Structure and Function of HIV-1 Reverse Transcriptase: Molecular Mechanisms of Polymerization and Inhibition
Sarafianos, Stefan G., Marchand, Bruno, Das, Kalyan, Himmel, Daniel M., Parniak, Michael A., Hughes, Stephen H., Arnold, Eddy
Published in Journal of molecular biology (23.01.2009)
Published in Journal of molecular biology (23.01.2009)
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Journal Article
Identification of Alternative Binding Sites for Inhibitors of HIV-1 Ribonuclease H Through Comparative Analysis of Virtual Enrichment Studies
Felts, Anthony K, LaBarge, Krystal, Bauman, Joseph D, Patel, Dishaben V, Himmel, Daniel M, Arnold, Eddy, Parniak, Michael A, Levy, Ronald M
Published in Journal of chemical information and modeling (22.08.2011)
Published in Journal of chemical information and modeling (22.08.2011)
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Journal Article
Myosin Subfragment 1 Structures Reveal a Partially Bound Nucleotide and a Complex Salt Bridge That Helps Couple Nucleotide and Actin Binding
Risal, Dipesh, Gourinath, S., Himmel, Daniel M., Szent-Györgyi, Andrew G., Cohen, Carolyn
Published in Proceedings of the National Academy of Sciences - PNAS (15.06.2004)
Published in Proceedings of the National Academy of Sciences - PNAS (15.06.2004)
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Journal Article
Exploring structural variability in X-ray crystallographic models using protein local optimization by torsion-angle sampling
Knight, Jennifer L., Zhou, Zhiyong, Gallicchio, Emilio, Himmel, Daniel M., Friesner, Richard A., Arnold, Eddy, Levy, Ronald M.
Published in Acta crystallographica. Section D, Biological crystallography. (01.04.2008)
Published in Acta crystallographica. Section D, Biological crystallography. (01.04.2008)
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Journal Article
Structure of HIV-1 Reverse Transcriptase with the Inhibitor β-Thujaplicinol Bound at the RNase H Active Site
Himmel, Daniel M., Maegley, Karen A., Pauly, Tom A., Bauman, Joseph D., Das, Kalyan, Dharia, Chhaya, Clark, Arthur D., Ryan, Kevin, Hickey, Michael J., Love, Robert A., Hughes, Stephen H., Bergqvist, Simon, Arnold, Eddy
Published in Structure (London) (09.12.2009)
Published in Structure (London) (09.12.2009)
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Journal Article
Structure of a Dihydroxycoumarin Active-Site Inhibitor in Complex with the RNase H Domain of HIV-1 Reverse Transcriptase and Structure–Activity Analysis of Inhibitor Analogs
Himmel, Daniel M., Myshakina, Nataliya S., Ilina, Tatiana, Van Ry, Alexander, Ho, William C., Parniak, Michael A., Arnold, Eddy
Published in Journal of molecular biology (15.07.2014)
Published in Journal of molecular biology (15.07.2014)
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Journal Article
Synthesis, Activity, and Structural Analysis of Novel α-Hydroxytropolone Inhibitors of Human Immunodeficiency Virus Reverse Transcriptase-Associated Ribonuclease H
Chung, Suhman, Himmel, Daniel M, Jiang, Jian-Kang, Wojtak, Krzysztof, Bauman, Joseph D, Rausch, Jason W, Wilson, Jennifer A, Beutler, John A, Thomas, Craig J, Arnold, Eddy, Le Grice, Stuart F.J
Published in Journal of medicinal chemistry (14.07.2011)
Published in Journal of medicinal chemistry (14.07.2011)
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Journal Article
Rigor-like Structures from Muscle Myosins Reveal Key Mechanical Elements in the Transduction Pathways of This Allosteric Motor
Yang, Yuting, Gourinath, S., Kovács, Mihály, Nyitray, László, Reutzel, Robbie, Himmel, Daniel M., O'Neall-Hennessey, Elizabeth, Reshetnikova, Ludmilla, Szent-Györgyi, Andrew G., Brown, Jerry H., Cohen, Carolyn
