Mitocryptides from Human Mitochondrial DNA-Encoded Proteins Activate Neutrophil Formyl Peptide Receptors: Receptor Preference and Signaling Properties
Gabl, Michael, Sundqvist, Martina, Holdfeldt, Andre, Lind, Simon, Mårtensson, Jonas, Christenson, Karin, Marutani, Takayuki, Dahlgren, Claes, Mukai, Hidehito, Forsman, Huamei
Published in The Journal of immunology (1950) (01.05.2018)
Published in The Journal of immunology (1950) (01.05.2018)
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Structure–Function Characteristics and Signaling Properties of Lipidated Peptidomimetic FPR2 Agonists: Peptoid Stereochemistry and Residues in the Vicinity of the Headgroup Affect Function
Holdfeldt, Andre, Skovbakke, Sarah Line, Gabl, Michael, Nielsen, Christina, Dahlgren, Claes, Franzyk, Henrik, Forsman, Huamei
Published in ACS omega (31.03.2019)
Published in ACS omega (31.03.2019)
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Journal Article
Basic characteristics of the neutrophil receptors that recognize formylated peptides, a danger-associated molecular pattern generated by bacteria and mitochondria
Dahlgren, Claes, Gabl, Michael, Holdfeldt, André, Winther, Malene, Forsman, Huamei
Published in Biochemical pharmacology (15.08.2016)
Published in Biochemical pharmacology (15.08.2016)
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Journal Article
The PAR4-derived pepducin P4Pal10 lacks effect on neutrophil GPCRs that couple to Gαq for signaling but distinctly modulates function of the Gαi-coupled FPR2 and FFAR2
Holdfeldt, André, Lind, Simon, Hesse, Camilla, Dahlgren, Claes, Forsman, Huamei
Published in Biochemical pharmacology (01.10.2020)
Published in Biochemical pharmacology (01.10.2020)
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Journal Article
Staphylococcus aureus -Derived PSMα Peptides Activate Neutrophil FPR2 but Lack the Ability to Mediate β-Arrestin Recruitment and Chemotaxis
Sundqvist, Martina, Christenson, Karin, Gabl, Michael, Holdfeldt, André, Jennbacken, Karin, Møller, Thor C, Dahlgren, Claes, Forsman, Huamei
Published in The Journal of immunology (1950) (15.12.2019)
Published in The Journal of immunology (1950) (15.12.2019)
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Journal Article
Similarities and differences between the responses induced in human phagocytes through activation of the medium chain fatty acid receptor GPR84 and the short chain fatty acid receptor FFA2R
Sundqvist, Martina, Christenson, Karin, Holdfeldt, André, Gabl, Michael, Mårtensson, Jonas, Björkman, Lena, Dieckmann, Regis, Dahlgren, Claes, Forsman, Huamei
Published in Biochimica et biophysica acta (01.05.2018)
Published in Biochimica et biophysica acta (01.05.2018)
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Journal Article
Combining Elements from Two Antagonists of Formyl Peptide Receptor 2 Generates More Potent Peptidomimetic Antagonists
Skovbakke, Sarah Line, Holdfeldt, André, Nielsen, Christina, Hansen, Anna Mette, Perez-Gassol, Iris, Dahlgren, Claes, Forsman, Huamei, Franzyk, Henrik
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
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Journal Article
Multiple ligand recognition sites in free fatty acid receptor 2 (FFA2R) direct distinct neutrophil activation patterns
Lind, Simon, Holdfeldt, André, Mårtensson, Jonas, Granberg, Kenneth L., Forsman, Huamei, Dahlgren, Claes
Published in Biochemical pharmacology (01.11.2021)
Published in Biochemical pharmacology (01.11.2021)
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Journal Article
Functional selective ATP receptor signaling controlled by the free fatty acid receptor 2 through a novel allosteric modulation mechanism
Lind, Simon, Holdfeldt, André, Mårtensson, Jonas, Sundqvist, Martina, Björkman, Lena, Forsman, Huamei, Dahlgren, Claes
Published in The FASEB journal (01.06.2019)
