Structure-Based Design of Potent Peptidomimetic Inhibitors Covalently Targeting SARS-CoV-2 Papain-like Protease
Wang, Qian, Chen, Guofeng, He, Jian, Li, Jiameng, Xiong, Muya, Su, Haixia, Li, Minjun, Hu, Hangchen, Xu, Yechun
Published in International journal of molecular sciences (11.05.2023)
Published in International journal of molecular sciences (11.05.2023)
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Journal Article
Identification of Cysteine 270 as a Novel Site for Allosteric Modulators of SARS‐CoV‐2 Papain‐Like Protease
Hu, Hangchen, Wang, Qian, Su, Haixia, Shao, Qiang, Zhao, Wenfeng, Chen, Guofeng, Li, Minjun, Xu, Yechun
Published in Angewandte Chemie International Edition (23.12.2022)
Published in Angewandte Chemie International Edition (23.12.2022)
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Journal Article
Unraveling the catalytic mechanism of SARS-CoV-2 papain-like protease with allosteric modulation of C270 mutation using multiscale computational approaches
Shao, Qiang, Xiong, Muya, Li, Jiameng, Hu, Hangchen, Su, Haixia, Xu, Yechun
Published in Chemical science (Cambridge) (10.05.2023)
Published in Chemical science (Cambridge) (10.05.2023)
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Journal Article
Chemical Space Profiling of SARS-CoV‑2 PLpro Using DNA-Encoded Focused Libraries
Wang, Xudong, Zhu, Ying, Zhao, Qingyi, Lu, Weiwei, Xu, Yechun, Hu, Hangchen, Lu, Xiaojie
Published in ACS medicinal chemistry letters (11.04.2024)
Published in ACS medicinal chemistry letters (11.04.2024)
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Journal Article
Chemical Space Profiling of SARS-CoV-2 PL pro Using DNA-Encoded Focused Libraries
Wang, Xudong, Zhu, Ying, Zhao, Qingyi, Lu, Weiwei, Xu, Yechun, Hu, Hangchen, Lu, Xiaojie
Published in ACS medicinal chemistry letters (11.04.2024)
Published in ACS medicinal chemistry letters (11.04.2024)
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Journal Article
Structure-based design of a novel inhibitor of the ZIKA virus NS2B/NS3 protease
Xiong, Yanchao, Cheng, Fei, Zhang, Junyi, Su, Haixia, Hu, Hangchen, Zou, Yi, Li, Minjun, Xu, Yechun
Published in Bioorganic chemistry (01.11.2022)
Published in Bioorganic chemistry (01.11.2022)
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Journal Article
Discovery, SAR Study of GST Inhibitors from a Novel Quinazolin-4(1H)‑one Focused DNA-Encoded Library
Wen, Xin, Zhang, Minmin, Duan, Zhiqiang, Suo, Yanrui, Lu, Weiwei, Jin, Rui, Mu, Baiyang, Li, Kaige, Zhang, Xu, Meng, Linghua, Hong, Yu, Wang, Xingyu, Hu, Hangchen, Zhu, Jian, Song, Weixiao, Shen, Aijun, Lu, Xiaojie
Published in Journal of medicinal chemistry (24.08.2023)
Published in Journal of medicinal chemistry (24.08.2023)
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Journal Article
Structure-Based Survey of the Binding Modes of BACE1 Inhibitors
Hu, Hangchen, Chen, Zhaoqiang, Xu, Xiang, Xu, Yechun
Published in ACS chemical neuroscience (20.02.2019)
Published in ACS chemical neuroscience (20.02.2019)
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Journal Article
Identification of Highly Selective Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Inhibitors by a Covalent Fragment-Based Approach
Huang, Fubao, Hu, Hangchen, Wang, Kai, Peng, Chengyuan, Xu, Wenwei, Zhang, Yu, Gao, Jing, Liu, Yishen, Zhou, Hu, Huang, Ruimin, Li, Minjun, Shen, Jianhua, Xu, Yechun
Published in Journal of medicinal chemistry (09.07.2020)
Published in Journal of medicinal chemistry (09.07.2020)
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Journal Article
Identification of Cysteine 270 as a Novel Site for Allosteric Modulators of SARS‐CoV‐2 Papain‐Like Protease
Hu, Hangchen, Wang, Qian, Su, Haixia, Shao, Qiang, Zhao, Wenfeng, Chen, Guofeng, Li, Minjun, Xu, Yechun
Published in Angewandte Chemie (23.12.2022)
Published in Angewandte Chemie (23.12.2022)
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Journal Article
Tricyclic compound as well as preparation method and application thereof
REN PENGXUAN, ZHANG XIANGLEI, LIU HONG, SU HAIXIA, YU CHANGYUE, LI JIAN, BAI FANG, HU HANGCHEN, ZHANG LEIRA, XU YECHUN
Year of Publication 03.01.2023
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Year of Publication 03.01.2023
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