Non-Amidine-Containing 1,2-Dibenzamidobenzene Inhibitors of Human Factor Xa with Potent Anticoagulant and Antithrombotic Activity
Masters, John J, Franciskovich, Jeffry B, Tinsley, Jennifer M, Campbell, Charles, Campbell, Jack B, Craft, Trelia J, Froelich, Larry L, Gifford-Moore, Donetta S, Hay, Lynne A, Herron, David K, Klimkowski, Valentine J, Kurz, Kenneth D, Metz, James T, Ratz, Andrew M, Shuman, Robert T, Smith, Gerald F, Smith, Tommy, Towner, Richard D, Wiley, Michael R, Wilson, Alex, Yee, Ying K
Published in Journal of medicinal chemistry (01.06.2000)
Published in Journal of medicinal chemistry (01.06.2000)
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Flow cytometric evaluation of the effects of leukotriene B4 receptor antagonists (LY255283 and SC-41930) on calcium mobilization and integrin expression of activated human neutrophils
MARDER, P, SCHULTZ, R. M, SPAETHE, S. M, SOFIA, M. J, HERRON, D. K
Published in Prostaglandins, leukotrienes and essential fatty acids (01.08.1992)
Published in Prostaglandins, leukotrienes and essential fatty acids (01.08.1992)
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Leukotriene B4 receptor antagonists: the LY255283 series of hydroxyacetophenones
Herron, David K, Goodson, Theodore, Bollinger, Nancy G, Swanson-Bean, Dorothy, Wright, Ian G, Staten, Gilbert S, Thompson, Alan R, Froelich, Larry L, Jackson, William T
Published in Journal of medicinal chemistry (01.05.1992)
Published in Journal of medicinal chemistry (01.05.1992)
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Leukotriene receptor on U-937 cells: discriminatory responses to leukotrienes C4 and D4
Wetmore, L A, Gerard, N P, Herron, D K, Bollinger, N G, Baker, S R, Feldman, H A, Drazen, J M
Published in The American journal of physiology (01.08.1991)
Published in The American journal of physiology (01.08.1991)
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Structure-Based Design of Potent, Amidine-Derived Inhibitors of Factor Xa: Evaluation of Selectivity, Anticoagulant Activity, and Antithrombotic Activity
Wiley, Michael R, Weir, Leonard C, Briggs, Steven, Bryan, Nancy A, Buben, John, Campbell, Charles, Chirgadze, Nickolay Y, Conrad, Richard C, Craft, Trelia J, Ficorilli, James V, Franciskovich, Jeffry B, Froelich, Larry L, Gifford-Moore, Donetta S, Goodson, Theodore, Herron, David K, Klimkowski, Valentine J, Kurz, Kenneth D, Kyle, Jeffery A, Masters, John J, Ratz, Andrew M, Milot, Guy, Shuman, Robert T, Smith, Tommy, Smith, Gerald F, Tebbe, Ann Louise, Tinsley, Jennifer M, Towner, Richard D, Wilson, Alexander, Yee, Ying K
Published in Journal of medicinal chemistry (09.03.2000)
Published in Journal of medicinal chemistry (09.03.2000)
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Effects of two leukotriene B4 (LTB4) receptor antagonists (LY255283 and SC-41930) on LTB4-induced human neutrophil adhesion and superoxide production
SCHULTZ, R. M, MARDER, P, SPAETHE, S. M, HERRON, D. K, SOFIA, M. J
Published in Prostaglandins, leukotrienes and essential fatty acids (01.08.1991)
Published in Prostaglandins, leukotrienes and essential fatty acids (01.08.1991)
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Evaluation of Antibiotic Efficacy Using Electron Microscopy: Morphological Effects of Guanylureido Cephalosporin, Chlorobenzoylureido Cephalosporin, BL-P1654, and Carbenicillin on Pseudomonas aeruginosa
Ellis, L F, Herron, D K, Preston, D A, Simmons, L K, Schlegel, R A
Published in Antimicrobial Agents and Chemotherapy (01.02.1976)
Published in Antimicrobial Agents and Chemotherapy (01.02.1976)
