European Medicinal Chemistry Leaders in Industry (EMCL) – On the Status and Future of Medicinal Chemistry Research in Europe
Ali, Amjad, Bauser, Marcus, Bertrand, Sophie, Blackaby, Wesley, Boss, Christoph, Bossart, Martin, Hall, Adrian, Binch, Hayley, Czechtizky, Werngard, Gijsen, Harrie, Haning, Helmut, Hartung, Ingo V., Kilburn, Paul, Lassalle, Gilbert, Lücking, Ulrich, Mack, Jürgen, Missbach, Martin, Otsomaa, Leena, Torrens, Antoni, Wagner, Michael, Walter, Magnus, Weinstabl, Harald, Hijfte, Luc, Nussbaum, Franz
Published in ChemMedChem (03.07.2023)
Published in ChemMedChem (03.07.2023)
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Journal Article
Mechanism Selection for Regiocontrol in Base-Assisted, Palladium-Catalysed Direct CH Coupling with Halides: First Approach for Oxazole- and Thiazole-4-Carboxylates
Théveau, Laure, Verrier, Cécile, Lassalas, Pierrik, Martin, Thibaut, Dupas, Georges, Querolle, Olivier, Van Hijfte, Luc, Marsais, Francis, Hoarau, Christophe
Published in Chemistry : a European journal (16.12.2011)
Published in Chemistry : a European journal (16.12.2011)
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Journal Article
The 52nd International Conference on Medicinal Chemistry (RICT 2016) of the French Medicinal Chemistry Society (SCT) Held in Caen (Normandy)
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Journal Article
Conference Proceeding
Identification of a series of substituted 2-piperazinyl-5-pyrimidylhydroxamic acids as potent histone deacetylase inhibitors
Angibaud, Patrick, Emelen, Kristof Van, Decrane, Laurence, Brandt, Sven van, Holte, Peter ten, Pilatte, Isabelle, Roux, Bruno, Poncelet, Virginie, Speybrouck, David, Queguiner, Laurence, Gaurrand, Sandrine, Mariën, Ann, Floren, Wim, Janssen, Lut, Verdonck, Marc, Dun, Jacky van, Gompel, Jacky van, Gilissen, Ron, Mackie, Claire, Jardin, Marc Du, Peeters, Jozef, Noppe, Marc, Hijfte, Luc Van, Freyne, Eddy, Page, Martin, Janicot, Michel, Arts, Janine
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Journal Article
Bivalent Ligands for Protein Degradation in Drug Discovery
Scheepstra, Marcel, Hekking, Koen F.W., van Hijfte, Luc, Folmer, Rutger H.A.
Published in Computational and structural biotechnology journal (01.01.2019)
Published in Computational and structural biotechnology journal (01.01.2019)
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Journal Article
Diastereodivergent Addition of Allenylzincs to Aryl Glyoxylates
Hameury, Thomas, Guillemont, Jérôme, Van Hijfte, Luc, Bellosta, Véronique, Cossy, Janine
Published in Organic letters (04.06.2009)
Published in Organic letters (04.06.2009)
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Journal Article
On the use of boronates in the Petasis reaction
Jourdan, Hélène, Gouhier, Géraldine, Van Hijfte, Luc, Angibaud, Patrick, Piettre, Serge R.
Published in Tetrahedron letters (01.11.2005)
Published in Tetrahedron letters (01.11.2005)
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Journal Article
Combinatorial chemistry, automation and molecular diversity: new trends in the pharmaceutical industry
Van Hijfte, Luc, Marciniak, Gilbert, Froloff, Nicolas
Published in Journal of Chromatography B: Biomedical Sciences and Applications (02.04.1999)
Published in Journal of Chromatography B: Biomedical Sciences and Applications (02.04.1999)
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Book Review
Journal Article
Ring enlargement and ring contraction induced by DAST
Ferret, Haidy, Déchamps, Ingrid, Pardo, Domingo Gomez, Hijfte, Luc Van, Cossy, and Janine
Published in ARKIVOC (16.04.2010)
Published in ARKIVOC (16.04.2010)
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Journal Article
Web Resource
Analyses of compound libraries obtained by high-throughput parallel synthesis: strategy of quality control by high-performance liquid chromatography, mass spectrometry and nuclear magnetic resonance techniques
Duléry, Bertrand D, Verne-Mismer, Joëlle, Wolf, Evelyne, Kugel, C, Van Hijfte, Luc
Published in Journal of chromatography. B, Biomedical sciences and applications (02.04.1999)
Published in Journal of chromatography. B, Biomedical sciences and applications (02.04.1999)
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Journal Article
Intramolecular Sila-Matteson Rearrangement: A General Access to Silylated Heterocycles
François, Cyril, Boddaert, Thomas, Durandetti, Muriel, Querolle, Olivier, Van Hijfte, Luc, Meerpoel, Lieven, Angibaud, Patrick, Maddaluno, Jacques
Published in Organic letters (20.04.2012)
Published in Organic letters (20.04.2012)
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Journal Article
Interfacing Chemical Biology and Drug Discovery: Report from the 50th International Conference on Medicinal Chemistry of the SCT (French Medicinal Chemistry Society), July 2–4, 2014, Rouen, France
Sapi, Janos, Schmidt, Frédéric, Van Hijfte, Luc, George, Pascal
Published in ACS chemical biology (19.12.2014)
Published in ACS chemical biology (19.12.2014)
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Journal Article
Conference Proceeding
Intramolecular 1,3-diyl trapping reactions. Total synthesis of (.+-.)-hypnophilin and (.+-.)-coriolin. Formation of the trans-fused bicyclo[3.3.0]octane ring system
Van Hijfte, Luc, Little, R. Daniel, Petersen, Jeffrey L, Moeller, Kevin D
Published in Journal of organic chemistry (01.10.1987)
Published in Journal of organic chemistry (01.10.1987)
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Journal Article
Studies on pyrrolidinones. synthesis of fused 1,5-naphthyridines
Akué-Gédu, Rufine, Couturier, Daniel, Hénichart, Jean-Pierre, Rigo, Benoît, Sanz, Gerard, Van Hijfte, Luc, Bourry, Anne
Published in Tetrahedron (08.07.2012)
Published in Tetrahedron (08.07.2012)
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Journal Article
Corrigendum: Mechanism Selection for Regiocontrol in Base-Assisted, Palladium-Catalysed Direct CH Coupling with Halides: First Approach for Oxazole- and Thiazole-4-Carboxylates
Théveau, Laure, Verrier, Cécile, Lassalas, Pierrik, Martin, Thibaut, Dupas, Georges, Querolle, Olivier, Van Hijfte, Luc, Marsais, Francis, Hoarau, Christophe
Published in Chemistry : a European journal (13.02.2012)
Published in Chemistry : a European journal (13.02.2012)
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Journal Article