Improved Solution- and Solid-Phase Preparation of Hydroxamic Acids from Esters
Ho, Chih Y, Strobel, Eric, Ralbovsky, Janet, Galemmo, Robert A
Published in Journal of organic chemistry (10.06.2005)
Published in Journal of organic chemistry (10.06.2005)
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Journal Article
Macrocyclic BACE inhibitors: Optimization of a micromolar hit to nanomolar leads
Huang, Yifang, Strobel, Eric D., Ho, Chih Y., Reynolds, Charles H., Conway, Kelly A., Piesvaux, Jennifer A., Brenneman, Douglas E., Yohrling, George J., Moore Arnold, H., Rosenthal, Daniel, Alexander, Richard S., Tounge, Brett A., Mercken, Marc, Vandermeeren, Marc, Parker, Michael H., Reitz, Allen B., Baxter, Ellen W.
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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Roles of Conformational and Positional Adaptability in Structure-Based Design of TMC125-R165335 (Etravirine) and Related Non-nucleoside Reverse Transcriptase Inhibitors That Are Highly Potent and Effective against Wild-Type and Drug-Resistant HIV-1 Variants
Das, Kalyan, Clark, Arthur D, Lewi, Paul J, Heeres, Jan, de Jonge, Marc R, Koymans, Lucien M. H, Vinkers, H. Maarten, Daeyaert, Frederik, Ludovici, Donald W, Kukla, Michael J, De Corte, Bart, Kavash, Robert W, Ho, Chih Y, Ye, Hong, Lichtenstein, Mark. A, Andries, Koen, Pauwels, Rudi, de Béthune, Marie-Pierre, Boyer, Paul L, Clark, Patrick, Hughes, Stephen H, Janssen, Paul A. J, Arnold, Eddy
Published in Journal of medicinal chemistry (06.05.2004)
Published in Journal of medicinal chemistry (06.05.2004)
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Journal Article
Evolution of anti-HIV drug candidates. Part 3: diarylpyrimidine (DAPY) analogues
Ludovici, Donald W., De Corte, Bart L., Kukla, Michael J., Ye, Hong, Ho, Chih Y., Lichtenstein, Mark A., Kavash, Robert W., Andries, Koen, de Béthune, Marie-Pierre, Azijn, Hilde, Pauwels, Rudi, Lewi, Paul J., Heeres, Jan, Koymans, Lucien M.H., de Jonge, Marc R., Van Aken, Koen J.A., Daeyaert, Frederik F.D., Das, Kalyan, Arnold, Edward, Janssen, Paul A.J.
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
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Journal Article
(6,7-Dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenylamines: Platelet-Derived Growth Factor Receptor Tyrosine Kinase Inhibitors with Broad Antiproliferative Activity against Tumor Cells
Ho, Chih Y, Ludovici, Donald W, Maharoof, Umar S. M, Mei, Jay, Sechler, Jan L, Tuman, Robert W, Strobel, Eric D, Andraka, Laura, Yen, Hwa-Kwo, Leo, Gregory, Li, Jian, Almond, Harold, Lu, Hong, DeVine, Ann, Tominovich, Rose M, Baker, Judith, Emanuel, Stuart, Gruninger, Robert H, Middleton, Steven A, Johnson, Dana L, Galemmo, Robert A
Published in Journal of medicinal chemistry (29.12.2005)
Published in Journal of medicinal chemistry (29.12.2005)
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Synthesis and Anti-HIV-1 Activity of 4,5,6,7-Tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one (TlBO) Derivatives. 4
Ho, Winston, Kukla, Michael J, Breslin, Henry J, Ludovici, Donald W, Grous, Philip P, Diamond, Craig J, Miranda, Milton, Rodgers, James D, Ho, Chih Y
Published in Journal of medicinal chemistry (03.03.1995)
Published in Journal of medicinal chemistry (03.03.1995)
