Evolutionary drivers of thermoadaptation in enzyme catalysis
Nguyen, Vy, Wilson, Christopher, Hoemberger, Marc, Stiller, John B., Agafonov, Roman V., Kutter, Steffen, English, Justin, Theobald, Douglas L., Kern, Dorothee
Published in Science (American Association for the Advancement of Science) (20.01.2017)
Published in Science (American Association for the Advancement of Science) (20.01.2017)
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Journal Article
Allosteric modulation of a human protein kinase with monobodies
Zorba, Adelajda, Nguyen, Vy, Koide, Akiko, Hoemberger, Marc, Zheng, Yuejiao, Kutter, Steffen, Kim, Chansik, Koide, Shohei, Kern, Dorothee
Published in Proceedings of the National Academy of Sciences - PNAS (09.07.2019)
Published in Proceedings of the National Academy of Sciences - PNAS (09.07.2019)
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Journal Article
From primordial clocks to circadian oscillators
Pitsawong, Warintra, Pádua, Ricardo A P, Grant, Timothy, Hoemberger, Marc, Otten, Renee, Bradshaw, Niels, Grigorieff, Nikolaus, Kern, Dorothee
Published in Nature (London) (06.04.2023)
Published in Nature (London) (06.04.2023)
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Journal Article
Optimization of a novel piperazinone series as potent selective peripheral covalent BTK inhibitors
Ma, Bin, Metrick, Claire M., Gu, Chungang, Hoemberger, Marc, Bajrami, Bekim, Bame, Eris, Huang, Jiansheng, Mingueneau, Michael, Murugan, Paramasivam, Santoro, Joseph C., Tang, Hao, Wang, Ti, Hopkins, Brian T.
Published in Bioorganic & medicinal chemistry letters (15.03.2022)
Published in Bioorganic & medicinal chemistry letters (15.03.2022)
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Journal Article
Discovery and Preclinical Characterization of BIIB091, a Reversible, Selective BTK Inhibitor for the Treatment of Multiple Sclerosis
Hopkins, Brian T, Bame, Eris, Bajrami, Bekim, Black, Cheryl, Bohnert, Tonika, Boiselle, Carrie, Burdette, Doug, Burns, Jeremy C, Delva, Luisette, Donaldson, Douglas, Grater, Richard, Gu, Chungang, Hoemberger, Marc, Johnson, Josh, Kapadnis, Sudarshan, King, Kris, Lulla, Mukesh, Ma, Bin, Marx, Isaac, Magee, Tom, Meissner, Robert, Metrick, Claire M, Mingueneau, Michael, Murugan, Paramasivam, Otipoby, Kevin L, Polack, Evelyne, Poreci, Urjana, Prince, Robin, Roach, Allie M, Rowbottom, Chris, Santoro, Joseph C, Schroeder, Patricia, Tang, Hao, Tien, Eric, Zhang, Fengmei, Lyssikatos, Joseph
Published in Journal of medicinal chemistry (27.01.2022)
Published in Journal of medicinal chemistry (27.01.2022)
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Journal Article
Corrigendum to “Optimization of a novel piperazinone series as potent selective peripheral covalent BTK inhibitors” [Bioorg. Med. Chem. Lett. 60 (2022) 128549]
Ma, Bin, Metrick, Claire M., Gu, Chungang, Hoemberger, Marc, Bajrami, Bekim, Bame, Eris, Huang, Jiansheng, Mingueneau, Michael, Murugan, Paramasivam, Nevalainen, Marta, Santoro, Joseph C., Tang, Hao, Wang, Ti, Hopkins, Brian T.
Published in Bioorganic & medicinal chemistry letters (15.09.2022)
Published in Bioorganic & medicinal chemistry letters (15.09.2022)
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Journal Article
Discovery and Preclinical Characterization of BIIB129, a Covalent, Selective, and Brain-Penetrant BTK Inhibitor for the Treatment of Multiple Sclerosis
Himmelbauer, Martin K., Bajrami, Bekim, Basile, Rebecca, Capacci, Andrew, Chen, TeYu, Choi, Colin K., Gilfillan, Rab, Gonzalez-Lopez de Turiso, Felix, Gu, Chungang, Hoemberger, Marc, Johnson, Douglas S., Jones, J. Howard, Kadakia, Ekta, Kirkland, Melissa, Lin, Edward Y., Liu, Ying, Ma, Bin, Magee, Tom, Mantena, Srinivasa, Marx, Isaac E., Metrick, Claire M., Mingueneau, Michael, Murugan, Paramasivam, Muste, Cathy A., Nadella, Prasad, Nevalainen, Marta, Parker Harp, Chelsea R., Pattaropong, Vatee, Pietrasiewicz, Alicia, Prince, Robin J., Purgett, Thomas J., Santoro, Joseph C., Schulz, Jurgen, Sciabola, Simone, Tang, Hao, Vandeveer, H. George, Wang, Ti, Yousaf, Zain, Helal, Christopher J., Hopkins, Brian T.
Published in Journal of medicinal chemistry (23.05.2024)
Published in Journal of medicinal chemistry (23.05.2024)
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Journal Article
Probing an Ancient Protein's Dynamics with NMR
Hoemberger, Marc S., Wilson, Christopher G., Kern, Dorothee
Published in Biophysical journal (28.01.2014)
Published in Biophysical journal (28.01.2014)
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Journal Article
Evolutionary drivers of thermoadaptation in enzyme catalysis
Nguyen, Vy, Wilson, Christopher, Hoemberger, Marc, Stiller, John B., Agafonov, Roman V., Kutter, Steffen, English, Justin, Theobald, Douglas L., Kern, Dorothee
Published in Science (American Association for the Advancement of Science) (22.12.2016)
Published in Science (American Association for the Advancement of Science) (22.12.2016)
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Journal Article
Probing the Transition State in Enzyme Catalysis by High-Pressure NMR Dynamics
Stiller, John B, Kerns, S Jordan, Hoemberger, Marc, Cho, Young-Jin, Otten, Renee, Hagan, Michael F, Kern, Dorothee
Published in Nature catalysis (01.08.2019)
Published in Nature catalysis (01.08.2019)
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