Melatonin stimulates the nonamyloidogenic processing of βAPP through the positive transcriptional regulation of ADAM10 and ADAM17
Shukla, Mayuri, Htoo, Htut Htut, Wintachai, Phitchayapak, Hernandez, Jean-Francois, Dubois, Claire, Postina, Rolf, Xu, Huaxi, Checler, Frédéric, Smith, Duncan R., Govitrapong, Piyarat, Vincent, Bruno
Published in Journal of pineal research (01.03.2015)
Published in Journal of pineal research (01.03.2015)
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Synthesis and Characterization of Andrographolide Derivatives as Regulators of βAPP Processing in Human Cells
Dey, Arpita, Chen, Ran, Li, Feng, Maitra, Subhamita, Hernandez, Jean-Francois, Zhou, Guo-Chun, Vincent, Bruno
Published in Molecules (Basel, Switzerland) (17.12.2021)
Published in Molecules (Basel, Switzerland) (17.12.2021)
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4-Amino-1,2,4-triazole-3-thione-derived Schiff bases as metallo-β-lactamase inhibitors
Gavara, Laurent, Sevaille, Laurent, De Luca, Filomena, Mercuri, Paola, Bebrone, Carine, Feller, Georges, Legru, Alice, Cerboni, Giulia, Tanfoni, Silvia, Baud, Damien, Cutolo, Giuliano, Bestgen, Benoît, Chelini, Giulia, Verdirosa, Federica, Sannio, Filomena, Pozzi, Cecilia, Benvenuti, Manuela, Kwapien, Karolina, Fischer, Marina, Becker, Katja, Frère, Jean-Marie, Mangani, Stefano, Gresh, Nohad, Berthomieu, Dorothée, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-François
Published in European journal of medicinal chemistry (15.12.2020)
Published in European journal of medicinal chemistry (15.12.2020)
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4-( N -Alkyl- and -Acyl-amino)-1,2,4-triazole-3-thione Analogs as Metallo-β-Lactamase Inhibitors: Impact of 4-Linker on Potency and Spectrum of Inhibition
Gavara, Laurent, Verdirosa, Federica, Legru, Alice, Mercuri, Paola Sandra, Nauton, Lionel, Sevaille, Laurent, Feller, Georges, Berthomieu, Dorothée, Sannio, Filomena, Marcoccia, Francesca, Tanfoni, Silvia, De Luca, Filomena, Gresh, Nohad, Galleni, Moreno, Docquier, Jean-Denis, Hernandez, Jean-François
Published in Biomolecules (Basel, Switzerland) (23.07.2020)
Published in Biomolecules (Basel, Switzerland) (23.07.2020)
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Unraveling the Speciation of β‑Amyloid Peptides during the Aggregation Process by Taylor Dispersion Analysis
Deleanu, Mihai, Hernandez, Jean-François, Cipelletti, Luca, Biron, Jean-Philippe, Rossi, Emilie, Taverna, Myriam, Cottet, Hervé, Chamieh, Joseph
Published in Analytical chemistry (Washington) (27.04.2021)
Published in Analytical chemistry (Washington) (27.04.2021)
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Intermolecular interactions of the extended recognition site of VIM‐2 metallo‐β‐lactamase with 1,2,4‐triazole‐3‐thione inhibitors. Validations of a polarizable molecular mechanics potential by ab initio QC
Kwapien, Karolina, Gavara, Laurent, Docquier, Jean‐Denis, Berthomieu, Dorothée, Hernandez, Jean‐François, Gresh, Nohad
Published in Journal of computational chemistry (15.01.2021)
Published in Journal of computational chemistry (15.01.2021)
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Methamphetamine regulates βAPP processing in human neuroblastoma cells
Shukla, Mayuri, Maitra, Subhamita, Hernandez, Jean-François, Govitrapong, Piyarat, Vincent, Bruno
Published in Neuroscience letters (14.05.2019)
Published in Neuroscience letters (14.05.2019)
