Synthesis and Pharmacological Evaluation of 3-[(4-Oxo-4H-pyrido[3,2-e][1,3]thiazin-2-yl)(phenyl)amino]propanenitrile Derivatives as Orally Active AMPA Receptor Antagonists
Inami, Hiroshi, Shishikura, Jun-ichi, Yasunaga, Tomoyuki, Hirano, Masaaki, Kimura, Takenori, Yamashita, Hiroshi, Ohno, Kazushige, Sakamoto, Shuichi
Published in Chemical & pharmaceutical bulletin (01.07.2019)
Published in Chemical & pharmaceutical bulletin (01.07.2019)
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Therapeutic effects of interleukin-1 receptor-associated kinase 4 inhibitor AS2444697 on diabetic nephropathy in type 2 diabetic mice
Kondo, Mitsuhiro, Tahara, Atsuo, Hayashi, Kazumi, Inami, Hiroshi, Ishikawa, Takeshi, Tomura, Yuichi
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.07.2020)
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.07.2020)
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Renoprotective effects of novel interleukin-1 receptor-associated kinase 4 inhibitor AS2444697 through anti-inflammatory action in 5/6 nephrectomized rats
Kondo, Mitsuhiro, Tahara, Atsuo, Hayashi, Kazumi, Abe, Masaki, Inami, Hiroshi, Ishikawa, Takeshi, Ito, Hiroyuki, Tomura, Yuichi
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.10.2014)
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.10.2014)
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Incidence of spinal instability among patients with discogenic low back pain with different backgrounds
Takahashi, Makoto, Iwamoto, Koji, Kuzuyama, Motoki, Inami, Hiroshi, Matsumoto, Yuto, Ueda, Shinji, Miyauchi, Yukio
Published in Journal of Physical Therapy Science (01.01.2021)
Published in Journal of Physical Therapy Science (01.01.2021)
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Synthesis, structure–activity relationships, and anticonvulsant activities of 2-amino-4H-pyrido[3,2-e][1,3]thiazin-4-one derivatives as orally active AMPA receptor antagonists
Inami, Hiroshi, Shishikura, Jun-ichi, Yasunaga, Tomoyuki, Ohno, Kazushige, Yamashita, Hiroshi, Kato, Kota, Sakamoto, Shuichi
Published in Bioorganic & medicinal chemistry (15.04.2015)
Published in Bioorganic & medicinal chemistry (15.04.2015)
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Functional Characterization of YM928, a Novel Noncompetitive α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonist
Ohno, Kazushige, Tsutsumi, Rie, Matsumoto, Naoyuki, Yamashita, Hiroshi, Amada, Yoko, Shishikura, Jun-Ichi, Yatsugi, Hiroshi Inami Shin-Ichi, Okada, Masamichi, Sakamoto, Shuichi, Yamaguchi, Tokio
Published in The Journal of pharmacology and experimental therapeutics (01.07.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2003)
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Suppression of fully kindled seizure and retardation of kindling acquisition by YM928 in the rat kindling model of epilepsy
Yamashita, Hiroshi, Ohno, Kazushige, Inami, Hiroshi, Shishikura, Jun-ichi, Sakamoto, Shuichi, Okada, Masamichi, Yamaguchi, Tokio
Published in European journal of pharmacology (28.06.2004)
Published in European journal of pharmacology (28.06.2004)
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Design, synthesis, and pharmacological evaluation of N-(3-carbamoyl-1H-pyrazol-4-yl)-1,3-oxazole-4-carboxamide derivatives as interleukin-1 receptor-associated kinase 4 inhibitors with reduced potential for cytochrome P450 1A2 induction
