A-85380 [3-(2( S)-azetidinylmethoxy) pyridine]: In Vitro pharmacological properties of a novel, high affinity α4β2 nicotinic acetylcholine receptor ligand
Sullivan, James P., Donnelly-Roberts, Diana, Briggs, Clark A., Anderson, David J., Gopalakrishnan, Murali, Piattoni-Kaplan, Marietta, Campbell, Jeffrey E., McKenna, David G., Molinari, Edwardo, Hettinger, Ann-Marie, Garvey, David S., Wasicak, James T., Holladay, Mark W., Williams, Michael, Arneric, Stephen P.
Published in Neuropharmacology (01.06.1996)
Published in Neuropharmacology (01.06.1996)
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Conference Proceeding
Novel 3-Pyridyl Ethers with Subnanomolar Affinity for Central Neuronal Nicotinic Acetylcholine Receptors
Abreo, Melwyn A, Lin, Nan-Horng, Garvey, David S, Gunn, David E, Hettinger, Ann-Marie, Wasicak, James T, Pavlik, Patricia A, Martin, Yvonne C, Donnelly-Roberts, Diana L, Anderson, David J, Sullivan, James P, Williams, Michael, Arneric, Stephen P, Holladay, Mark W
Published in Journal of medicinal chemistry (16.02.1996)
Published in Journal of medicinal chemistry (16.02.1996)
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Ligands for Brain Cholinergic Channel Receptors: Synthesis and in Vitro Characterization of Novel Isoxazoles and Isothiazoles as Bioisosteric Replacements for the Pyridine Ring in Nicotine
Garvey, David S, Wasicak, James T, Elliott, Richard L, Lebold, Suzanne, Hettinger, Ann-Marie, Carrera, George M, Lin, Nan-Horng, He, Yun, Holladay, Mark W
Published in Journal of medicinal chemistry (01.12.1994)
Published in Journal of medicinal chemistry (01.12.1994)
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Structure-activity studies on a novel series of cholinergic channel activators based on a heteroaryl ether framework
Lin, Nan-Horng, Abreo, Melwyn A., Gunn, David E., Lebold, Suzanne A., Lee, Edmund L., Wasicak, James T., Hettinger, Ann-Marie, Daanen, Jerome F., Garvey, David S., Campbell, Jeffrey E., Sullivan, James P., Williams, Michael, Arneric, Stephen P.
Published in Bioorganic & medicinal chemistry letters (20.09.1999)
Published in Bioorganic & medicinal chemistry letters (20.09.1999)
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