Sulfonium Ligands of the α7 nAChR
Horenstein, Nicole A, Stokes, Clare, Papke, Roger L
Published in Molecules (Basel, Switzerland) (17.09.2021)
Published in Molecules (Basel, Switzerland) (17.09.2021)
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A silent agonist of α7 nicotinic acetylcholine receptors modulates inflammation ex vivo and attenuates EAE
Godin, Jean-Rémi, Roy, Patrick, Quadri, Marta, Bagdas, Deniz, Toma, Wisam, Narendrula-Kotha, Ramya, Kishta, Osama A., Damaj, M. Imad, Horenstein, Nicole A., Papke, Roger L., Simard, Alain R.
Published in Brain, behavior, and immunity (01.07.2020)
Published in Brain, behavior, and immunity (01.07.2020)
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Design, synthesis, and electrophysiological evaluation of NS6740 derivatives: Exploration of the structure-activity relationship for alpha7 nicotinic acetylcholine receptor silent activation
Pismataro, Maria Chiara, Horenstein, Nicole A., Stokes, Clare, Quadri, Marta, De Amici, Marco, Papke, Roger L., Dallanoce, Clelia
Published in European journal of medicinal chemistry (01.11.2020)
Published in European journal of medicinal chemistry (01.11.2020)
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Comparison of the Anti-inflammatory Properties of Two Nicotinic Acetylcholine Receptor Ligands, Phosphocholine and pCF3-diEPP
Richter, Katrin, Papke, Roger L., Stokes, Clare, Roy, Danika C., Espinosa, Eduardo S., Wolf, Philipp M. K., Hecker, Andreas, Liese, Juliane, Singh, Vijay K., Padberg, Winfried, Schlüter, Klaus-Dieter, Rohde, Marius, McIntosh, J. Michael, Morley, Barbara J., Horenstein, Nicole A., Grau, Veronika, Simard, Alain R.
Published in Frontiers in cellular neuroscience (31.03.2022)
Published in Frontiers in cellular neuroscience (31.03.2022)
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Differential Regulation of Receptor Activation and Agonist Selectivity by Highly Conserved Tryptophans in the Nicotinic Acetylcholine Receptor Binding Site
Williams, Dustin K, Stokes, Clare, Horenstein, Nicole A, Papke, Roger L
Published in The Journal of pharmacology and experimental therapeutics (01.07.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2009)
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Reversal of Agonist Selectivity by Mutations of Conserved Amino Acids in the Binding Site of Nicotinic Acetylcholine Receptors
Horenstein, Nicole A., McCormack, Thomas J., Stokes, Clare, Ren, Ke, Papke, Roger L.
Published in The Journal of biological chemistry (23.02.2007)
Published in The Journal of biological chemistry (23.02.2007)
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Cracking the Betel Nut: Cholinergic Activity of Areca Alkaloids and Related Compounds
Horenstein, Nicole A, Quadri, Marta, Stokes, Clare, Shoaib, Mohammed, Papke, Roger L
Published in Nicotine & tobacco research (21.05.2019)
Published in Nicotine & tobacco research (21.05.2019)
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Allosteric Agonism of α7 Nicotinic Acetylcholine Receptors: Receptor Modulation Outside the Orthosteric Site
Gulsevin, Alican, Papke, Roger L, Stokes, Clare, Garai, Sumanta, Thakur, Ganesh A, Quadri, Marta, Horenstein, Nicole A
Published in Molecular pharmacology (01.06.2019)
Published in Molecular pharmacology (01.06.2019)
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Dissection of N,N-diethyl-N′-phenylpiperazines as α7 nicotinic receptor silent agonists
Quadri, Marta, Papke, Roger L., Horenstein, Nicole A.
Published in Bioorganic & medicinal chemistry (15.01.2016)
Published in Bioorganic & medicinal chemistry (15.01.2016)
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Stable desensitization of α7 nicotinic acetylcholine receptors by NS6740 requires interaction with S36 in the orthosteric agonist binding site
Pismataro, Maria Chiara, Horenstein, Nicole A., Stokes, Clare, Dallanoce, Clelia, Thakur, Ganesh A., Papke, Roger L.
Published in European journal of pharmacology (15.08.2021)
Published in European journal of pharmacology (15.08.2021)
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