Improvement of the Pharmacokinetics and In Vivo Antibacterial Efficacy of a Novel Type IIa Topoisomerase Inhibitor by Formulation in Liposomes
SHAPIRO, Adam B, NEWMAN, Joseph, GOTETI, Kosalaram, BEAUDOIN, Marie-Eve, HARRISON, Rane, HOPKINS, Sussie, AGRAWAL, Nikunj, RIVIN, Olga
Published in Antimicrobial Agents and Chemotherapy (01.10.2013)
Published in Antimicrobial Agents and Chemotherapy (01.10.2013)
Get full text
Journal Article
NBTI 5463 Is a Novel Bacterial Type II Topoisomerase Inhibitor with Activity against Gram-Negative Bacteria and In Vivo Efficacy
DOUGHERTY, Thomas J, NAYAR, Asha, NEWMAN, Joseph V, HOPKINS, Sussie, STONE, Gregory G, JOHNSTONE, Michele, SHAPIRO, Adam B, CRONIN, Mark, RECK, Folkert, EHMANN, David E
Published in Antimicrobial agents and chemotherapy (01.05.2014)
Published in Antimicrobial agents and chemotherapy (01.05.2014)
Get full text
Journal Article
Optimization of physicochemical properties and safety profile of novel bacterial topoisomerase type II inhibitors (NBTIs) with activity against Pseudomonas aeruginosa
Reck, Folkert, Ehmann, David E., Dougherty, Thomas J., Newman, Joseph V., Hopkins, Sussie, Stone, Gregory, Agrawal, Nikunj, Ciaccio, Paul, McNulty, John, Barthlow, Herbert, O’Donnell, Jennifer, Goteti, Kosalaram, Breen, John, Comita-Prevoir, Janelle, Cornebise, Mark, Cronin, Mark, Eyermann, Charles J., Geng, Bolin, Carr, Greg R., Pandarinathan, Lakshmipathi, Tang, Xuejun, Cottone, Andrew, Zhao, Liang, Bezdenejnih-Snyder, Natascha
Published in Bioorganic & medicinal chemistry (01.10.2014)
Published in Bioorganic & medicinal chemistry (01.10.2014)
Get full text
Journal Article
NBTI 5463 Is a Novel Bacterial Type II Topoisomerase Inhibitor with Activity against Gram-Negative Bacteria and In Vivo Efficacy
Dougherty, Thomas J, Nayar, Asha, Newman, Joseph V, Hopkins, Sussie, Stone, Gregory G, Johnstone, Michele, Shapiro, Adam B, Cronin, Mark, Reck, Folkert, Ehmann, David E
Published in Antimicrobial agents and chemotherapy (01.07.2014)
Published in Antimicrobial agents and chemotherapy (01.07.2014)
Get full text
Journal Article