Inami, Hiroshi, Mizutani, Tsuyoshi, Watanabe, Junko, Hayashida, Hisashi, Ito, Tomonori, Terasawa, Takeshi, Kontani, Toru, Yamagishi, Hiroaki, Usuda, Hiroyuki, Aoyama, Naohiro, Imamura, Emiko, Ishikawa, Takeshi
Published in Bioorganic & medicinal chemistry (03.05.2023)
Published in Bioorganic & medicinal chemistry (03.05.2023)
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Effect of YM928, a novel AMPA receptor antagonist, on seizures in EL mice and kainate-induced seizures in rats
Yamashita, Hiroshi, Ohno, Kazushige, Amada, Yoko, Inami, Hiroshi, Shishikura, Jun-Ichi, Sakamoto, Shuichi, Okada, Masamichi, Yamaguchi, Tokio
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.08.2004)
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.08.2004)
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Prevalence and Healing Process of Lateral Malleolus Fracture in Ankle Sprains: A Retrospective Study: 一整形外科における後方視的調査
TAKAHASHI, Makoto, IWAMOTO, Koji, MIZUKAMI, Masafumi, INAMI, Hiroshi, KUWAZURU, Manabu, MIYATA, Kenji, YAMAGUCHI, Katsuya, TAKEMOTO, Nobutoshi, IGAWA, Takeshi, MIYAUCHI, Yukio
Published in Rigaku ryoho kagaku (2018)
Published in Rigaku ryoho kagaku (2018)
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Design and synthesis of 6-fluoro-2-naphthyl derivatives as novel CCR3 antagonists with reduced CYP2D6 inhibition
Sato, Ippei, Morihira, Koichiro, Inami, Hiroshi, Kubota, Hirokazu, Morokata, Tatsuaki, Suzuki, Keiko, Iura, Yosuke, Nitta, Aiko, Imaoka, Takayuki, Takahashi, Toshiya, Takeuchi, Makoto, Ohta, Mitsuaki, Tsukamoto, Shin-ichi
Published in Bioorganic & medicinal chemistry (15.09.2008)
Published in Bioorganic & medicinal chemistry (15.09.2008)
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Synthesis, biological evaluation, and metabolic stability of acrylamide derivatives as novel CCR3 antagonists
Sato, Ippei, Morihira, Koichiro, Inami, Hiroshi, Kubota, Hirokazu, Morokata, Tatsuaki, Suzuki, Keiko, Ohno, Kazuki, Iura, Yosuke, Nitta, Aiko, Imaoka, Takayuki, Takahashi, Toshiya, Takeuchi, Makoto, Ohta, Mitsuaki, Tsukamoto, Shin-ichi
Published in Bioorganic & medicinal chemistry (15.08.2009)
Published in Bioorganic & medicinal chemistry (15.08.2009)
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Journal Article
Synthesis and structure–activity relationships of N-{1-[(6-fluoro-2-naphthyl)methyl]piperidin-4-yl}benzamide derivatives as novel CCR3 antagonists
Sato, Ippei, Morihira, Koichiro, Inami, Hiroshi, Kubota, Hirokazu, Morokata, Tatsuaki, Suzuki, Keiko, Hamada, Noritaka, Iura, Yosuke, Nitta, Aiko, Imaoka, Takayuki, Takahashi, Toshiya, Takeuchi, Makoto, Ohta, Mitsuaki, Tsukamoto, Shin-ichi
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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Corrigendum to “Synthesis and structure–activity relationships of N-{1-[(6-fluoro-2-naphthyl)methyl]piperidin-4-yl}benzamide derivatives as novel CCR3 antagonists” [Bioorg. Med. Chem. 16 (2008) 144–156]
Sato, Ippei, Morihira, Koichiro, Inami, Hiroshi, Kubota, Hirokazu, Morokata, Tatsuaki, Suzuki, Keiko, Hamada, Noritaka, Iura, Yosuke, Nitta, Aiko, Imaoka, Takayuki, Takahashi, Toshiya, Takeuchi, Makoto, Ohta, Mitsuaki, Tsukamoto, Shin-ichi
Published in Bioorganic & medicinal chemistry (15.07.2008)
Published in Bioorganic & medicinal chemistry (15.07.2008)
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