Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876
Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Müller, Thomas, Bauser, Marcus, Buchmann, Bernd
Published in ChemMedChem (19.10.2016)
Published in ChemMedChem (19.10.2016)
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Mechanism of inhibition of human glucose transporter GLUT1 is conserved between cytochalasin B and phenylalanine amides
Kapoor, Khyati, Finer-Moore, Janet S., Pedersen, Bjørn P., Caboni, Laura, Waight, Andrew, Hillig, Roman C., Bringmann, Peter, Heisler, Iring, Müller, Thomas, Siebeneicher, Holger, Stroud, Robert M.
Published in Proceedings of the National Academy of Sciences - PNAS (26.04.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (26.04.2016)
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Preclinical Efficacy of the Novel Monocarboxylate Transporter 1 Inhibitor BAY-8002 and Associated Markers of Resistance
Quanz, Maria, Bender, Eckhard, Kopitz, Charlotte, Grünewald, Sylvia, Schlicker, Andreas, Schwede, Wolfgang, Eheim, Ashley, Toschi, Luisella, Neuhaus, Roland, Richter, Carmen, Toedling, Joern, Merz, Claudia, Lesche, Ralf, Kamburov, Atanas, Siebeneicher, Holger, Bauser, Marcus, Hägebarth, Andrea
Published in Molecular cancer therapeutics (01.11.2018)
Published in Molecular cancer therapeutics (01.11.2018)
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A Flexible and Catalytic One-Pot Procedure for the Synthesis of Indoles
Siebeneicher, Holger, Bytschkov, Igor, Doye, Sven
Published in Angewandte Chemie International Edition (07.07.2003)
Published in Angewandte Chemie International Edition (07.07.2003)
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A Flexible Synthesis of Indoline, Indolizidine, and Pyrrolizidine Derivatives
Bytschkov, Igor, Siebeneicher, Holger, Doye, Sven
Published in European journal of organic chemistry (01.08.2003)
Published in European journal of organic chemistry (01.08.2003)
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Journal Article
Discovery of IRAK4 Inhibitors BAY1834845 (Zabedosertib) and BAY1830839
Bothe, Ulrich, Günther, Judith, Nubbemeyer, Reinhard, Siebeneicher, Holger, Ring, Sven, Bömer, Ulf, Peters, Michaele, Rausch, Alexandra, Denner, Karsten, Himmel, Herbert, Sutter, Andreas, Terebesi, Ildiko, Lange, Martin, Wengner, Antje M., Guimond, Nicolas, Thaler, Tobias, Platzek, Johannes, Eberspächer, Uwe, Schäfer, Martina, Steuber, Holger, Zollner, Thomas M., Steinmeyer, Andreas, Schmidt, Nicole
Published in Journal of medicinal chemistry (25.01.2024)
Published in Journal of medicinal chemistry (25.01.2024)
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Journal Article
Identification of novel GLUT inhibitors
Siebeneicher, Holger, Bauser, Marcus, Buchmann, Bernd, Heisler, Iring, Müller, Thomas, Neuhaus, Roland, Rehwinkel, Hartmut, Telser, Joachim, Zorn, Ludwig
Published in Bioorganic & medicinal chemistry letters (01.04.2016)
Published in Bioorganic & medicinal chemistry letters (01.04.2016)
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Abstract 4333: Identification and optimization of the first highly selective GLUT-1 inhibitors
Bauser, Marcus, Buchmann, Bernd, Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Mueller, Thomas, Kopitz, Charlotte Christine
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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sup 18^F-GP1, a Novel PET Tracer Designed for High-Sensitivity, Low-Background Detection of Thrombi
Lohrke, Jessica, Siebeneicher, Holger, Berger, Markus, Reinhardt, Michael, Berndt, Mathias, Mueller, Andre, Zerna, Marion, Koglin, Norman, Oden, Felix, Bauser, Marcus, Friebe, Matthias, Dinkelborg, Ludger M, Huetter, Joachim, Stephens, Andrew W
Published in The Journal of nuclear medicine (1978) (01.07.2017)
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Published in The Journal of nuclear medicine (1978) (01.07.2017)
Journal Article
18 F-GP1, a Novel PET Tracer Designed for High-Sensitivity, Low-Background Detection of Thrombi
Lohrke, Jessica, Siebeneicher, Holger, Berger, Markus, Reinhardt, Michael, Berndt, Mathias, Mueller, Andre, Zerna, Marion, Koglin, Norman, Oden, Felix, Bauser, Marcus, Friebe, Matthias, Dinkelborg, Ludger M, Huetter, Joachim, Stephens, Andrew W
Published in Journal of Nuclear Medicine (01.07.2017)
Published in Journal of Nuclear Medicine (01.07.2017)
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Abstract 1887: Preclinical evaluation of a novel interleukin-1 receptor-associated kinase 4 (IRAK4) inhibitor in combination with PI3K inhibitor copanlisib or BTK inhibitors in ABC-DLBCL
Lange, Martin, Wengner, Antje Margret, Bothe, Ulrich, Boemer, Ulf, Nubbemeyer, Reinhard, Siebeneicher, Holger, Steuber, Holger, Guenther, Judith, Potze, Lisette, Schmidt, Nicole, Politz, Oliver, Doecke, Wolf-Dietrich, Lagkadinou, Eleni, Zollner, Thomas M., Nussbaum, Franz von, Mumberg, Dominik, Steinmeyer, Andreas, Brands, Michael, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Cover Picture: Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876 (ChemMedChem 20/2016)
Siebeneicher, Holger, Cleve, Arwed, Rehwinkel, Hartmut, Neuhaus, Roland, Heisler, Iring, Müller, Thomas, Bauser, Marcus, Buchmann, Bernd
Published in ChemMedChem (19.10.2016)
Published in ChemMedChem (19.10.2016)
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Journal Article
[ 18 F]Fluoropyruvate: radiosynthesis and initial biological evaluation: [ 18 F]Fluoropyruvate
Graham, Keith, Müller, Andre, Lehmann, Lutz, Koglin, Norman, Dinkelborg, Ludger, Siebeneicher, Holger
Published in Journal of labelled compounds & radiopharmaceuticals (01.03.2014)
Published in Journal of labelled compounds & radiopharmaceuticals (01.03.2014)
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Journal Article
18F-GP1, a Novel PET Tracer Designed for High-Sensitivity, Low-Background Detection of Thrombi
Lohrke, Jessica, Siebeneicher, Holger, Berger, Markus, Reinhardt, Michael, Berndt, Mathias, Mueller, Andre, Zerna, Marion, Koglin, Norman, Oden, Felix, Bauser, Marcus, Friebe, Matthias, Dinkelborg, Ludger M, Huetter, Joachim, Stephens, Andrew W
Published in The Journal of nuclear medicine (1978) (01.07.2017)
Published in The Journal of nuclear medicine (1978) (01.07.2017)
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Journal Article