Determination of New 4-Aryl-pyrido[1,2-c]pyrimidine Derivatives, Potential Antidepressant Agents with a High Affinity to 5-Hydroxytryptamin 1A Receptor and Serotonin Transporter Protein Receptor, with Capillary Electrophoresis
Grodner, Błażej, Król, Marek, Ślifirski, Grzegorz, Ślifirski, Piotr, Herold, Franciszek
Published in Chromatographia (01.02.2024)
Published in Chromatographia (01.02.2024)
Get full text
Journal Article
The Synthesis and Absolute Configuration of Enantiomeric Pure (R)- and (S)-3-(piperidin-3-yl)-1H-Indole Derivatives
Król, Marek, Ślifirski, Grzegorz, Kleps, Jerzy, Podsadni, Piotr, Materek, Ilona, Kozioł, Anna E, Herold, Franciszek
Published in International journal of molecular sciences (28.12.2022)
Published in International journal of molecular sciences (28.12.2022)
Get full text
Journal Article
Synthesis of Novel Pyrido[1,2-c]pyrimidine Derivatives with 6-Fluoro-3-(4-piperidynyl)-1,2-benzisoxazole Moiety as Potential SSRI and 5-HT1A Receptor Ligands
Król, Marek, Ślifirski, Grzegorz, Kleps, Jerzy, Ulenberg, Szymon, Belka, Mariusz, Bączek, Tomasz, Siwek, Agata, Stachowicz, Katarzyna, Szewczyk, Bernadeta, Nowak, Gabriel, Duszyńska, Beata, Herold, Franciszek
Published in International journal of molecular sciences (01.03.2021)
Published in International journal of molecular sciences (01.03.2021)
Get full text
Journal Article
Prediction of overall in vitro microsomal stability of drug candidates based on molecular modeling and support vector machines. Case study of novel arylpiperazines derivatives
Ulenberg, Szymon, Belka, Mariusz, Król, Marek, Herold, Franciszek, Hewelt-Belka, Weronika, Kot-Wasik, Agata, Bączek, Tomasz
Published in PloS one (31.03.2015)
Published in PloS one (31.03.2015)
Get full text
Journal Article
Synthesis and anticonvulsant activity of novel 2,6-diketopiperazine derivatives. Part 1: Perhydropyrrole[1,2- a]pyrazines
Dawidowski, Maciej, Herold, Franciszek, Chodkowski, Andrzej, Kleps, Jerzy, Szulczyk, Paweł, Wilczek, Marcin
Published in European journal of medicinal chemistry (01.10.2011)
Published in European journal of medicinal chemistry (01.10.2011)
Get full text
Journal Article
Molecular Docking Supplements an In vitro Determination of the Leading CYP Isoform for Arylpiperazine Derivatives
Ulenberg, Szymon, Bączek, Tomasz, Zieliñska, Joanna, Belka, Mariusz, Król, Marek, Herold, Franciszek
Published in Combinatorial chemistry & high throughput screening (01.01.2019)
Published in Combinatorial chemistry & high throughput screening (01.01.2019)
Get more information
Journal Article
Synthesis of a new scaffold: the 7H,8H-pyrimido[1,6-b]pyridazin-6,8-dione nucleus
Herold, Franciszek, Kałucka, Małgorzata, Król, Marek, Herold, Joanna, Kleps, Jerzy, Turło, Jadwiga
Published in Molecules (Basel, Switzerland) (30.12.2007)
Published in Molecules (Basel, Switzerland) (30.12.2007)
Get full text
Journal Article
Use of biomimetic chromatography and in vitro assay to develop predictive GA-MLR model for use in drug-property prediction among anti-depressant drug candidates
Ulenberg, Szymon, Ciura, Krzesimir, Georgiev, Paweł, Pastewska, Monika, Ślifirski, Grzegorz, Król, Marek, Herold, Franciszek, Bączek, Tomasz
Published in Microchemical journal (01.04.2022)
Published in Microchemical journal (01.04.2022)
Get full text
Journal Article
Understanding performance of 3D-printed sorbent in study of metabolic stability
