Multi-Component Mechanism of H2 Relaxin Binding to RXFP1 through NanoBRET Kinetic Analysis
Hoare, Bradley L., Bruell, Shoni, Sethi, Ashish, Gooley, Paul R., Lew, Michael J., Hossain, Mohammed A., Inoue, Asuka, Scott, Daniel J., Bathgate, Ross A.D.
Published in iScience (25.01.2019)
Published in iScience (25.01.2019)
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Journal Article
Developing insulin-like peptide 5-based antagonists for the G protein-coupled receptor, RXFP4
Wu, Hongkang, Handley, Thomas N.G., Hoare, Bradley L., Hartono, Herodion A., Scott, Daniel J., Chalmers, David K., Bathgate, Ross A.D., Hossain, Mohammed Akhter
Published in Biochemical pharmacology (01.06.2024)
Published in Biochemical pharmacology (01.06.2024)
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Journal Article
Bi-allelic variants in INSL3 and RXFP2 cause bilateral cryptorchidism and male infertility
Dicke, Ann-Kristin, Albrethsen, Jakob, Hoare, Bradley L, Wyrwoll, Margot J, Busch, Alexander S, Fietz, Daniela, Pilatz, Adrian, Bühlmann, Clara, Juul, Anders, Kliesch, Sabine, Gromoll, Jörg, Bathgate, Ross A D, Tüttelmann, Frank, Stallmeyer, Birgit
Published in Human reproduction (Oxford) (05.07.2023)
Published in Human reproduction (Oxford) (05.07.2023)
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Journal Article
ThermoBRET: A Ligand‐Engagement Nanoscale Thermostability Assay Applied to GPCRs
Hoare, Bradley L., Tippett, David N., Kaur, Amandeep, Cullum, Sean A., Miljuš, Tamara, Koers, Eline J., Harwood, Clare R., Dijon, Nicola, Holliday, Nicholas D., Sykes, David A., Veprintsev, Dmitry B.
Published in Chembiochem : a European journal of chemical biology (15.01.2024)
Published in Chembiochem : a European journal of chemical biology (15.01.2024)
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Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe
Gazzi, Thais, Brennecke, Benjamin, Atz, Kenneth, Korn, Claudia, Sykes, David, Forn-Cuni, Gabriel, Pfaff, Patrick, Sarott, Roman C, Westphal, Matthias V, Mostinski, Yelena, Mach, Leonard, Wasinska-Kalwa, Malgorzata, Weise, Marie, Hoare, Bradley L, Milju, Tamara, Mexi, Maira, Roth, Nicolas, Koers, Eline J, Guba, Wolfgang, Alker, Andr, Rufer, Arne C, Kusznir, Eric A, Huber, Sylwia, Raposo, Catarina, Zirwes, Elisabeth A, Osterwald, Anja, Pavlovic, Anto, Moes, Svenja, Beck, Jennifer, Nettekoven, Matthias, Benito-Cuesta, Irene, Grande, Teresa, Drawnel, Faye, Widmer, Gabriella, Holzer, Daniela, van der Wel, Tom, Mandhair, Harpreet, Honer, Michael, Fingerle, Jürgen, Scheffel, Jörg, Broichhagen, Johannes, Gawrisch, Klaus, Romero, Julián, Hillard, Cecilia J, Varga, Zoltan V, van der Stelt, Mario, Pacher, Pal, Gertsch, Jürg, Ullmer, Christoph, McCormick, Peter J, Oddi, Sergio, Spaink, Herman P, Maccarrone, Mauro, Veprintsev, Dmitry B, Carreira, Erick M, Grether, Uwe, Nazaré, Marc
Published in Chemical science (Cambridge) (18.05.2022)
Published in Chemical science (Cambridge) (18.05.2022)
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Activation of Multiple G Protein Pathways to Characterize the Five Dopamine Receptor Subtypes Using Bioluminescence Technology
Mönnich, Denise, Humphrys, Laura J., Höring, Carina, Hoare, Bradley L., Forster, Lisa, Pockes, Steffen
Published in ACS pharmacology & translational science (08.03.2024)
Published in ACS pharmacology & translational science (08.03.2024)
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Journal Article
Long-Circulating Vasoactive 1,18-Octadecanedioic Acid–Terlipressin Conjugate
Berger, Or, Choi, Wonmin, Ko, Caroline H., Thompson, Matthew P., Avram, Michael J., Scott, Daniel J., Hoare, Bradley L., Cridge, Riley, Wheatley, Mark, Bathgate, Ross A. D., Batlle, Daniel, Gianneschi, Nathan C.
Published in ACS pharmacology & translational science (10.05.2024)
Published in ACS pharmacology & translational science (10.05.2024)
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