PA-6 inhibits inward rectifier currents carried by V93I and D172N gain-of-function KIR2.1 channels, but increases channel protein expression
Ji, Yuan, Veldhuis, Marlieke G, Zandvoort, Jantien, Romunde, Fee L, Houtman, Marien J. C, Duran, Karen, van Haaften, Gijs, Zangerl-Plessl, Eva-Maria, Takanari, Hiroki, Stary-Weinzinger, Anna, van der Heyden, Marcel A. G
Published in Journal of biomedical science (15.07.2017)
Published in Journal of biomedical science (15.07.2017)
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Development of IKATP Ion Channel Blockers Targeting Sulfonylurea Resistant Mutant KIR6.2 Based Channels for Treating DEND Syndrome
Houtman, Marien J. C., Friesacher, Theres, Chen, Xingyu, Zangerl-Plessl, Eva-Maria, Heyden, Marcel A. G. van der, Stary-Weinzinger, Anna
Published in Frontiers in pharmacology (14.01.2022)
Published in Frontiers in pharmacology (14.01.2022)
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Short-term Variability of Repolarization Is Superior to Other Repolarization Parameters in the Evaluation of Diverse Antiarrhythmic Interventions in the Chronic Atrioventricular Block Dog
Bossu, Alexandre, Varkevisser, Rosanne, Beekman, Henriette D M, Houtman, Marien J C, van der Heyden, Marcel A G, Vos, Marc A
Published in Journal of cardiovascular pharmacology (01.06.2017)
Published in Journal of cardiovascular pharmacology (01.06.2017)
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Identification of a PEST Sequence in Vertebrate KIR2.1 That Modifies Rectification
Qile, Muge, Ji, Yuan, Houtman, Marien J. C., Veldhuis, Marlieke, Romunde, Fee, Kok, Bart, van der Heyden, Marcel A. G.
Published in Frontiers in physiology (05.07.2019)
Published in Frontiers in physiology (05.07.2019)
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Computational Identification of Novel Kir6 Channel Inhibitors
Chen, Xingyu, Garon, Arthur, Wieder, Marcus, Houtman, Marien J C, Zangerl-Plessl, Eva-Maria, Langer, Thierry, van der Heyden, Marcel A G, Stary-Weinzinger, Anna
Published in Frontiers in pharmacology (24.05.2019)
Published in Frontiers in pharmacology (24.05.2019)
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Late Na+ Current Inhibition by Ranolazine Reduces Torsades de Pointes in the Chronic Atrioventricular Block Dog Model
Antoons, Gudrun, PhD, Oros, Avram, MD, PhD, Beekman, Jet D.M., BSc, Engelen, Markus A., MD, Houtman, Marien J.C., BSc, Belardinelli, Luiz, MD, Stengl, Milan, PhD, Vos, Marc A., PhD
Published in Journal of the American College of Cardiology (23.02.2010)
Published in Journal of the American College of Cardiology (23.02.2010)
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Inhibition of cardiomyocyte automaticity by electrotonic application of inward rectifier current from Kir2.1 expressing cells
de Boer, Teun P, van Veen, Toon A B, Houtman, Marien J C, Jansen, John A, van Amersfoorth, Shirley C M, Doevendans, Pieter A, Vos, Marc A, van der Heyden, Marcel A G
Published in Medical & biological engineering & computing (01.07.2006)
Published in Medical & biological engineering & computing (01.07.2006)
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Drug-Induced Torsade de Pointes Arrhythmias in the Chronic AV Block Dog Are Perpetuated by Focal Activity
Boulaksil, Mohamed, Jungschleger, Jerome G, Antoons, Gudrun, Houtman, Marien J.C, de Boer, Teun P, Wilders, Ronald, Beekman, Jet D, Maessen, Jos G, van der Hulst, Ferenc F, van der Heyden, Marcel A.G, van Veen, Toon A.B, van Rijen, Harold V.M, de Bakker, Jacques M.T, Vos, Marc A
Published in Circulation. Arrhythmia and electrophysiology (01.08.2011)
Published in Circulation. Arrhythmia and electrophysiology (01.08.2011)
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LUF7244 plus Dofetilide Rescues Aberrant K v 11.1 Trafficking and Produces Functional I Kv11.1
Qile, Muge, Ji, Yuan, Golden, Tyona D, Houtman, Marien J C, Romunde, Fee, Fransen, Doreth, van Ham, Willem B, IJzerman, Ad P, January, Craig T, Heitman, Laura H, Stary-Weinzinger, Anna, Delisle, Brian P, van der Heyden, Marcel A G
Published in Molecular pharmacology (01.06.2020)
Published in Molecular pharmacology (01.06.2020)
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Selective late sodium current inhibitor GS‐458967 suppresses Torsades de Pointes by mostly affecting perpetuation but not initiation of the arrhythmia
Bossu, Alexandre, Houtman, Marien J C, Meijborg, Veronique M F, Varkevisser, Rosanne, Beekman, Henriette D M, Dunnink, Albert, Bakker, Jacques M T, Mollova, Nevena, Rajamani, Sridharan, Belardinelli, Luiz, Heyden, Marcel A G, Vos, Marc A
Published in British journal of pharmacology (01.06.2018)
Published in British journal of pharmacology (01.06.2018)
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Glibenclamide and HMR1098 normalize Cantú syndrome‐associated gain‐of‐function currents
Houtman, Marien J. C., Chen, Xingyu, Qile, Muge, Duran, Karen, Haaften, Gijs, Stary‐Weinzinger, Anna, Heyden, Marcel A. G.