Ulenberg, Szymon, Georgiev, Paweł, Belka, Mariusz, Ślifirski, Grzegorz, Wróbel, Martyna, Chodkowski, Andrzej, Król, Marek, Herold, Franciszek, Bączek, Tomasz
Published in Journal of Chromatography A (11.10.2020)
Published in Journal of Chromatography A (11.10.2020)
Get full text
Journal Article
Synthesis and biological evaluation of new multi-target 3-(1H-indol-3-yl)pyrrolidine-2,5-dione derivatives with potential antidepressant effect
Wróbel, Martyna Z., Chodkowski, Andrzej, Herold, Franciszek, Marciniak, Monika, Dawidowski, Maciej, Siwek, Agata, Starowicz, Gabriela, Stachowicz, Katarzyna, Szewczyk, Bernadeta, Nowak, Gabriel, Belka, Mariusz, Bączek, Tomasz, Satała, Grzegorz, Bojarski, Andrzej J., Turło, Jadwiga
Published in European journal of medicinal chemistry (01.12.2019)
Published in European journal of medicinal chemistry (01.12.2019)
Get full text
Journal Article
The influence of phase II enzymes on in vitro half-life of pirydo[1,2-c]pirymidine derivatives as structural analogues of arylpiperazine
Ulenberg, Szymon, Belka, Mariusz, Georgiev, Paweł, Ślifirski, Grzegorz, Król, Marek, Herold, Franciszek, Bączek, Tomasz
Published in Microchemical journal (01.12.2020)
Published in Microchemical journal (01.12.2020)
Get full text
Journal Article
Synthesis of novel pyrido[1,2-c]pyrimidine derivatives with rigidized tryptamine moiety as potential SSRI and 5-HT1A receptor ligands
Ślifirski, Grzegorz, Król, Marek, Kleps, Jerzy, Ulenberg, Szymon, Belka, Mariusz, Bączek, Tomasz, Siwek, Agata, Stachowicz, Katarzyna, Szewczyk, Bernadeta, Nowak, Gabriel, Bojarski, Andrzej, Kozioł, Anna E., Turło, Jadwiga, Herold, Franciszek
Published in European journal of medicinal chemistry (15.03.2019)
Published in European journal of medicinal chemistry (15.03.2019)
Get full text
Journal Article
Synthesis of new 5,6,7,8-tetrahydropyrido[1,2-c]pyrimidine derivatives with rigidized tryptamine moiety as potential SSRI and 5-HT1A receptor ligands
Ślifirski, Grzegorz, Król, Marek, Kleps, Jerzy, Podsadni, Piotr, Belka, Mariusz, Bączek, Tomasz, Siwek, Agata, Stachowicz, Katarzyna, Szewczyk, Bernadeta, Nowak, Gabriel, Bojarski, Andrzej, Kozioł, Anna E., Turło, Jadwiga, Herold, Franciszek
Published in European journal of medicinal chemistry (15.10.2019)
Published in European journal of medicinal chemistry (15.10.2019)
Get full text
Journal Article
Improved simultaneous production of mycelial biomass and polysaccharides by submerged culture of Hericium erinaceum: optimization using a central composite rotatable design (CCRD)
Malinowska, Eliza, Krzyczkowski, Wojciech, Łapienis, Grzegorz, Herold, Franciszek
Published in Journal of industrial microbiology & biotechnology (01.12.2009)
Published in Journal of industrial microbiology & biotechnology (01.12.2009)
Get full text
Journal Article
Biosynthesis of selenium-containing polysaccharides with antioxidant activity in liquid culture of Hericium erinaceum
Malinowska, Eliza, Krzyczkowski, Wojciech, Herold, Franciszek, Łapienis, Grzegorz, Ślusarczyk, Joanna, Suchocki, Piotr, Kuraś, Mieczysław, Turło, Jadwiga
Published in Enzyme and microbial technology (06.05.2009)
Published in Enzyme and microbial technology (06.05.2009)
Get full text
Journal Article
Prediction of Overall
Ulenberg, Szymon, Belka, Mariusz, Król, Marek, Herold, Franciszek, Hewelt-Belka, Weronika, Kot-Wasik, Agata, Baczek, Tomasz
Published in PloS one (31.03.2015)
Published in PloS one (31.03.2015)
Get full text
Journal Article