Abstract 4332: Discovery of BAY 1163877 - A pan-FGFR inhibitor: De novo structure-based design and lead optimization of benzothiophenyl-pyrrolotriazines
Collin, Marie-Pierre L., Lobell, Mario, Huebsch, Walter, Brohm, Dirk, Héroult, Mélanie, Lustig, Klemens, Gruenewald, Sylvia, Boemer, Ulf, Jautelat, Rolf, Hess-Stump, Holger, Jaroch, Stefan, Brands, Michael, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
VEGFR-2 AND VEGFR-3 INHIBITORY ANTHRANILAMIDE PYRIDINES
KRUEGER, MARTIN, HABEREY, MARTIN, HESS-STUMP, HOLGER, THIERAUCH, KARL-HEINZ, INCE, STUART, MENRAD, ANDREAS, HUTH, ANDREAS, ZORN, LUDWIG
Year of Publication 24.05.2011
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Year of Publication 24.05.2011
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VEGFR-2 AND VEGFR-3 INHIBITORY ANTHRANYLAMIDE PYRIDINE
HABEREY MARTIN, HUTH ANDREAS, ZORN LUDWIG, THIERAUCH KARL-HEINZ, KRUEGER MARTIN, INCE STUART, HESS-STUMP HOLGER, MENRAD ANDREAS
Year of Publication 10.02.2011
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Year of Publication 10.02.2011
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VEGFR-2 AND VEGFR-3 INHIBITORY ANTHRANYLAMIDOPYRIDINES, INTERMEDIATE (VARIANTS)
HABEREY MARTIN, HUTH ANDREAS, ZORN LUDWIG, KRUEGER MARTIN, INCE STUART, HESS-STUMP HOLGER, MENRAD ANDREAS
Year of Publication 10.04.2008
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Year of Publication 10.04.2008
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VEGFR-2 and VEGFR-3 inhibitory anthranylamidopy-ridines
HABEREY, MARTIN, KRUEGER, MARTIN, HESS-STUMP, HOLGER, THIERAUCH, KARL-HEINZ, INCE, STUART, MENRAD, ANDREAS, HUTH, ANDREAS, ZORN, LUDWIG
Year of Publication 30.09.2009
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Year of Publication 30.09.2009
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Thiozolidinones production and use thereof as medicaments
HESS-STUMP, HOLGER, SIEMEISTER, GERHARD, BRIEM, HANS, EBERSPAECHER, UWE, SCHNEIDER, HERBERT, WORTMANN, LARS, ELS, KNUT, SCHWEDE, WOLFGANG, SCHULZE, VOLKER
Year of Publication 30.09.2009
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Year of Publication 30.09.2009
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PHARMACEUTICAL USE OF FIBULIN-1
HESS-STUMP, HOLGER, HAENDLER, BERNARD, CHWALISZ, KRISTOF, LESSEY, BRUCE
Year of Publication 16.04.2003
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Year of Publication 16.04.2003
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PHARMACEUTICAL USE OF FIBULIN-1
HESS-STUMP, HOLGER, HAENDLER, BERNARD, CHWALISZ, KRISTOF, LESSEY, BRUCE
Year of Publication 23.01.2003
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Year of Publication 23.01.2003
Patent
Tetrahydrocarbazol derivatives as ligands for G-protein-coupled receptors (GPCR)
KOPPITZ MARCUS KARL, PAULINI KLAUS, HESS-STUMP HOLGER, MUHN HANS PETER, SHAW KENNETH JAY
Year of Publication 17.10.2006
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Year of Publication 17.10.2006
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Tetrahydrocarbazol derivatives as ligands for G-protein-coupled receptors (GPCR)
Koppitz, Marcus Karl, Muhn, Hans Peter, Shaw, Kenneth Jay, Hess-Stump, Holger, Paulini, Klaus
Year of Publication 17.10.2006
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Year of Publication 17.10.2006
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VEGFR-2 AND VEGFR-3 INHIBITORY ANTHRANYLAMIDOPYRYDINES
HABEREY MARTIN, HUTH ANDREAS, ZORN LUDWIG, THIERAUCH KARL-HEINZ, HESS-STUMP HOLGER, INCE STUART, KRUGER MARTIN, MENRAD ANDREAS
Year of Publication 21.09.2007
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Year of Publication 21.09.2007
Patent
PHARMACEUTICAL USE OF FIBULIN-1
HESS-STUMP, HOLGER, HAENDLER, BERNARD, CHWALISZ, KRISTOF, LESSEY, BRUCE
Year of Publication 29.11.2001
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Year of Publication 29.11.2001
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TETRAHYDROCARBOZOLE DERIVATIVES AS LIGANDS FOR G-PROTEIN COUPLED RECEPTORS (GPCR)
KLAUS PAULINI, HANS-PETER MUHN, MARCUS KOPPITZ, KEN SHAW, HOLGER HESS-STUMP
Year of Publication 30.06.2005
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Year of Publication 30.06.2005
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VEGFR-2 and VEGFR-3 inhibitory anthranylamidopyridines for the treatment of diseases caused by persistent angiogenesis
KRUGER, MARTIN, HABEREY, MARTIN, HESS-STUMP, HOLGER, THIERAUCH, KARL-HEINZ, INCE, STUART, MENRAD, ANDREAS, HUTH, ANDREAS, ZORN, LUDWIG
Year of Publication 23.02.2007
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Year of Publication 23.02.2007
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VEGFR-2 AND VEGFR-3 INHIBITORY ANTHRANYLAMIDOPYRIDINES
KRUEGER, MARTIN, HABEREY, MARTIN, HESS-STUMP, HOLGER, THIERAUCH, KARL-HEINZ, INCE, STUART, MENRAD, ANDREAS, HUTH, ANDREAS, ZORN, LUDWIG
Year of Publication 16.11.2005
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Year of Publication 16.11.2005
Patent
VEGFR-2 AND VEGFR-3 INHIBITORY ANTHRANYLAMIDOPYRIDINES
HABEREY MARTIN, HUTH ANDREAS, ZORN LUDWIG, THIERAUCH KARL-HEINZ, KRUEGER MARTIN, INCE STUART, HESS-STUMP HOLGER, MENRAD ANDREAS
Year of Publication 31.10.2005
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Year of Publication 31.10.2005
Patent
VEGFR-2 AND VEGFR-3 INHIBITORY ANTHRANYLAMIDOPYRIDINES
MARTIN KRUEGER, STUART INCE, KARL-HEINZ THIERAUCH, MARTIN HABEREY, ANDREAS HUTH, HOLGER HESS-STUMP, LUDWIG ZORN, ANDREAS MENRAD
Year of Publication 31.10.2005
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Year of Publication 31.10.2005
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