Combating Enhanced Intracellular Survival (Eis)-Mediated Kanamycin Resistance of Mycobacterium tuberculosis by Novel Pyrrolo[1,5‑a]pyrazine-Based Eis Inhibitors
Garzan, Atefeh, Willby, Melisa J, Ngo, Huy X, Gajadeera, Chathurada S, Green, Keith D, Holbrook, Selina Y. L, Hou, Caixia, Posey, James E, Tsodikov, Oleg V, Garneau-Tsodikova, Sylvie
Published in ACS infectious diseases (14.04.2017)
Published in ACS infectious diseases (14.04.2017)
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Repurposing antipsychotic drugs into antifungal agents: Synergistic combinations of azoles and bromperidol derivatives in the treatment of various fungal infections
Holbrook, Selina Y.L., Garzan, Atefeh, Dennis, Emily K., Shrestha, Sanjib K., Garneau-Tsodikova, Sylvie
Published in European journal of medicinal chemistry (20.10.2017)
Published in European journal of medicinal chemistry (20.10.2017)
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Discovery of substituted benzyloxy-benzylamine inhibitors of acetyltransferase Eis and their anti-mycobacterial activity
Pang, Allan H., Green, Keith D., Chandrika, Nishad Thamban, Garzan, Atefeh, Punetha, Ankita, Holbrook, Selina Y.L., Willby, Melisa J., Posey, James E., Tsodikov, Oleg V., Garneau-Tsodikova, Sylvie
Published in European journal of medicinal chemistry (15.11.2022)
Published in European journal of medicinal chemistry (15.11.2022)
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Structure-Guided Optimization of Inhibitors of Acetyltransferase Eis from Mycobacterium tuberculosis
Punetha, Ankita, Ngo, Huy X, Holbrook, Selina Y L, Green, Keith D, Willby, Melisa J, Bonnett, Shilah A, Krieger, Kyle, Dennis, Emily K, Posey, James E, Parish, Tanya, Tsodikov, Oleg V, Garneau-Tsodikova, Sylvie
Published in ACS chemical biology (19.06.2020)
Published in ACS chemical biology (19.06.2020)
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Structure-based design of haloperidol analogues as inhibitors of acetyltransferase Eis from Mycobacterium tuberculosis to overcome kanamycin resistance
Punetha, Ankita, Green, Keith D., Garzan, Atefeh, Thamban Chandrika, Nishad, Willby, Melisa J., Pang, Allan H., Hou, Caixia, Holbrook, Selina Y. L., Krieger, Kyle, Posey, James E., Parish, Tanya, Tsodikov, Oleg V., Garneau-Tsodikova, Sylvie
Published in MedChemComm (17.11.2021)
Published in MedChemComm (17.11.2021)
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Potent 1,2,4-Triazino[5,6b]indole-3-thioether Inhibitors of the Kanamycin Resistance Enzyme Eis from Mycobacterium tuberculosis
Ngo, Huy X., Green, Keith D., Gajadeera, Chathurada S., Willby, Melisa J., Holbrook, Selina Y. L., Hou, Caixia, Garzan, Atefeh, Mayhoub, Abdelrahman S., Posey, James E., Tsodikov, Oleg. V., Garneau-Tsodikova, Sylvie
Published in ACS infectious diseases (08.06.2018)
Published in ACS infectious diseases (08.06.2018)
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Nucleoside triphosphate cosubstrates control the substrate profile and efficiency of aminoglycoside 3′-O-phosphotransferase type IIaElectronic supplementary information (ESI) available. See DOI: 10.1039/c8md00234g
Holbrook, Selina Y. L, Gentry, Matthew S, Tsodikov, Oleg V, Garneau-Tsodikova, Sylvie
Year of Publication 15.08.2018
Year of Publication 15.08.2018
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Nucleoside triphosphate cosubstrates control the substrate profile and efficiency of aminoglycoside 3′-O-phosphotransferase type IIa† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c8md00234g
Holbrook, Selina Y. L., Gentry, Matthew S., Tsodikov, Oleg V., Garneau-Tsodikova, Sylvie
Published in MedChemComm (16.07.2018)
Published in MedChemComm (16.07.2018)
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Structure-based design of haloperidol analogues as inhibitors of acetyltransferase Eis from to overcome kanamycin resistance
Punetha, Ankita, Green, Keith D, Garzan, Atefeh, Thamban Chandrika, Nishad, Willby, Melisa J, Pang, Allan H, Hou, Caixia, Holbrook, Selina Y. L, Krieger, Kyle, Posey, James E, Parish, Tanya, Tsodikov, Oleg V, Garneau-Tsodikova, Sylvie
Published in RSC medicinal chemistry (17.11.2021)
Published in RSC medicinal chemistry (17.11.2021)
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