2-(Thienothiazolylimino)-1,3-thiazolidin-4-ones inhibit cell division cycle 25 A phosphatase
Huber-Villaume, Sophie, Revelant, Germain, Sibille, Estelle, Philippot, Stéphanie, Morabito, Angelica, Dunand, Sandrine, Chaimbault, Patrick, Bagrel, Denyse, Kirsch, Gilbert, Hesse, Stéphanie, Schohn, Hervé
Published in Bioorganic & medicinal chemistry (01.07.2016)
Published in Bioorganic & medicinal chemistry (01.07.2016)
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Direct Metalation of Heteroaromatic Esters and Nitriles Using a Mixed Lithium−Cadmium Base. Subsequent Conversion to Dipyridopyrimidinones
Bentabed-Ababsa, Ghenia, Cheikh Sid Ely, Sidaty, Hesse, Stéphanie, Nassar, Ekhlass, Chevallier, Floris, Nguyen, Tan Tai, Derdour, Aïcha, Mongin, Florence
Published in Journal of organic chemistry (05.02.2010)
Published in Journal of organic chemistry (05.02.2010)
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One-pot synthesis of new 2,4,5-trisubstituted 1,3-thiazoles and 1,3-selenazoles
Thomae, David, Perspicace, Enrico, Xu, Zhanjie, Henryon, Dorothée, Schneider, Serge, Hesse, Stéphanie, Kirsch, Gilbert, Seck, Pierre
Published in Tetrahedron (11.04.2009)
Published in Tetrahedron (11.04.2009)
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Direct metallation of thienopyrimidines using a mixed lithium-cadmium base and antitumor activity of functionalized derivatives
Snegaroff, Katia, Lassagne, Frederic, Bentabed-Ababsa, Ghenia, Nassar, Ekhlass, Ely, Sidaty Cheikh Sid, Hesse, Stephanie, Perspicace, Enrico, Derdour, Aicha, Mongin, Florence
Published in Organic & biomolecular chemistry (01.01.2009)
Published in Organic & biomolecular chemistry (01.01.2009)
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Synthesis and biological evaluation of novel 2-heteroarylimino-1,3-thiazolidin-4-ones as potential anti-tumor agents
Revelant, Germain, Huber-Villaume, Sophie, Dunand, Sandrine, Kirsch, Gilbert, Schohn, Hervé, Hesse, Stéphanie
Published in European journal of medicinal chemistry (13.04.2015)
Published in European journal of medicinal chemistry (13.04.2015)
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Microwave-Assisted Synthesis of 5-Substituted 2-Aminothiophenes Starting from Arylacetaldehydes
Revelant, Germain, Dunand, Sandrine, Hesse, Stephanie, Kirsch, Gilbert
Published in Synthesis (Stuttgart) (01.09.2011)
Published in Synthesis (Stuttgart) (01.09.2011)
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Journal Article
Synthesis and biological evaluation of di-aryl urea derivatives as c-Kit inhibitors
Ravez, Séverine, Arsenlis, Stéphane, Barczyk, Amélie, Dupont, Anthony, Frédérick, Raphaël, Hesse, Stéphanie, Kirsch, Gilbert, Depreux, Patrick, Goossens, Laurence
Published in Bioorganic & medicinal chemistry (15.11.2015)
Published in Bioorganic & medicinal chemistry (15.11.2015)
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Journal Article
Synthesis and Properties of New Multiple TCNE Adducts from Dialkynyl‐N‐(het)arylpyrroles
Pierrat, Philippe, Cebrián, Cristina, Beley, Marc, Gros, Philippe C., Torres‐Moya, Iván, Prieto, Pilar, Hesse, Stéphanie
Published in European journal of organic chemistry (23.07.2019)
Published in European journal of organic chemistry (23.07.2019)
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Journal Article
Synthesis of substituted [1,3]thiazolo[4,5- b]pyridines and [1,3]thiazolo[4,5- d][1,2,3]triazines
Thomae, David, Perspicace, Enrico, Hesse, Stéphanie, Kirsch, Gilbert, Seck, Pierre
Published in Tetrahedron (22.09.2008)
Published in Tetrahedron (22.09.2008)
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Journal Article
Design, synthesis and biological evaluation of new classes of thieno[3,2-d]pyrimidinone and thieno[1,2,3]triazine as inhibitor of vascular endothelial growth factor receptor-2 (VEGFR-2)
Perspicace, Enrico, Jouan-Hureaux, Valérie, Ragno, Rino, Ballante, Flavio, Sartini, Stefania, La Motta, Concettina, Da Settimo, Federico, Chen, Binbin, Kirsch, Gilbert, Schneider, Serge, Faivre, Béatrice, Hesse, Stéphanie
Published in European journal of medicinal chemistry (01.05.2013)
Published in European journal of medicinal chemistry (01.05.2013)
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Journal Article
One-pot synthesis of new tetrasubstituted thiophenes and selenophenes
Thomae, David, Perspicace, Enrico, Henryon, Dorothée, Xu, Zhanjie, Schneider, Serge, Hesse, Stéphanie, Kirsch, Gilbert, Seck, Pierre
Published in Tetrahedron (12.12.2009)
Published in Tetrahedron (12.12.2009)
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Vascular endothelial growth factor receptor-2 (VEGFR-2) inhibitors: development and validation of predictive 3-D QSAR models through extensive ligand- and structure-based approaches
Ragno, Rino, Ballante, Flavio, Pirolli, Adele, Wickersham, Richard B., Patsilinakos, Alexandros, Hesse, Stéphanie, Perspicace, Enrico, Kirsch, Gilbert
Published in Journal of computer-aided molecular design (01.08.2015)
Published in Journal of computer-aided molecular design (01.08.2015)
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Nanoparticles on the Basis of Highly Functionalized Dextrans
Liebert, Tim, Hornig, Stephanie, Hesse, Stephanie, Heinze, Thomas
Published in Journal of the American Chemical Society (03.08.2005)
Published in Journal of the American Chemical Society (03.08.2005)
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Journal Article
Synthesis of Novel N-Substituted 2-(Hetero)arylimino-1,3-thiazolidin-4-ones
Revelant, Germain, Hesse, Stephanie, Kirsch, Gilbert
Published in Synthesis (Stuttgart) (01.10.2010)
Published in Synthesis (Stuttgart) (01.10.2010)
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