Stereochemical Requirements for the Mineralocorticoid Receptor Antagonist Activity of Dihydropyridines
Arhancet, Graciela B, Woodard, Scott S, Dietz, Jessica D, Garland, Danny J, Wagner, Grace M, Iyanar, Kaliappan, Collins, Joe T, Blinn, James R, Numann, Randal E, Hu, Xiao, Huang, Horng-Chih
Published in Journal of medicinal chemistry (27.05.2010)
Published in Journal of medicinal chemistry (27.05.2010)
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Structural and Thermodynamic Characterization of the TYK2 and JAK3 Kinase Domains in Complex with CP-690550 and CMP-6
Chrencik, Jill E., Patny, Akshay, Leung, Iris K., Korniski, Brian, Emmons, Thomas L., Hall, Troii, Weinberg, Robin A., Gormley, Jennifer A., Williams, Jennifer M., Day, Jacqueline E., Hirsch, Jeffrey L., Kiefer, James R., Leone, Joseph W., Fischer, H. David, Sommers, Cynthia D., Huang, Horng-Chih, Jacobsen, E.J., Tenbrink, Ruth E., Tomasselli, Alfredo G., Benson, Timothy E.
Published in Journal of molecular biology (16.07.2010)
Published in Journal of molecular biology (16.07.2010)
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Discovery of (3 S ,3a R )-2-(3-Chloro-4-cyanophenyl)-3-cyclopentyl-3,3a,4,5-tetrahydro-2 H -benzo[ g ]indazole-7-carboxylic Acid (PF-3882845), an Orally Efficacious Mineralocorticoid Receptor (MR) Antagonist for Hypertension and Nephropathy
Meyers, Marvin J., Arhancet, Graciela B., Hockerman, Susan L., Chen, Xiangyang, Long, Scott A., Mahoney, Matthew W., Rico, Joseph R., Garland, Danny J., Blinn, James. R., Collins, Joe T., Yang, Shengtian, Huang, Horng-Chih, McGee, Kevin F., Wendling, Jay M., Dietz, Jessica D., Payne, Maria A., Homer, Bruce L., Heron, Marcia I., Reitz, David B., Hu, Xiao
Published in Journal of medicinal chemistry (26.08.2010)
Published in Journal of medicinal chemistry (26.08.2010)
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Discovery of (3S,3aR)-2-(3-Chloro-4-cyanophenyl)-3-cyclopentyl-3,3a,4,5-tetrahydro-2H-benzo[g]indazole-7-carboxylic Acid (PF-3882845), an Orally Efficacious Mineralocorticoid Receptor (MR) Antagonist for Hypertension and Nephropathy
Meyers, Marvin J, Arhancet, Graciela B, Hockerman, Susan L, Chen, Xiangyang, Long, Scott A, Mahoney, Matthew W, Rico, Joseph R, Garland, Danny J, Blinn, James. R, Collins, Joe T, Yang, Shengtian, Huang, Horng-Chih, McGee, Kevin F, Wendling, Jay M, Dietz, Jessica D, Payne, Maria A, Homer, Bruce L, Heron, Marcia I, Reitz, David B, Hu, Xiao
Published in Journal of medicinal chemistry (26.08.2010)
Published in Journal of medicinal chemistry (26.08.2010)
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A Highly Enantioselective Benzothiepine Synthesis
Wang, Ching-Cheng, Li, James J, Huang, Horng-Chih, Lee, Len F, Reitz, David B
Published in Journal of organic chemistry (05.05.2000)
Published in Journal of organic chemistry (05.05.2000)
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Discovery of Novel Cyanodihydropyridines as Potent Mineralocorticoid Receptor Antagonists
Arhancet, Graciela B, Woodard, Scott S, Iyanar, Kaliappan, Case, Brenda L, Woerndle, Rhonda, Dietz, Jessica D, Garland, Danny J, Collins, Joe T, Payne, Maria A, Blinn, James R, Pomposiello, Silvia I, Hu, Xiao, Heron, Marcia I, Huang, Horng-Chih, Lee, Len F
Published in Journal of medicinal chemistry (26.08.2010)
Published in Journal of medicinal chemistry (26.08.2010)
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Novel Tight-Binding Inhibitory Factor-κB Kinase (IKK-2) Inhibitors Demonstrate Target-Specific Anti-Inflammatory Activities in Cellular Assays and following Oral and Local Delivery in an in Vivo Model of Airway Inflammation
Sommers, Cynthia D., Thompson, Janice M., Guzova, Julia A., Bonar, Sheri L., Rader, Randall K., Mathialagan, Sumathy, Venkatraman, Neetu, Holway, Vicky Walker, Kahn, Larry E., Hu, George, Garner, Debra S., Huang, Horng-Chih, Chiang, Po-Chang, Schindler, John F., Hu, Yiding, Meyer, Debra M., Kishore, Nandini N.