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Evaluation of Antibiotic Efficacy Using Electron Microscopy: Morphological Effects of Guanylureido Cephalosporin, BL-P1654, and Carbenicillin on Escherichia coli
Ellis, L F, Herron, D K, Preston, D A, Simmons, L K, Schlegel, R A
Published in Antimicrobial Agents and Chemotherapy (01.02.1976)
Published in Antimicrobial Agents and Chemotherapy (01.02.1976)
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Pulmonary actions of LY255283, a leukotriene B4 receptor antagonist
Silbaugh, S A, Stengel, P W, Cockerham, S L, Roman, C R, Saussy, Jr, D L, Spaethe, S M, Goodson, Jr, T, Herron, D K, Fleisch, J H
Published in European journal of pharmacology (13.11.1992)
Published in European journal of pharmacology (13.11.1992)
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Development of a series of phenyltetrazole leukotriene D4 (LTD4) receptor antagonists
Harper, R W, Herron, D K, Bollinger, N G, Sawyer, J S, Baldwin, R F, Roman, C R, Rinkema, L E, Fleisch, J H
Published in Journal of medicinal chemistry (03.04.1992)
Published in Journal of medicinal chemistry (03.04.1992)
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Synthesis and activity of new aryl- and heteroaryl- substituted pyrazole inhibitors of the transforming growth factor-b type I receptor kinase domain
Sawyer, JS, Anderson, BD, Beight, DW, Campbell, RM, Jones, ML, Herron, DK, Lampe, JW, McCowan, McMillen, WT, Mort, N, Parsons, S, Smith, ECR, Vieth, M, Wier, LC, Yan, L, Zhang, FM, Yingling, JM
Published in Journal of medicinal chemistry (11.09.2003)
Published in Journal of medicinal chemistry (11.09.2003)
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N(2)-Aroylanthranilamide inhibitors of human factor Xa
Yee, Y K, Tebbe, A L, Linebarger, J H, Beight, D W, Craft, T J, Gifford-Moore, D, Goodson, Jr, T, Herron, D K, Klimkowski, V J, Kyle, J A, Sawyer, J S, Smith, G F, Tinsley, J M, Towner, R D, Weir, L, Wiley, M R
Published in Journal of medicinal chemistry (09.03.2000)
Published in Journal of medicinal chemistry (09.03.2000)
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Leukotriene receptor antagonists. III. Pharmacological and chemical studies with LY137617, a leukotriene D4 and leukotriene E4 receptor antagonist
Herron, D K, Whitesitt, C A, Mallet, B E, Rinkema, L E, Haisch, K D, Fleisch, J H
Published in Drugs under experimental and clinical research (1988)
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Published in Drugs under experimental and clinical research (1988)
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Synthesis and activity of new aryl- and heteroaryl-substituted 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole inhibitors of the transforming growth factor-β type I receptor kinase domain
SAWYER, J. Scott, BEIGHT, Douglas W, PARSONS, Stephen, SMITH, Edward C. R, WAGNER, Jill R, LEI YAN, FAMING ZHANG, YINGLING, Jonathan M, BRITT, Karen S, ANDERSON, Bryan D, CAMPBELL, Robert M, GOODSON, Theodore JR, HERRON, David K, LI, Hong-Yu, MCMILLEN, William T, MORT, Nicholas
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
Published in Bioorganic & medicinal chemistry letters (05.07.2004)
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Kinetic Characterization of Novel Pyrazole TGF-β Receptor I Kinase Inhibitors and Their Blockade of the Epithelial−Mesenchymal Transition
Peng, Sheng-Bin, Yan, Lei, Xia, Xiaoling, Watkins, Scott A, Brooks, Harold B, Beight, Douglas, Herron, David K, Jones, Michael L, Lampe, John W, McMillen, William T, Mort, Nicholas, Sawyer, J. Scott, Yingling, Jonathan M
Published in Biochemistry (Easton) (22.02.2005)
Published in Biochemistry (Easton) (22.02.2005)
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