Design, synthesis, and evaluation of potent, structurally novel peroxisome proliferator-activated receptor (PPAR) δ-selective agonists
Kasuga, Jun-ichi, Nakagome, Izumi, Aoyama, Atsushi, Sako, Kumiko, Ishizawa, Michiyasu, Ogura, Michitaka, Makishima, Makoto, Hirono, Shuichi, Hashimoto, Yuichi, Miyachi, Hiroyuki
Published in Bioorganic & medicinal chemistry (01.08.2007)
Published in Bioorganic & medicinal chemistry (01.08.2007)
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Design and synthesis of a series of I--benzyl phenylpropanoic acid-type peroxisome proliferator-activated receptor (PPAR) gamma partial agonists with improved aqueous solubility
Ohashi, Masao, Oyama, Takuji, Putranto, Endy, Waku, Tsuyoshi, Nobusada, Hiromi, Kataoka, Ken, Matsuno, Kenji, Yashiro, Masakazu, Morikawa, Kosuke, Huh, Nam-ho, Miyachi, Hiroyuki
Published in Bioorganic & medicinal chemistry (01.04.2013)
Published in Bioorganic & medicinal chemistry (01.04.2013)
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LIVER X RECEPTOR (LXR) MODULATORS WITH DIBENZ[b,f]-[1,4]OXAZEPIN-11-ONE, (Z)-DIBENZ[b,f]AZOCIN-6-ONE, AND 11,12-DIHYDRODIBENZ[b,f]AZOCIN-6-ONE SKELETONS
Aoyama, Atsushi, Aoyama, Hiroshi, Makishima, Makoto, Hashimoto, Yuichi, Miyachi, Hiroyuki
Published in Heterocycles (01.09.2009)
Published in Heterocycles (01.09.2009)
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Abstract 2627: Antitumor effect in human lung cancer by a combination treatment of novel histone deacetylase inhibitors: SL142 or SL325 and retinoic acids
Fukazawa, Takuya, Han, Shaoteng, Yamatsuji, Tomoki, Mastuoka, Junji, Miyachi, Hiroyuki, Morita, Ichiro, Takaoka, Munenori, Maeda, Yutaka, Naomoto, Yoshio
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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SAR-oriented discovery of peroxisome proliferator-activated receptor pan agonist with a 4-adamantylphenyl group as a hydrophobic tail
Kasuga, Jun-ichi, Yamasaki, Daisuke, Ogura, Kiyoshi, Shimizu, Motomu, Sato, Mayumi, Makishima, Makoto, Doi, Takefumi, Hashimoto, Yuichi, Miyachi, Hiroyuki
Published in Bioorganic & medicinal chemistry (01.02.2008)
Published in Bioorganic & medicinal chemistry (01.02.2008)
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Improvement of water-solubility of biarylcarboxylic acid peroxisome proliferator-activated receptor (PPAR) d-selective partial agonists by disruption of molecular planarity/symmetry
Kasuga, Jun-Ichi, Ishikawa, Minoru, Yonehara, Mitsuhiro, Makishima, Makoto, Hashimoto, Yuichi, Miyachi, Hiroyuki
Published in Bioorganic & medicinal chemistry (15.10.2010)
Published in Bioorganic & medicinal chemistry (15.10.2010)
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Design and synthesis of substituted phenylpropanoic acid derivatives as human peroxisome proliferator-activated receptor α/δ dual agonists
Kasuga, Jun-ichi, Makishima, Makoto, Hashimoto, Yuichi, Miyachi, Hiroyuki
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Ligands with a 3,3-diphenylpentane skeleton for nuclear vitamin D and androgen receptors: Dual activities and metabolic activation
Hosoda, Shinnosuke, Tanatani, Aya, Wakabayashi, Ken-ichi, Makishima, Makoto, Imai, Keisuke, Miyachi, Hiroyuki, Nagasawa, Kazuo, Hashimoto, Yuichi
Published in Bioorganic & medicinal chemistry (15.08.2006)
Published in Bioorganic & medicinal chemistry (15.08.2006)
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Ligands with dual vitamin D3-agonistic and androgen-antagonistic activities
HOSODA, Shinnosuke, TANATANI, Aya, WAKABAYASHI, Ken-Ichi, NAKANO, Yusuke, MIYACHI, Hiroyuki, NAGASAWA, Kazuo, HASHIMOTO, Yuichi
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
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Design, synthesis, and evaluation of substituted phenylpropanoic acid derivatives as human peroxisome proliferator activated receptor activators. Discovery of potent and human peroxisome proliferator activated receptor a subtype-selective activators
Nomura, M, Tanase, T, Ide, T, Tsunoda, M, Suzuki, M, Uchiki, H, Murakami, K, Miyachi, H
Published in Journal of medicinal chemistry (14.08.2003)
Published in Journal of medicinal chemistry (14.08.2003)
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Angiogenesis inhibitors derived from thalidomide
Noguchi, Tomomi, Fujimoto, Haruka, Sano, Hiroko, Miyajima, Atsushi, Miyachi, Hiroyuki, Hashimoto, Yuichi
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
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Novel Notch-sparing y-secretase inhibitors derived from a peroxisome proliferator-activated receptor agonist library
KUROSUMI, Motonori, NISHIO, Yoshino, OSAWA, Satoko, KOBAYASHI, Hisayoshi, IWATSUBO, Takeshi, TOMITA, Taisuke, MIYACHI, Hiroyuki
Published in Bioorganic & medicinal chemistry letters (2010)
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Published in Bioorganic & medicinal chemistry letters (2010)
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Analysis of the Critical Structural Determinant(s) of Species-Selective Peroxisome Proliferator-Activated Receptor Alpha (PPARα)-Activation by Phenylpropanoic Acid-Type PPARα Agonists
Miyachi, Hiroyuki, Uchiki, Hideharu
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
Published in Bioorganic & medicinal chemistry letters (06.10.2003)
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LXR ANTAGONISTS WITH A 5-SUBSTITUTED PHENANTHRIDIN-6-ONE SKELETON: SYNTHESIS AND LXR TRANSREPRESSION ACTIVITIES OF CONFORMATIONALLY RESTRICTED CARBA-T0901317 ANALOGS
Aoyama, Atsushi, Aoyama, Hiroshi, Dodo, Kosuke, Makishima, Makoto, Hashimoto, Yuichi, Miyachi, Hiroyuki
Published in Heterocycles (2008)
Published in Heterocycles (2008)
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Ligands with dual vitamin D 3-agonistic and androgen-antagonistic activities
Hosoda, Shinnosuke, Tanatani, Aya, Wakabayashi, Ken-ichi, Nakano, Yusuke, Miyachi, Hiroyuki, Nagasawa, Kazuo, Hashimoto, Yuichi
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
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