Contemporary approaches to site-selective protein modification
Hoyt, Emily A., Cal, Pedro M. S. D., Oliveira, Bruno L., Bernardes, Gonçalo J. L.
Published in Nature reviews. Chemistry (01.03.2019)
Published in Nature reviews. Chemistry (01.03.2019)
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Alkynyl Benzoxazines and Dihydroquinazolines as Cysteine Targeting Covalent Warheads and Their Application in Identification of Selective Irreversible Kinase Inhibitors
McAulay, Kirsten, Hoyt, Emily A., Thomas, Morgan, Schimpl, Marianne, Bodnarchuk, Michael S., Lewis, Hilary J., Barratt, Derek, Bhavsar, Deepa, Robinson, David M., Deery, Michael J., Ogg, Derek J., Bernardes, Goncalo J. L., Ward, Richard A., Waring, Michael J., Kettle, Jason G.
Published in Journal of the American Chemical Society (10.06.2020)
Published in Journal of the American Chemical Society (10.06.2020)
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Stable Pyrrole‐Linked Bioconjugates through Tetrazine‐Triggered Azanorbornadiene Fragmentation
Gil de Montes, Enrique, Istrate, Alena, Navo, Claudio D., Jiménez‐Moreno, Ester, Hoyt, Emily A., Corzana, Francisco, Robina, Inmaculada, Jiménez‐Osés, Gonzalo, Moreno‐Vargas, Antonio J., Bernardes, Gonçalo J. L.
Published in Angewandte Chemie International Edition (06.04.2020)
Published in Angewandte Chemie International Edition (06.04.2020)
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Single Mutation on Trastuzumab Modulates the Stability of Antibody–Drug Conjugates Built Using Acetal-Based Linkers and Thiol-Maleimide Chemistry
Ferhati, Xhenti, Jiménez-Moreno, Ester, Hoyt, Emily A, Salluce, Giulia, Cabeza-Cabrerizo, Mar, Navo, Claudio D, Compañón, Ismael, Akkapeddi, Padma, Matos, Maria J, Salaverri, Noelia, Garrido, Pablo, Martínez, Alfredo, Laserna, Víctor, Murray, Thomas V, Jiménez-Osés, Gonzalo, Ravn, Peter, Bernardes, Gonçalo J. L, Corzana, Francisco
Published in Journal of the American Chemical Society (30.03.2022)
Published in Journal of the American Chemical Society (30.03.2022)
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Journal Article
Stable Pyrrole‐Linked Bioconjugates through Tetrazine‐Triggered Azanorbornadiene Fragmentation
Gil de Montes, Enrique, Istrate, Alena, Navo, Claudio D., Jiménez‐Moreno, Ester, Hoyt, Emily A., Corzana, Francisco, Robina, Inmaculada, Jiménez‐Osés, Gonzalo, Moreno‐Vargas, Antonio J., Bernardes, Gonçalo J. L.
Published in Angewandte Chemie (06.04.2020)
Published in Angewandte Chemie (06.04.2020)
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Adaptive Optimization of Chemical Reactions with Minimal Experimental Information
Reker, Daniel, Hoyt, Emily A., Bernardes, Gonçalo J.L., Rodrigues, Tiago
Published in Cell reports physical science (18.11.2020)
Published in Cell reports physical science (18.11.2020)
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