Constraining Cyclic Peptides To Mimic Protein Structure Motifs
Hill, Timothy A., Shepherd, Nicholas E., Diness, Frederik, Fairlie, David P.
Published in Angewandte Chemie (International ed.) (24.11.2014)
Published in Angewandte Chemie (International ed.) (24.11.2014)
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Journal Article
Connecting Hydrophobic Surfaces in Cyclic Peptides Increases Membrane Permeability
Hoang, Huy N., Hill, Timothy A., Fairlie, David P.
Published in Angewandte Chemie International Edition (06.04.2021)
Published in Angewandte Chemie International Edition (06.04.2021)
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Journal Article
Improving on Nature: Making a Cyclic Heptapeptide Orally Bioavailable
Nielsen, Daniel S., Hoang, Huy N., Lohman, Rink-Jan, Hill, Timothy A., Lucke, Andrew J., Craik, David J., Edmonds, David J., Griffith, David A., Rotter, Charles J., Ruggeri, Roger B., Price, David A., Liras, Spiros, Fairlie, David P.
Published in Angewandte Chemie (International ed.) (03.11.2014)
Published in Angewandte Chemie (International ed.) (03.11.2014)
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Journal Article
Ras-Related Protein Rab5a Regulates Complement C5a Receptor Trafficking, Chemotaxis, and Chemokine Secretion in Human Macrophages
Wu, Kai-Chen, Condon, Nicholas D, Hill, Timothy A., Reid, Robert C., Fairlie, David P., Lim, Junxian
Published in Journal of innate immunity (01.01.2023)
Published in Journal of innate immunity (01.01.2023)
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Journal Article
Downsizing human, bacterial, and viral proteins to short water-stable alpha helices that maintain biological potency
Harrison, Rosemary S., Shepherd, Nicholas E., Hoang, Huy N., Ruiz-Gómez, Gloria, Hill, Timothy A., Driver, Russell W., Desai, Vishal S., Young, Paul R., Abbenante, Giovanni, Fairlie, David P., Klibanov, Alexander M.
Published in Proceedings of the National Academy of Sciences - PNAS (29.06.2010)
Published in Proceedings of the National Academy of Sciences - PNAS (29.06.2010)
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Journal Article
Inhibition of Dynamin Mediated Endocytosis by the DynolesSynthesis and Functional Activity of a Family of Indoles
Hill, Timothy A, Gordon, Christopher P, McGeachie, Andrew B, Venn-Brown, Barbara, Odell, Luke R, Chau, Ngoc, Quan, Annie, Mariana, Anna, Sakoff, Jennette A, Chircop (nee Fabbro), Megan, Robinson, Phillip J, McCluskey, Adam
Published in Journal of medicinal chemistry (25.06.2009)
Published in Journal of medicinal chemistry (25.06.2009)
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Journal Article
Wollamide Cyclic Hexapeptides Synergize with Established and New Tuberculosis Antibiotics in Targeting Mycobacterium tuberculosis
Rollo, Rachel F, Mori, Giorgia, Hill, Timothy A, Hillemann, Doris, Niemann, Stefan, Homolka, Susanne, Fairlie, David P, Blumenthal, Antje
Published in Microbiology spectrum (17.08.2023)
Published in Microbiology spectrum (17.08.2023)
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Journal Article
Truncated and helix-constrained peptides with high affinity and specificity for the cFos coiled-coil of AP-1
Rao, Tara, Ruiz-Gómez, Gloria, Hill, Timothy A, Hoang, Huy N, Fairlie, David P, Mason, Jody M
Published in PloS one (27.03.2013)
Published in PloS one (27.03.2013)
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Journal Article
Iminochromene Inhibitors of Dynamins I and II GTPase Activity and Endocytosis
Hill, Timothy A, Mariana, Anna, Gordon, Christopher P, Odell, Luke R, Robertson, Mark J, McGeachie, Andrew B, Chau, Ngoc, Daniel, James A, Gorgani, Nick N, Robinson, Phillip J, McCluskey, Adam