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Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates
Legru, Alice, Verdirosa, Federica, Vo-Hoang, Yen, Tassone, Giusy, Vascon, Filippo, Thomas, Caitlyn A., Sannio, Filomena, Corsica, Giuseppina, Benvenuti, Manuela, Feller, Georges, Coulon, Rémi, Marcoccia, Francesca, Devente, Savannah Rowane, Bouajila, Ezeddine, Piveteau, Catherine, Leroux, Florence, Deprez-Poulain, Rebecca, Deprez, Benoît, Licznar-Fajardo, Patricia, Crowder, Michael W., Cendron, Laura, Pozzi, Cecilia, Mangani, Stefano, Docquier, Jean-Denis, Hernandez, Jean-François, Gavara, Laurent
Published in Journal of medicinal chemistry (22.12.2022)
Published in Journal of medicinal chemistry (22.12.2022)
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Taylor Dispersion Analysis and Atomic Force Microscopy Provide a Quantitative Insight into the Aggregation Kinetics of Aβ (1–40)/Aβ (1–42) Amyloid Peptide Mixtures
Deleanu, Mihai, Deschaume, Olivier, Cipelletti, Luca, Hernandez, Jean-François, Bartic, Carmen, Cottet, Hervé, Chamieh, Joseph
Published in ACS chemical neuroscience (16.03.2022)
Published in ACS chemical neuroscience (16.03.2022)
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S -Ethyl-Isothiocitrullin-Based Dipeptides and 1,2,4-Oxadiazole Pseudo-Dipeptides: Solid Phase Synthesis and Evaluation as NO Synthase Inhibitors
Mauchauffée, Elodie, Leroy, Jérémy, Chamcham, Jihanne, Ejjoummany, Abdelaziz, Maurel, Manon, Nauton, Lionel, Ramassamy, Booma, Mezghenna, Karima, Boucher, Jean-Luc, Lajoix, Anne-Dominique, Hernandez, Jean-François
Published in Molecules (Basel, Switzerland) (29.06.2023)
Published in Molecules (Basel, Switzerland) (29.06.2023)
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1,2,4‐Triazole‐3‐Thione Analogues with a 2‐Ethylbenzoic Acid at Position 4 as VIM‐type Metallo‐β‐Lactamase Inhibitors
Verdirosa, Federica, Gavara, Laurent, Sevaille, Laurent, Tassone, Giusy, Corsica, Giuseppina, Legru, Alice, Feller, Georges, Chelini, Giulia, Mercuri, Paola Sandra, Tanfoni, Silvia, Sannio, Filomena, Benvenuti, Manuela, Cerboni, Giulia, De Luca, Filomena, Bouajila, Ezeddine, Vo Hoang, Yen, Licznar‐Fajardo, Patricia, Galleni, Moreno, Pozzi, Cecilia, Mangani, Stefano, Docquier, Jean‐Denis, Hernandez, Jean‐François
Published in ChemMedChem (05.04.2022)
Published in ChemMedChem (05.04.2022)
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1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity
Legru, Alice, Verdirosa, Federica, Hernandez, Jean-François, Tassone, Giusy, Sannio, Filomena, Benvenuti, Manuela, Conde, Pierre-Alexis, Bossis, Guillaume, Thomas, Caitlyn A., Crowder, Michael W., Dillenberger, Melissa, Becker, Katja, Pozzi, Cecilia, Mangani, Stefano, Docquier, Jean-Denis, Gavara, Laurent
Published in European journal of medicinal chemistry (15.12.2021)
Published in European journal of medicinal chemistry (15.12.2021)
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N‑Acyl Benzotriazole Derivatives for the Synthesis of Dipeptides and Tripeptides and Peptide Biotinylation by Mechanochemistry
Gonnet, Lori, Tintillier, Thibault, Venturini, Natacha, Konnert, Laure, Hernandez, Jean-François, Lamaty, Frédéric, Laconde, Guillaume, Martinez, Jean, Colacino, Evelina
Published in ACS sustainable chemistry & engineering (03.04.2017)
Published in ACS sustainable chemistry & engineering (03.04.2017)
