia J, Kiefer, James R, Lai, Tommy, Li, Yingjie, Liao, Jiangpeng, Liu, Wenfeng, Lu, Henry, Pardo, Eneida, Tsui, Vickie, Wang, Jian, Wang, Yongyun, Xu, Zhaowu, Yan, Fen, Yu, Dong, Zawadzke, Laura, Zhu, Xiaoqin, Zhu, Xiaoyu, Sims, Robert J, Cochran, Andrea G, Bellon, Steve, Audia, James E, Magnuson, Steven, Albrecht, Brian K
Published in ACS medicinal chemistry letters (12.05.2016)
Published in ACS medicinal chemistry letters (12.05.2016)
Get full text
Journal Article
Phosphorylation-dependent activity of the deubiquitinase DUBA
Huang, Oscar W., Ma, Xiaolei, Yin, JianPing, Flinders, Jeremy, Maurer, Till, Kayagaki, Nobuhiko, Phung, Qui, Bosanac, Ivan, Arnott, David, Dixit, Vishva M., Hymowitz, Sarah G., Starovasnik, Melissa A., Cochran, Andrea G.
Published in Nature structural & molecular biology (15.01.2012)
Published in Nature structural & molecular biology (15.01.2012)
Get full text
Journal Article
Wnt Antagonists Bind through a Short Peptide to the First [beta]-Propeller Domain of LRP5/6
Bourhis, Eric, Wang, Weiru, Tam, Christine, Hwang, Jiyoung, Zhang, Yingnan, Spittler, Didier, Huang, Oscar W, Gong, Yan, Estevez, Alberto, Zilberleyb, Inna, Rouge, Lionel, Chiu, Cecilia, Wu, Yan, Costa, Mike, Hannoush, Rami N, Franke, Yvonne, Cochran, Andrea G
Published in Structure (London) (12.10.2011)
Published in Structure (London) (12.10.2011)
Get full text
Journal Article
Exploiting the Cullin E3 Ligase Adaptor Protein SKP1 for Targeted Protein Degradation
Hong, Seong Ho, Osa, Akane, Huang, Oscar W, Wertz, Ingrid E, Nomura, Daniel K
Published in bioRxiv (02.11.2023)
Published in bioRxiv (02.11.2023)
Get full text
Journal Article
Covalent Degrader of the Oncogenic Transcription Factor β-Catenin
Gowans, Flor A, Forte, Nafsika, Hatcher, Justin, Huang, Oscar W, Wang, Yangzhi, Poblano, Belen E Altamirano, Wertz, Ingrid E, Nomura, Daniel K
Published in bioRxiv : the preprint server for biology (02.11.2023)
Get more information
Published in bioRxiv : the preprint server for biology (02.11.2023)
Journal Article