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Journal Article
Synthesis and anti-HIV-1 activity of 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one (TIBO) derivatives. 2
Kukla, Michael J, Breslin, Henry J, Diamond, Craig J, Grous, Philip P, Ho, Chih Y, Miranda, Milton, Rodgers, James D, Sherrill, Ronald G, De Clercq, Erik, Pauwels, Rudi, Andries, Koen, Moens, Luc J, Janssen, Marcel A. C, Janssen, Paul A. J
Published in Journal of medicinal chemistry (01.11.1991)
Published in Journal of medicinal chemistry (01.11.1991)
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Journal Article
Synthesis and Anti-HIV-1 Activity of 4,5,6,7-Tetrahydro-5-methylimidazo[4,5,1-jk][1,4]benzodiazepin-2(1H)-one (TIBO) Derivatives. 3
Breslin, Henry J, Kukla, Michael J, Ludovici, Donald W, Mohrbacher, Richard, Ho, Winston, Miranda, Milton, Rodgers, James D, Hitchens, T. Kevin, Leo, Gregory
Published in Journal of medicinal chemistry (01.03.1995)
Published in Journal of medicinal chemistry (01.03.1995)
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Journal Article
Indolo[2,1-c][1,4]benzodiazepines: a new class of antiallergic agents
Ho, Chih Y, Hageman, William E, Persico, Francis J
Published in Journal of medicinal chemistry (01.06.1986)
Published in Journal of medicinal chemistry (01.06.1986)
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Journal Article
Evolution of Anti-HIV Drug CandidatesPart 2: Diaryltriazine (DATA) Analogues
Ludovici, Donald W., Kavash, Robert W., Kukla, Michael J., Ho, Chih Y., Ye, Hong, De Corte, Bart L., Andries, Koen, de Béthune, Marie-Pierre, Azijn, Hilde, Pauwels, Rudi, Moereels, Henry E.L., Heeres, Jan, Koymans, Lucien M.H., de Jonge, Marc R., Van Aken, Koen J.A., Daeyaert, Frederik F.D., J. Lewi, Paul, Das, Kalyan, Arnold, Edward, Janssen, Paul A.J.
Published in Bioorganic & medicinal chemistry letters (01.09.2001)
Published in Bioorganic & medicinal chemistry letters (01.09.2001)
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Journal Article
Synthesis and anti-HIV-1 activity of 4,5,6,7-tetrahydro-5-methylimidazo [4,5,1-jk][1,4] benzodiazepin-2(1H)-one (TIBO) derivatives
Breslin, HJ, Kukla, MJ, Ludovici, D W, Mohrbacher, R, Ho, Winston, Miranda, M, Rodgers, J D, Hitchens, T K, Leo, G, Gauthier, DA, Ho, Chih Y, Scott, M K, De Clercq, E, Pauwels, R
Published in Journal of medicinal chemistry (01.01.1995)
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Published in Journal of medicinal chemistry (01.01.1995)
Journal Article
Synthesis and anti-HIV-1 activity of 4,5,6,7-tetrahydro-5-methylimidazo [4,5,1-jk][1,4] benzodiazepin 2(1H)-one (TlBO) derivatives
Ho, Winston, Kukla, MJ, Breslin, HJ, Ludovici, D W, Grous, P P, Diamond, C J, Miranda, M, Rodgers, J D, Ho, Chih Y, De Clercq, E, Pauwels, R, Andries, K, Janssen, MAC, Janssen, PAJ
Published in Journal of medicinal chemistry (01.01.1995)
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Published in Journal of medicinal chemistry (01.01.1995)
Journal Article
Improved Solution- and Solid-Phase Preparation of Hydroxamic Acids from Esters
Ho, Chih Y., Strobel, Eric, Ralbovsky, Janet, Galemmo, Robert A. Jr
Published in ChemInform (25.10.2005)
Published in ChemInform (25.10.2005)
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Journal Article