Published in Journal of medicinal chemistry (27.05.2010)
Published in Journal of medicinal chemistry (27.05.2010)
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Journal Article
Crystal Structures of Protein-Bound Cyclic Peptides
Malde, Alpeshkumar K, Hill, Timothy A, Iyer, Abishek, Fairlie, David P
Published in Chemical reviews (11.09.2019)
Published in Chemical reviews (11.09.2019)
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Journal Article
Novel Helix-Constrained Nociceptin Derivatives Are Potent Agonists and Antagonists of ERK Phosphorylation and Thermal Analgesia in Mice
Harrison, Rosemary S, Ruiz-Gómez, Gloria, Hill, Timothy A, Chow, Shiao Y, Shepherd, Nicholas E, Lohman, Rink-Jan, Abbenante, Giovanni, Hoang, Huy N, Fairlie, David P
Published in Journal of medicinal chemistry (09.12.2010)
Published in Journal of medicinal chemistry (09.12.2010)
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Journal Article
Norcantharidin Analogues: Synthesis, Anticancer Activity and Protein Phosphatase 1 and 2A Inhibition
Hill, Timothy A., Stewart, Scott G., Gordon, Christopher P., Ackland, Stephen P., Gilbert, Jayne, Sauer, Benjamin, Sakoff, Jennette A., McCluskey, Adam
Published in ChemMedChem (15.12.2008)
Published in ChemMedChem (15.12.2008)
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Journal Article
Comparative α-Helicity of Cyclic Pentapeptides in Water
de Araujo, Aline D., Hoang, Huy N., Kok, W. Mei, Diness, Frederik, Gupta, Praveer, Hill, Timothy A., Driver, Russell W., Price, David A., Liras, Spiros, Fairlie, David P.
Published in Angewandte Chemie (International ed.) (01.07.2014)
Published in Angewandte Chemie (International ed.) (01.07.2014)
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Journal Article
28 GHz Taylor feed network for sidelobe level reduction in 5G phased array antennas
Hill, Timothy A., Kelly, James R.
Published in Microwave and optical technology letters (01.01.2019)
Published in Microwave and optical technology letters (01.01.2019)
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Journal Article
Helical structure in cyclic peptides: effect of N-methyl amides versus esters
Wu, Chongyang, Hoang, Huy N., Hill, Timothy A., Lim, Junxian, Kok, W. Mei, Akondi, Kalyani, Liu, Ligong, Fairlie, David P.
Published in Chemical communications (Cambridge, England) (08.11.2022)
Published in Chemical communications (Cambridge, England) (08.11.2022)
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Journal Article
Modifying a Hydroxyl Patch in Glucagon-like Peptide 1 Produces Biased Agonists with Unique Signaling Profiles
Wang, Peiqi, Hill, Timothy A., Mitchell, Justin, Fitzsimmons, Rebecca L., Xu, Weijun, Loh, Zhixuan, Suen, Jacky Y., Lim, Junxian, Iyer, Abishek, Fairlie, David P.
Published in Journal of medicinal chemistry (08.09.2022)
Published in Journal of medicinal chemistry (08.09.2022)
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Journal Article
A Novel Class of Anticancer Compounds Targets the Actin Cytoskeleton in Tumor Cells
STEHN, Justine R, HAASS, Nikolas K, FATH, Thomas, HILL, Timothy A, McCLUSKEY, Adam, SCHEVZOV, Galina, PALMER, Stephen J, HARDEMAN, Edna C, WINLAW, David, REEVE, Vivienne E, DIXON, Ian, WENINGER, Wolfgang, BONELLO MELISSA DESOUZA, Teresa, CRIPE, Timothy P, GUNNING, Peter W, KOTTYAN, Gregg, TREUTLEIN, Herbert, JUN ZENG, NASCIMENTO, Paula R. B. B, SEQUEIRA, Vanessa B, BUTLER, Tanya L, ALLANSON, Munif
Published in Cancer research (Chicago, Ill.) (15.08.2013)
Published in Cancer research (Chicago, Ill.) (15.08.2013)
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