Published in The Journal of pharmacology and experimental therapeutics (01.08.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2009)
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1,2-Diarylcyclopentenes as Selective Cyclooxygenase-2 Inhibitors and Orally Active Anti-inflammatory Agents
Li, James J, Anderson, Gary D, Burton, Earl G, Cogburn, J. Nita, Collins, Joe T, Garland, Danny J, Gregory, Susan A, Huang, Horng-Chih, Isakson, Peter C
Published in Journal of medicinal chemistry (01.10.1995)
Published in Journal of medicinal chemistry (01.10.1995)
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Aminopyridinecarboxamide-based inhaled IKK-2 inhibitors for asthma and COPD: Structure–activity relationship
Xie, Jin, Poda, Gennadiy I., Hu, Yiding, Chen, Natalie X., Heier, Richard F., Wolfson, Serge G., Reding, Matthew T., Lennon, Patrick J., Kurumbail, Ravi G., Selness, Shaun R., Li, Xiong, Kishore, Nandini N., Sommers, Cynthia D., Christine, Lori, Bonar, Sheri L., Venkatraman, Neetu, Mathialagan, Sumathy, Brustkern, Sarah J., Huang, Horng-Chih
Published in Bioorganic & medicinal chemistry (01.02.2011)
Published in Bioorganic & medicinal chemistry (01.02.2011)
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Discovery of Potent, Nonsystemic Apical Sodium-Codependent Bile Acid Transporter Inhibitors (Part 1)
Tremont, Samuel J, Lee, Len F, Huang, Horng-Chih, Keller, Bradley T, Banerjee, Shyamal C, Both, Scott R, Carpenter, Andrew J, Wang, Ching-Cheng, Garland, Danny J, Huang, Wei, Jones, Claude, Koeller, Kevin J, Kolodziej, Steve A, Li, James, Manning, Robert E, Mahoney, Matthew W, Miller, Raymond E, Mischke, Deborah A, Rath, Nigam P, Fletcher, Theresa, Reinhard, Emily J, Tollefson, Michael B, Vernier, William F, Wagner, Grace M, Rapp, Steve R, Beaudry, Judy, Glenn, Kevin, Regina, Karen, Schuh, Joe R, Smith, Mark E, Trivedi, Jay S, Reitz, David B
Published in Journal of medicinal chemistry (08.09.2005)
Published in Journal of medicinal chemistry (08.09.2005)
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Design, synthesis, and biological evaluation of pyrazinones containing novel P1 needles as inhibitors of TF/VIIa
Trujillo, John I., Huang, Horng-Chih, Neumann, William L., Mahoney, Matthew W., Long, Scott, Huang, Wei, Garland, Danny J., Kusturin, Carrie, Abbas, Zaheer, South, Michael S., Reitz, David B.
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
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Discovery of Potent, Nonsystemic Apical Sodium-Codependent Bile Acid Transporter Inhibitors (Part 2)
Huang, Horng-Chih, Tremont, Samuel J, Lee, Len F, Keller, Bradley T, Carpenter, Andrew J, Wang, Ching-Cheng, Banerjee, Shyamal C, Both, Scott R, Fletcher, Theresa, Garland, Danny J, Huang, Wei, Jones, Claude, Koeller, Kevin J, Kolodziej, Steve A, Li, James, Manning, Robert E, Mahoney, Matthew W, Miller, Raymond E, Mischke, Deborah A, Rath, Nigam P, Reinhard, Emily J, Tollefson, Michael B, Vernier, William F, Wagner, Grace M, Rapp, Steve R, Beaudry, Judy, Glenn, Kevin, Regina, Karen, Schuh, Joe R, Smith, Mark E, Trivedi, Jay S, Reitz, David B
Published in Journal of medicinal chemistry (08.09.2005)
Published in Journal of medicinal chemistry (08.09.2005)
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A novel one-pot conversion of methyl sulfones to sulfonamides
Huang, Horng-Chih, Reinhard, Emily J., Reitz, David B.
Published in Tetrahedron letters (26.09.1994)
Published in Tetrahedron letters (26.09.1994)
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Aminopyridinecarboxamide-based inhibitors: Structure–activity relationship
Bonafoux, Dominique F., Bonar, Sheri L., Clare, Michael, Donnelly, Ann M., Glaenzer, Jeanette L., Guzova, Julia A., Huang, He, Kishore, Nandidni N., Koszyk, Francis J., Lennon, Patrick J., Libby, Adam, Mathialagan, Sumathy, Oburn, David S., Rouw, Sharon A, Sommers, Cynthia D., Tripp, Catherine S., Vanella, Lori J., Weier, Richard, Wolfson, Serge G., Huang, Horng-Chih
Published in Bioorganic & medicinal chemistry (2010)
Published in Bioorganic & medicinal chemistry (2010)
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Kinetic characterization of human glutamine-fructose-6-phosphate amidotransferase I: potent feedback inhibition by glucosamine 6-phosphate
Broschat, Kay O, Gorka, Christine, Page, Jimmy D, Martin-Berger, Cynthia L, Davies, Michael S, Huang Hc, Horng-chih, Gulve, Eric A, Salsgiver, William J, Kasten, Thomas P
Published in The Journal of biological chemistry (26.04.2002)
Published in The Journal of biological chemistry (26.04.2002)
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In vivo pharmacology of SC-51316, a nonpeptidic angiotensin II receptor antagonist
Olins, G M, Smits, G J, Koepke, J P, Huang, H C, Reitz, D B, Manning, R E, Blaine, E H
Published in American journal of hypertension (01.07.1993)
Published in American journal of hypertension (01.07.1993)
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Diaryl indenes and benzofurans: Novel classes of potent and selective cyclooxygenase-2 inhibitors
Huang, Horng-Chih, Chamberlain, Timothy S., Selbert, Karen, Koboldt, Carol M., Isakson, Peter C., Reitz, David B.
Published in Bioorganic & medicinal chemistry letters (19.10.1995)
Published in Bioorganic & medicinal chemistry letters (19.10.1995)
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