Chemical and structural studies provide a mechanistic basis for recognition of the MYC G-quadruplex
Calabrese, David R, Chen, Xiang, Leon, Elena C, Gaikwad, Snehal M, Phyo, Zaw, Hewitt, William M, Alden, Stephanie, Hilimire, Thomas A, He, Fahu, Michalowski, Aleksandra M, Simmons, John K, Saunders, Lindsey B, Zhang, Shuling, Connors, Daniel, Walters, Kylie J, Mock, Beverly A, Schneekloth, Jr, John S
Published in Nature communications (12.10.2018)
Published in Nature communications (12.10.2018)
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Journal Article
Targeting the Oncogenic Long Non-coding RNA SLNCR1 by Blocking Its Sequence-Specific Binding to the Androgen Receptor
Schmidt, Karyn, Weidmann, Chase A., Hilimire, Thomas A., Yee, Elaine, Hatfield, Breanne M., Schneekloth, John S., Weeks, Kevin M., Novina, Carl D.
Published in Cell reports (Cambridge) (14.01.2020)
Published in Cell reports (Cambridge) (14.01.2020)
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Journal Article
Peptides Derived from the Tight Junction Protein CLDN1 Disrupt the Skin Barrier and Promote Responsiveness to an Epicutaneous Vaccine
Brewer, Matthew G., Anderson, Elizabeth A., Pandya, Radha P., De Benedetto, Anna, Yoshida, Takeshi, Hilimire, Thomas A., Martinez-Sobrido, Luis, Beck, Lisa A., Miller, Benjamin L.
Published in Journal of investigative dermatology (01.02.2020)
Published in Journal of investigative dermatology (01.02.2020)
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Journal Article
Increasing the Safety Profile of the Master Donor Live Attenuated Influenza Vaccine
Hilimire, Thomas A, Nogales, Aitor, Chiem, Kevin, Ortego, Javier, Martinez-Sobrido, Luis
Published in Pathogens (Basel) (29.01.2020)
Published in Pathogens (Basel) (29.01.2020)
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Correction for Piepenbrink et al., "Highly Cross-Reactive and Protective Influenza A Virus H3N2 Hemagglutinin- and Neuraminidase-Specific Human Monoclonal Antibodies"
Piepenbrink, Michael, Oladunni, Fatai, Nogales, Aitor, Khalil, Ahmed M, Fitzgerald, Theresa, Hilimire, Thomas A, Basu, Madhubanti, Fucile, Christopher, Topham, David J, Rosenberg, Alexander F, Martinez-Sobrido, Luis, Kobie, James J
Published in Microbiology spectrum (05.03.2024)
Published in Microbiology spectrum (05.03.2024)
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Journal Article
Measuring RNA–Ligand Interactions with Microscale Thermophoresis
Moon, Michelle H, Hilimire, Thomas A, Sanders, Allix M, Schneekloth, John S
Published in Biochemistry (Easton) (07.08.2018)
Published in Biochemistry (Easton) (07.08.2018)
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Journal Article
Small molecule microarray identifies inhibitors of tyrosyl-DNA phosphodiesterase 1 that simultaneously access the catalytic pocket and two substrate binding sites
Zhao, Xue Zhi, Kiselev, Evgeny, Lountos, George T, Wang, Wenjie, Tropea, Joseph E, Needle, Danielle, Hilimire, Thomas A, Schneekloth, John S, Waugh, David S, Pommier, Yves, Burke, Terrence R
Published in Chemical science (Cambridge) (28.01.2021)
Published in Chemical science (Cambridge) (28.01.2021)
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Journal Article
Mediator kinase inhibition reverses castration resistance of advanced prostate cancer
Li, Jing, Hilimire, Thomas A, Liu, Yueying, Wang, Lili, Liang, Jiaxin, Gyorffy, Balazs, Sikirzhytski, Vitali, Ji, Hao, Zhang, Li, Cheng, Chen, Ding, Xiaokai, Kerr, Kendall R, Dowling, Charles E, Chumanevich, Alexander A, Mack, Zachary T, Schools, Gary P, Lim, Chang-Uk, Ellis, Leigh, Zi, Xiaolin, Porter, Donald C, Broude, Eugenia V, McInnes, Campbell, Wilding, George, Lilly, Michael B, Roninson, Igor B, Chen, Mengqian
Published in The Journal of clinical investigation (15.05.2024)
Published in The Journal of clinical investigation (15.05.2024)
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Journal Article
Enhancing the ligand efficiency of anti-HIV compounds targeting frameshift-stimulating RNA
Anokhina, Viktoriya S., McAnany, John D., Ciesla, Jessica H., Hilimire, Thomas A., Santoso, Netty, Miao, Hongyu, Miller, Benjamin L.
Published in Bioorganic & medicinal chemistry (01.07.2019)
Published in Bioorganic & medicinal chemistry (01.07.2019)
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Journal Article
High-Affinity Recognition of HIV‑1 Frameshift-Stimulating RNA Alters Frameshifting in Vitro and Interferes with HIV‑1 Infectivity
Ofori, Leslie O, Hilimire, Thomas A, Bennett, Ryan P, Brown, Nathaniel W, Smith, Harold C, Miller, Benjamin L
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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Journal Article
HIV‑1 Frameshift RNA-Targeted Triazoles Inhibit Propagation of Replication-Competent and Multi-Drug-Resistant HIV in Human Cells
Hilimire, Thomas A, Chamberlain, Jeffrey M, Anokhina, Viktoriya, Bennett, Ryan P, Swart, Oliver, Myers, Jason R, Ashton, John M, Stewart, Ryan A, Featherston, Aaron L, Gates, Kathleen, Helms, Eric D, Smith, Harold C, Dewhurst, Stephen, Miller, Benjamin L
Published in ACS chemical biology (16.06.2017)
Published in ACS chemical biology (16.06.2017)
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Journal Article
N‑Methylation as a Strategy for Enhancing the Affinity and Selectivity of RNA-binding Peptides: Application to the HIV‑1 Frameshift-Stimulating RNA
Hilimire, Thomas A., Bennett, Ryan P., Stewart, Ryan A., Garcia-Miranda, Pablo, Blume, Alex, Becker, Jordan, Sherer, Nathan, Helms, Eric D., Butcher, Samuel E., Smith, Harold C., Miller, Benjamin L.
Published in ACS chemical biology (15.01.2016)
Published in ACS chemical biology (15.01.2016)
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Journal Article
Mediator kinase inhibition reverses castration resistance of advanced prostate cancer
Li, Jing, Hilimire, Thomas A, Liu, Yueying, Wang, Lili, Liang, Jiaxin, Gyorffy, Balazs, Sikirzhytski, Vitali, Ji, Hao, Zhang, Li, Cheng, Chen, Ding, Xiaokai, Kerr, Kendall R, Dowling, Charles E, Chumanevich, Alexander A, Mack, Zachary T, Schools, Gary R, Lim, Chang-uk, Ellis, Leigh, Zi, Xiaolin, Porter, Donald C, Broude, Eugenia V, McInnes, Campbell, Wilding, George, Lilly, Michael B, Roninson, Igor B, Chen, Mengqian
Published in The Journal of clinical investigation (01.05.2024)
Published in The Journal of clinical investigation (01.05.2024)
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