Published in The FASEB journal (01.06.2019)
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Journal Article
GRK2 selectively attenuates the neutrophil NADPH-oxidase response triggered by β-arrestin recruiting GPR84 agonists
Fredriksson, Johanna, Holdfeldt, André, Mårtensson, Jonas, Björkman, Lena, Møller, Thor C., Müllers, Erik, Dahlgren, Claes, Sundqvist, Martina, Forsman, Huamei
Published in Biochimica et biophysica acta. Molecular cell research (01.07.2022)
Published in Biochimica et biophysica acta. Molecular cell research (01.07.2022)
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Journal Article
Identification of Residues Critical for FPR2 Activation by the Cryptic Peptide Mitocryptide-2 Originating from the Mitochondrial DNA-Encoded Cytochrome b
Lind, Simon, Gabl, Michael, Holdfeldt, André, Mårtensson, Jonas, Sundqvist, Martina, Nishino, Kodai, Dahlgren, Claes, Mukai, Hidehito, Forsman, Huamei
Published in The Journal of immunology (1950) (01.05.2019)
Published in The Journal of immunology (1950) (01.05.2019)
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Journal Article
Neutrophil Signaling That Challenges Dogmata of G Protein-Coupled Receptor Regulated Functions
Dahlgren, Claes, Holdfeldt, André, Lind, Simon, Mårtensson, Jonas, Gabl, Michael, Björkman, Lena, Sundqvist, Martina, Forsman, Huamei
Published in ACS pharmacology & translational science (10.04.2020)
Published in ACS pharmacology & translational science (10.04.2020)
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Journal Article
Lack of Receptor for Advanced Glycation End Products Leads to Less Severe Staphylococcal Skin Infection but More Skin Abscesses and Prolonged Wound Healing
Na, Manli, Mohammad, Majd, Fei, Ying, Wang, Wanzhong, Holdfeldt, André, Forsman, Huamei, Ali, Abukar, Pullerits, Rille, Jin, Tao
Published in The Journal of infectious diseases (24.07.2018)
Published in The Journal of infectious diseases (24.07.2018)
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Journal Article
Interdependent allosteric free fatty acid receptor 2 modulators synergistically induce functional selective activation and desensitization in neutrophils
Lind, Simon, Holdfeldt, André, Mårtensson, Jonas, Sundqvist, Martina, Kenakin, Terry P., Björkman, Lena, Forsman, Huamei, Dahlgren, Claes
Published in Biochimica et biophysica acta. Molecular cell research (01.06.2020)
Published in Biochimica et biophysica acta. Molecular cell research (01.06.2020)
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Journal Article
Formyl peptide derived lipopeptides disclose differences between the receptors in mouse and men and call the pepducin concept in question
Winther, Malene, Holdfeldt, André, Sundqvist, Martina, Rajabkhani, Zahra, Gabl, Michael, Bylund, Johan, Dahlgren, Claes, Forsman, Huamei
Published in PloS one (21.09.2017)
Published in PloS one (21.09.2017)
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Journal Article
Neutrophil priming that turns natural FFA2R agonists into potent activators of the superoxide generating NADPH‐oxidase
Mårtensson, Jonas, Holdfeldt, André, Sundqvist, Martina, Gabl, Michael, Kenakin, Terry P., Björkman, Lena, Forsman, Huamei, Dahlgren, Claes
Published in Journal of leukocyte biology (01.12.2018)
Published in Journal of leukocyte biology (01.12.2018)
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Journal Article
Barbadin selectively modulates FPR2-mediated neutrophil functions independent of receptor endocytosis
Sundqvist, Martina, Holdfeldt, André, Wright, Shane C., Møller, Thor C., Siaw, Esther, Jennbacken, Karin, Franzyk, Henrik, Bouvier, Michel, Dahlgren, Claes, Forsman, Huamei
Published in Biochimica et biophysica acta. Molecular cell research (01.12.2020)
Published in Biochimica et biophysica acta. Molecular cell research (01.12.2020)
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