Published in Journal of cellular and molecular medicine (01.08.2019)
Published in Journal of cellular and molecular medicine (01.08.2019)
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Istaroxime, a positive inotropic agent devoid of proarrhythmic properties in sensitive chronic atrioventricular block dogs
Bossu, Alexandre, Kostense, Amée, Beekman, Henriette D.M., Houtman, Marien J.C., van der Heyden, Marcel A.G., Vos, Marc A.
Published in Pharmacological research (01.07.2018)
Published in Pharmacological research (01.07.2018)
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Calcium release near l -type calcium channels promotes beat-to-beat variability in ventricular myocytes from the chronic AV block dog
Antoons, Gudrun, Johnson, Daniel M, Dries, Eef, Santiago, Demetrio J, Ozdemir, Semir, Lenaerts, Ilse, Beekman, Jet D.M, Houtman, Marien J.C, Sipido, Karin R, Vos, Marc A
Published in Journal of molecular and cellular cardiology (01.12.2015)
Published in Journal of molecular and cellular cardiology (01.12.2015)
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Reduction of fibrosis-related arrhythmias by chronic renin-angiotensin-aldosterone system inhibitors in an aged mouse model
Stein, Mera, Boulaksil, Mohamed, Jansen, John A, Herold, Eva, Noorman, Maartje, Joles, Jaap A, van Veen, Toon A B, Houtman, Marien J C, Engelen, Markus A, Hauer, Richard N W, de Bakker, Jacques M T, van Rijen, Harold V M
Published in American journal of physiology. Heart and circulatory physiology (01.08.2010)
Published in American journal of physiology. Heart and circulatory physiology (01.08.2010)
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Inhibiting the clathrin-mediated endocytosis pathway rescues K(IR)2.1 downregulation by pentamidine
Varkevisser, Rosanne, Houtman, Marien J C, Waasdorp, Maaike, Man, Joyce C K, Heukers, Raimond, Takanari, Hiroki, Tieland, Ralph G, van Bergen En Henegouwen, Paul M P, Vos, Marc A, van der Heyden, Marcel A G
Published in Pflügers Archiv (01.02.2013)
Published in Pflügers Archiv (01.02.2013)
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Inhibition of lysosomal degradation rescues pentamidine-mediated decreases of K(IR)2.1 ion channel expression but not that of K(v)11.1
Nalos, Lukas, de Boer, Teun P, Houtman, Marien J C, Rook, Martin B, Vos, Marc A, van der Heyden, Marcel A G
Published in European journal of pharmacology (10.02.2011)
Published in European journal of pharmacology (10.02.2011)
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Relevance of calmodulin/CaMKII activation for arrhythmogenesis in the AV block dog
Bourgonje, Vincent J.A., Msc, Schoenmakers, Marieke, MD, PhD, Beekman, Jet D.M, van der Nagel, Roel, Bsc, Houtman, Marien J.C., Bsc, Miedema, Lars F., Bsc, Antoons, Gudrun, PhD, Sipido, Karin, MD, PhD, de Windt, Leon J., PhD, van Veen, Toon A.B., PhD, Vos, Marc A., PhD
Published in Heart rhythm (01.11.2012)
Published in Heart rhythm (01.11.2012)
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Journal Article
Inhibiting the clathrin-mediated endocytosis pathway rescues KIR2.1 downregulation by pentamidine
Varkevisser, Rosanne, Houtman, Marien J. C., Waasdorp, Maaike, Man, Joyce C. K., Heukers, Raimond, Takanari, Hiroki, Tieland, Ralph G., van Bergen en Henegouwen, Paul M. P., Vos, Marc A., van der Heyden, Marcel A. G.
Published in Pflügers Archiv (01.02.2013)
Published in Pflügers Archiv (01.02.2013)
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Experimental Mapping of the Canine KCNJ2 and KCNJ12 Gene Structures and Functional Analysis of the Canine K(IR)2.2 ion Channel
Houtman, Marien J C, Takanari, Hiroki, Kok, Bart G J M, van Eck, Margot, Montagne, Denise R, Vos, Marc A, de Boer, Teun P, van der Heyden, Marcel A G
Published in Frontiers in physiology (2012)
Published in Frontiers in physiology (2012)
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