Extracellular loops 2 and 3 of the calcitonin receptor selectively modify agonist binding and efficacy
Dal Maso, Emma, Zhu, Yue, Pham, Vi, Reynolds, Christopher A., Deganutti, Giuseppe, Hick, Caroline A., Yang, Dehua, Christopoulos, Arthur, Hay, Debbie L., Wang, Ming-Wei, Sexton, Patrick M., Furness, Sebastian G.B., Wootten, Denise
Published in Biochemical pharmacology (01.04.2018)
Published in Biochemical pharmacology (01.04.2018)
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The Molecular Control of Calcitonin Receptor Signaling
dal Maso, Emma, Glukhova, Alisa, Zhu, Yue, Garcia-Nafria, Javier, Tate, Christopher G, Atanasio, Silvia, Reynolds, Christopher A, Ramírez-Aportela, Erney, Carazo, Jose-Maria, Hick, Caroline A, Furness, Sebastian G. B, Hay, Debbie L, Liang, Yi-Lynn, Miller, Laurence J, Christopoulos, Arthur, Wang, Ming-Wei, Wootten, Denise, Sexton, Patrick M
Published in ACS pharmacology & translational science (08.02.2019)
Published in ACS pharmacology & translational science (08.02.2019)
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Deconvoluting the Molecular Control of Binding and Signaling at the Amylin 3 Receptor: RAMP3 Alters Signal Propagation through Extracellular Loops of the Calcitonin Receptor
Pham, Vi, Zhu, Yue, Dal Maso, Emma, Reynolds, Christopher A, Deganutti, Giuseppe, Atanasio, Silvia, Hick, Caroline A, Yang, Dehua, Christopoulos, Arthur, Hay, Debbie L, Furness, Sebastian G. B, Wang, Ming-Wei, Wootten, Denise, Sexton, Patrick M
Published in ACS pharmacology & translational science (14.06.2019)
Published in ACS pharmacology & translational science (14.06.2019)
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Development of a Novel Assay for Direct Assessment of Selective Amylin Receptor Activation Reveals Novel Differences in Behavior of Selective and Nonselective Peptide Agonists
Keov, Peter, Christopoulos, George, Hick, Caroline A, Glendorf, Tine, Ballarín-González, Borja, Wootten, Denise, Sexton, Patrick M
Published in Molecular pharmacology (01.05.2024)
Published in Molecular pharmacology (01.05.2024)
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AM833 Is a Novel Agonist of Calcitonin Family G Protein-Coupled Receptors: Pharmacological Comparison with Six Selective and Nonselective Agonists
Fletcher, Madeleine M, Keov, Peter, Truong, Tin T, Mennen, Grace, Hick, Caroline A, Zhao, Peishen, Furness, Sebastian G B, Kruse, Thomas, Clausen, Trine R, Wootten, Denise, Sexton, Patrick M
Published in The Journal of pharmacology and experimental therapeutics (01.06.2021)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2021)
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Identification of novel antivirals inhibiting recognition of Venezuelan equine encephalitis virus capsid protein by the Importin α/β1 heterodimer through high-throughput screening
Thomas, David R., Lundberg, Lindsay, Pinkham, Chelsea, Shechter, Sharon, DeBono, Aaron, Baell, Jonathan, Wagstaff, Kylie M., Hick, Caroline A., Kehn-Hall, Kylene, Jans, David A.
Published in Antiviral research (01.03.2018)
Published in Antiviral research (01.03.2018)
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