Published in Structure (London) (01.05.2007)
Published in Structure (London) (01.05.2007)
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Journal Article
HIV-1 Reverse Transcriptase Structure with RNase H Inhibitor Dihydroxy Benzoyl Naphthyl Hydrazone Bound at a Novel Site
Himmel, Daniel M, Sarafianos, Stefan G, Dharmasena, Sanjeewa, Hossain, Mohammed M, McCoy-Simandle, Kessler, Ilina, Tatiana, Clark, Arthur D, Knight, Jennifer L, Julias, John G, Clark, Patrick K, Krogh-Jespersen, Karsten, Levy, Ronald M, Hughes, Stephen H, Parniak, Michael A, Arnold, Eddy
Published in ACS chemical biology (20.12.2006)
Published in ACS chemical biology (20.12.2006)
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Journal Article
Crystal Structures for HIV-1 Reverse Transcriptase in Complexes with Three Pyridinone Derivatives: A New Class of Non-Nucleoside Inhibitors Effective against a Broad Range of Drug-Resistant Strains
Himmel, Daniel M, Das, Kalyan, Clark, Arthur D, Hughes, Stephen H, Benjahad, Abdellah, Oumouch, Said, Guillemont, Jérôme, Coupa, Sophie, Poncelet, Alain, Csoka, Imre, Meyer, Christophe, Andries, Koen, Nguyen, Chi Hung, Grierson, David S, Arnold, Eddy
Published in Journal of medicinal chemistry (01.12.2005)
Published in Journal of medicinal chemistry (01.12.2005)
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Journal Article
Crystal Structure of Scallop Myosin S1 in the Pre-Power Stroke State to 2.6 Å Resolution: Flexibility and Function in the Head
Gourinath, S., Himmel, Daniel M., Brown, Jerry H., Reshetnikova, Ludmilla, Szent-Györgyi, Andrew G., Cohen, Carolyn
Published in Structure (London) (01.12.2003)
Published in Structure (London) (01.12.2003)
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Journal Article
Crystal engineering of HIV-1 reverse transcriptase for structure-based drug design
Bauman, Joseph D, Das, Kalyan, Ho, William C, Baweja, Mukta, Himmel, Daniel M, Clark, Arthur D. Jr, Oren, Deena A, Boyer, Paul L, Hughes, Stephen H, Shatkin, Aaron J, Arnold, Eddy
Published in Nucleic acids research (01.09.2008)
Published in Nucleic acids research (01.09.2008)
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Journal Article
4-Benzyl and 4-Benzoyl-3-dimethylaminopyridin-2(1H)-ones: In Vitro Evaluation of New C-3-Amino-Substituted and C-5,6-Alkyl-Substituted Analogues against Clinically Important HIV Mutant Strains
Benjahad, Abdellah, Croisy, Martine, Monneret, Claude, Bisagni, Emile, Mabire, Dominique, Coupa, Sophie, Poncelet, Alain, Csoka, Imre, Guillemont, Jérôme, Meyer, Christophe, Andries, Koen, Pauwels, Rudi, de Béthune, Marie-Pierre, Himmel, Daniel M, Das, Kalyan, Arnold, Eddy, Nguyen, Chi Hung, Grierson, David S
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Journal Article
Introducing Our Authors
Hang, Howard C, Warthaka, Mangalika, Worthington, Andrew, Sayut, Daniel J, Himmel, Daniel M, Sarafianos, Stefan G
Published in ACS chemical biology (15.12.2006)
Published in ACS chemical biology (15.12.2006)
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Journal Article
Structure of HIV-1 Reverse Transcriptase with the Inhibitor b-Thujaplicinol Bound at the RNase H Active Site
Himmel, Daniel M, Maegley, Karen A, Pauly, Tom A, Bauman, Joseph D, Das, Kalyan, Dharia, Chhaya, Clark, Arthur D, Ryan, Kevin, Hickey, Michael J, Love, Robert A, Hughes, Stephen H, Bergqvist, Simon, Arnold, Eddy
Published in Structure (London) (09.12.2009)
Published in Structure (London) (09.12.2009)
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Journal Article