Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii : From Screening Impurity to In Vivo Efficacy
Skudlarek, Jason W., Cooke, Andrew J., Mitchell, Helen J., Babaoglu, Kerim, Shaw, Anthony W., Tong, Ling, Nomland, Ashley B., Labroli, Marc, Sha, Deyou, Mulhearn, James J., Wu, Chengwei, Li, Sarah W., Beshore, Douglas C., Hughes, Jonathan M. E., Jouffroy, Matthieu, Wang, Hao, Balibar, Carl J., Painter, Ronald E., Shen, Pamela, Lange, Henry S., Ishchenko, Andrii, Chen, Yun-Ting, Klein, Daniel J., Tracy, Rodger W., Miller, Randy R., Cabalu, Tamara D., Wu, Zhe, Leithead, Andrew, Scapin, Giovanna, Hruza, Alan W., Dzhekieva, Liudmila, Bukhtiyarova, Marina, Homsher, Michelle F., Xu, Min, Bahnck-Teets, Carolyn, McKenney, David, Buevich, Alexei V., Liu, Jian, Zhang, Li-Kang, Meng, Tao, Kelly, Terri, DiNunzio, Edward, Soisson, Stephen, Cheng, Robert K. Y., Hennig, Michael, Raheem, Izzat, Walker, Scott S.
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Published in Journal of medicinal chemistry (12.09.2024)
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Deng, Yongqi, Shipps, Gerald W, Cooper, Alan, English, Jessie M, Annis, D. Allen, Carr, Donna, Nan, Yang, Wang, Tong, Zhu, Hugh Y, Chuang, Cheng-Chi, Dayananth, Priya, Hruza, Alan W, Xiao, Li, Jin, Weihong, Kirschmeier, Paul, Windsor, William T, Samatar, Ahmed A
Published in Journal of medicinal chemistry (13.11.2014)
Published in Journal of medicinal chemistry (13.11.2014)
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MK-8353: Discovery of an Orally Bioavailable Dual Mechanism ERK Inhibitor for Oncology
Boga, Sobhana Babu, Deng, Yongqi, Zhu, Liang, Nan, Yang, Cooper, Alan B., Shipps, Gerald W., Doll, Ronald, Shih, Neng-Yang, Zhu, Hugh, Sun, Robert, Wang, Tong, Paliwal, Sunil, Tsui, Hon-Chung, Gao, Xiaolei, Yao, Xin, Desai, Jagdish, Wang, James, Alhassan, Abdul Basit, Kelly, Joseph, Patel, Mehul, Muppalla, Kiran, Gudipati, Subrahmanyam, Zhang, Li-Kang, Buevich, Alexei, Hesk, David, Carr, Donna, Dayananth, Priya, Black, Stuart, Mei, Hong, Cox, Kathleen, Sherborne, Bradley, Hruza, Alan W., Xiao, Li, Jin, Weihong, Long, Brian, Liu, Gongjie, Taylor, Stacey A., Kirschmeier, Paul, Windsor, William T., Bishop, Robert, Samatar, Ahmed A.
Published in ACS medicinal chemistry letters (12.07.2018)
Published in ACS medicinal chemistry letters (12.07.2018)
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Bukhtiyarova, Marina, Cook, Erica M., Hancock, Paula J., Hruza, Alan W., Shaw, Anthony W., Adam, Gregory C., Barnard, Richard J. O., McKenna, Philip M., Holloway, M. Katharine, Bell, Ian M., Carroll, Steve, Cornella-Taracido, Ivan, Cox, Christopher D., Kutchukian, Peter S., Powell, David A., Strickland, Corey, Trotter, B. Wesley, Tudor, Matthew, Wolkenberg, Scott, Li, Jing, Tellers, David M.
Published in ACS medicinal chemistry letters (14.01.2021)
Published in ACS medicinal chemistry letters (14.01.2021)
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Modulating the interaction between CDK2 and cyclin A with a quinoline-based inhibitor
Deng, Yongqi, Shipps, Gerald W., Zhao, Lianyun, Siddiqui, M. Arshad, Popovici-Muller, Janeta, Curran, Patrick J., Duca, Jose S., Hruza, Alan W., Fischmann, Thierry O., Madison, Vincent S., Zhang, Rumin, McNemar, Charles W., Mayhood, Todd W., Syto, Rosalinda, Annis, Allen, Kirschmeier, Paul, Lees, Emma M., Parry, David A., Windsor, William T.
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
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Synthesis, Properties, and Applications of Diazotrifluropropanoyl-Containing Photoactive Analogs of Farnesyl Diphosphate Containing Modified Linkages for Enhanced Stability
Hovlid, Marisa L, Edelstein, Rebecca L, Henry, Olivier, Ochocki, Joshua, DeGraw, Amanda, Lenevich, Stepan, Talbot, Trista, Young, Victor G, Hruza, Alan W, Lopez-Gallego, Fernando, Labello, Nicholas P, Strickland, Corey L, Schmidt-Dannert, Claudia, Distefano, Mark D
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Published in Chemical biology & drug design (2010)
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FACTOR XIA INHIBITORS
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Year of Publication 18.11.2020
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Year of Publication 17.04.2018
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Year of Publication 13.06.2017
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Year of Publication 03.01.2018
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Year of Publication 21.12.2016
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