Discovery of a new chemical series of BRD4(1) inhibitors using protein-ligand docking and structure-guided design
Duffy, Bryan C., Liu, Shuang, Martin, Gregory S., Wang, Ruifang, Hsia, Ming Min, Zhao, He, Guo, Cheng, Ellis, Michael, Quinn, John F., Kharenko, Olesya A., Norek, Karen, Gesner, Emily M., Young, Peter R., McLure, Kevin G., Wagner, Gregory S., Lakshminarasimhan, Damodharan, White, Andre, Suto, Robert K., Hansen, Henrik C., Kitchen, Douglas B.
Published in Bioorganic & medicinal chemistry letters (15.07.2015)
Published in Bioorganic & medicinal chemistry letters (15.07.2015)
Get full text
Journal Article
An efficient synthesis of (7S,10R)-2-bromo-5,6,7,8,9,10-hexahydro-7,10-epiminocyclohepta[b]indole: application in the preparation and structural confirmation of a potent 5-HT6 antagonist
Isherwood, Matthew L., Guzzo, Peter R., Henderson, Alan J., Hsia, Ming Min, Kaur, Jagjit, Nacro, Kassoum, Narreddula, Venkateswara R., Panduga, Shailaja, Pathak, Rashmi, Shimpukade, Bharat, Tan, Valentina, Xiang, Kai, Qiang, Zhu, Ghosh, Animesh
Published in Tetrahedron: asymmetry (15.12.2012)
Published in Tetrahedron: asymmetry (15.12.2012)
Get full text
Journal Article
BRIDGED AND FUSED HETEROCYCLIC ANTIDIABETIC COMPOUNDS
CLADER, JOHN, W, DAVIS, JASON, L, DENG, KAI, HSIA, MING MIN, JOSIEN, HUBERT, B, HERR, ROBERT, JASON, GREENLEE, WILLIAM, J, WAN, SHUANGYI, MAYER, MICHAEL, JOHN
Year of Publication 20.11.2013
Get full text
Year of Publication 20.11.2013
Patent
PENTAFLUOROSULPHOLANE-CONTAINING ANTIDIABETIC COMPOUNDS
GREENLEE WILLIAM J, JOSIEN HUBERT B, MAYER MICHAEL JOHN, DAVIS JASON L, CLADER JOHN W, HSIA MING MIN, STAMFORD ANDREW, WAN SHUANGYI
Year of Publication 22.12.2011
Get full text
Year of Publication 22.12.2011
Patent
BRIDGED AND FUSED HETEROCYCLIC ANTIDIABETIC COMPOUNDS
HERR ROBERT JASON, GREENLEE WILLIAM J, JOSIEN HUBERT B, MAYER MICHAEL JOHN, DAVIS JASON L, CLADER JOHN W, HSIA MING MIN, DENG KAI, WAN SHUANGYI
Year of Publication 22.12.2011
Get full text
Year of Publication 22.12.2011
Patent
PENTAFLUOROSULPHOLANE-CONTAINING ANTIDIABETIC COMPOUNDS
CLADER, JOHN, W, DAVIS, JASON, L, HSIA, MING MIN, JOSIEN, HUBERT, B, GREENLEE, WILLIAM, J, STAMFORD, ANDREW, WAN, SHUANGYI, MAYER, MICHAEL, JOHN
Year of Publication 30.11.2011
Get full text
Year of Publication 30.11.2011
Patent
BRIDGED AND FUSED HETEROCYCLIC ANTIDIABETIC COMPOUNDS
CLADER, JOHN, W, DAVIS, JASON, L, DENG, KAI, HSIA, MING MIN, JOSIEN, HUBERT, B, HERR, ROBERT, JASON, GREENLEE, WILLIAM, J, WAN, SHUANGYI, MAYER, MICHAEL, JOHN
Year of Publication 30.11.2011
Get full text
Year of Publication 30.11.2011
Patent
Bridged and fused heterocyclic antidiabetic compounds
DENG, KAI, GREENLEE, WILLIAM J, MAYER, MICHAEL JOHN, HSIA, MING MIN, HERR, ROBERT JASON, WAN, SHUANGYI, JOSIEN, HUBERT B, CLADER, JOHN W, DAVIS, JASON L
Year of Publication 28.07.2011
Get full text
Year of Publication 28.07.2011
Patent
Pentafluorosulpholane-containing antidiabetic compounds
GREENLEE, WILLIAM J, MAYER, MICHAEL JOHN, HSIA, MING MIN, STAMFORD, ANDREW, WAN, SHUANGYI, JOSIEN, HUBERT B, CLADER, JOHN W, DAVIS, JASON L
Year of Publication 28.07.2011
Get full text
Year of Publication 28.07.2011
Patent
PENTAFLUOROSULPHOLANE-CONTAINING ANTIDIABETIC COMPOUNDS
CLADER, JOHN, W, DAVIS, JASON, L, HSIA, MING MIN, JOSIEN, HUBERT, B, GREENLEE, WILLIAM, J, STAMFORD, ANDREW, WAN, SHUANGYI, MAYER, MICHAEL, JOHN
Year of Publication 29.07.2010
Get full text
Year of Publication 29.07.2010
Patent
BRIDGED AND FUSED HETEROCYCLIC ANTIDIABETIC COMPOUNDS
CLADER, JOHN, W, DAVIS, JASON, L, DENG, KAI, HSIA, MING MIN, JOSIEN, HUBERT, B, HERR, ROBERT, JASON, GREENLEE, WILLIAM, J, WAN, SHUANGYI, MAYER, MICHAEL, JOHN
Year of Publication 29.07.2010
Get full text
Year of Publication 29.07.2010
Patent
PENTAFLUOROSULPHOLANE-CONTAINING ANTIDIABETIC COMPOUNDS
GREENLEE, WILLIAM J, MAYER, MICHAEL JOHN, HSIA, MING MIN, STAMFORD, ANDREW, WAN, SHUANGYI, JOSIEN, HUBERT B, CLADER, JOHN W, DAVIS, JASON L
Year of Publication 29.07.2010
Get full text
Year of Publication 29.07.2010
Patent
BRIDGED AND FUSED HETEROCYCLIC ANTIDIABETIC COMPOUNDS
DENG, KAI, GREENLEE, WILLIAM J, MAYER, MICHAEL JOHN, HSIA, MING MIN, HERR, ROBERT JASON, WAN, SHUANGYI, JOSIEN, HUBERT B, CLADER, JOHN W, DAVIS, JASON L
Year of Publication 29.07.2010
Get full text
Year of Publication 29.07.2010
Patent
Pentafluorosulpholane-containing antidiabetic compounds
GREENLEE, WILLIAM J, MAYER, MICHAEL JOHN, HSIA, MING MIN, WAN, SHUANG-YI, STAMFORD, ANDREW, JOSIEN, HUBERT B, CLADER, JOHN W, DAVIS, JASON L
Year of Publication 16.11.2010
Get full text
Year of Publication 16.11.2010
Patent
Bridged and fused heterocyclic antidiabetic compounds
DENG, KAI, GREENLEE, WILLIAM J, MAYER, MICHAEL JOHN, HSIA, MING MIN, WAN, SHUANG-YI, HERR, ROBERT JASON, JOSIEN, HUBERT B, CLADER, JOHN W, DAVIS, JASON L
Year of Publication 16.11.2010
Get full text
Year of Publication 16.11.2010
Patent