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3D structures of the Plasmodium vivax subtilisin-like drug target SUB1 reveal conformational changes to accommodate a substrate-derived α-ketoamide inhibitor
Martinez, Mariano, Batista, Fernando A, Maurel, Manon, Bouillon, Anthony, Ortega Varga, Laura, Wehenkel, Anne Marie, Le Chevalier-Sontag, Lucile, Blondel, Arnaud, Haouz, Ahmed, Hernandez, Jean François, Alzari, Pedro M, Barale, Jean Christophe
Published in Acta crystallographica. Section D, Biological crystallography. (01.08.2023)
Published in Acta crystallographica. Section D, Biological crystallography. (01.08.2023)
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Insights from structure-activity relationships and the binding mode of peptidic α-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1
Legru, Alice, Batista, Fernando A., Puszko, Anna K., Bouillon, Anthony, Maurel, Manon, Martinez, Mariano, Ejjoummany, Abdelaziz, Ortega Varga, Laura, Adler, Pauline, Méchaly, Ariel, Hadjadj, Margot, Sosnowski, Piotr, Hopfgartner, Gérard, Alzari, Pedro M., Blondel, Arnaud, Haouz, Ahmed, Barale, Jean-Christophe, Hernandez, Jean-François
Published in European journal of medicinal chemistry (05.04.2024)
Published in European journal of medicinal chemistry (05.04.2024)
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The standardized Centella asiatica extract ECa 233 regulates the catalytic activities of βAPP-cleaving secretases in human cell lines
Protha, Mehbuba Nur, Srisutjarit, Therathep, Dey, Arpita, Maitra, Subhamita, Hernandez, Jean-Francois, Tantisira, Mayuree H., Boondam, Yingrak, Pakaprot, Narawut, Vincent, Bruno
Published in ScienceAsia : journal of the Science Society of Thailand (01.04.2023)
Published in ScienceAsia : journal of the Science Society of Thailand (01.04.2023)
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1,2,4‐Triazole‐3‐thione Compounds as Inhibitors of Dizinc Metallo‐β‐lactamases
Sevaille, Laurent, Gavara, Laurent, Bebrone, Carine, De Luca, Filomena, Nauton, Lionel, Achard, Maud, Mercuri, Paola, Tanfoni, Silvia, Borgianni, Luisa, Guyon, Carole, Lonjon, Pauline, Turan‐Zitouni, Gülhan, Dzieciolowski, Julia, Becker, Katja, Bénard, Lionel, Condon, Ciaran, Maillard, Ludovic, Martinez, Jean, Frère, Jean‐Marie, Dideberg, Otto, Galleni, Moreno, Docquier, Jean‐Denis, Hernandez, Jean‐François
Published in ChemMedChem (21.06.2017)
Published in ChemMedChem (21.06.2017)
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Calibration of 1,2,4-Triazole-3-Thione, an Original Zn-Binding Group of Metallo-β-Lactamase Inhibitors. Validation of a Polarizable MM/MD Potential by Quantum Chemistry
Kwapien, Karolina, Damergi, Mirna, Nader, Serge, El Khoury, Léa, Hobaika, Zeina, Maroun, Richard G, Piquemal, Jean-Philip, Gavara, Laurent, Berthomieu, Dorothée, Hernandez, Jean-François, Gresh, Nohad
Published in The journal of physical chemistry. B (06.07.2017)
Published in The journal of physical chemistry. B (06.07.2017)
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Solid‐Phase Synthesis of Substrate‐Based Dipeptides and Heterocyclic Pseudo‐dipeptides as Potential NO Synthase Inhibitors
Touati‐Jallabe, Youness, Tintillier, Thibault, Mauchauffée, Elodie, Boucher, Jean‐Luc, Leroy, Jérémy, Ramassamy, Booma, Hamzé, Abdallah, Mezghenna, Karima, Bouzekrini, Amine, Verna, Claudia, Martinez, Jean, Lajoix, Anne‐Dominique, Hernandez, Jean‐François
Published in ChemMedChem (18.03.2020)
Published in ChemMedChem (18.03.2020)
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