Discovery and SAR of Novel 2,3-Dihydroimidazo[1,2-c]quinazoline PI3K Inhibitors: Identification of Copanlisib (BAY 80-6946)
Scott, William J., Hentemann, Martin F., Rowley, R. Bruce, Bull, Cathy O., Jenkins, Susan, Bullion, Ann M., Johnson, Jeffrey, Redman, Anikó, Robbins, Arthur H., Esler, William, Fracasso, R. Paul, Garrison, Timothy, Hamilton, Mark, Michels, Martin, Wood, Jill E., Wilkie, Dean P., Xiao, Hong, Levy, Joan, Stasik, Enrico, Liu, Ningshu, Schaefer, Martina, Brands, Michael, Lefranc, Julien
Published in ChemMedChem (19.07.2016)
Published in ChemMedChem (19.07.2016)
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On the Total Synthesis and Determination of the Absolute Configuration of Rishirilide B: Exploitation of Subtle Effects to Control the Sense of Cycloaddition of o-Quinodimethides
Yamamoto, Kana, Hentemann, Martin F., Allen, John G., Danishefsky, Samuel J.
Published in Chemistry : a European journal (21.07.2003)
Published in Chemistry : a European journal (21.07.2003)
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A Powerful o-Quinone Dimethide Strategy for Intermolecular Diels−Alder Cycloadditions
Allen, John G, Hentemann, Martin F, Danishefsky, Samuel J
Published in Journal of the American Chemical Society (02.02.2000)
Published in Journal of the American Chemical Society (02.02.2000)
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Antibacterial Inhibitors of Gram-Positive Thymidylate Kinase: Structure–Activity Relationships and Chiral Preference of a New Hydrophobic Binding Region
Kawatkar, Sameer P, Keating, Thomas A, Olivier, Nelson B, Breen, John N, Green, Oluyinka M, Guler, Satenig Y, Hentemann, Martin F, Loch, James T, McKenzie, Andrew R, Newman, Joseph V, Otterson, Linda G, Martínez-Botella, Gabriel
Published in Journal of medicinal chemistry (12.06.2014)
Published in Journal of medicinal chemistry (12.06.2014)
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Discovery of Selective and Potent Inhibitors of Gram-Positive Bacterial Thymidylate Kinase (TMK)
Martínez-Botella, Gabriel, Breen, John N, Duffy, James E. S, Dumas, Jacques, Geng, Bolin, Gowers, Ian K, Green, Oluyinka M, Guler, Satenig, Hentemann, Martin F, Hernandez-Juan, Felix A, Joseph-McCarthy, Diane, Kawatkar, Sameer, Larsen, Nicholas A, Lazari, Ovadia, Loch, James T, Macritchie, Jacqueline A, McKenzie, Andrew R, Newman, Joseph V, Olivier, Nelson B, Otterson, Linda G, Owens, Andrew P, Read, Jon, Sheppard, David W, Keating, Thomas A
Published in Journal of medicinal chemistry (26.11.2012)
Published in Journal of medicinal chemistry (26.11.2012)
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In Vivo Validation of Thymidylate Kinase (TMK) with a Rationally Designed, Selective Antibacterial Compound
Keating, Thomas A, Newman, Joseph V, Olivier, Nelson B, Otterson, Linda G, Andrews, Beth, Boriack-Sjodin, P. Ann, Breen, John N, Doig, Peter, Dumas, Jacques, Gangl, Eric, Green, Oluyinka M, Guler, Satenig Y, Hentemann, Martin F, Joseph-McCarthy, Diane, Kawatkar, Sameer, Kutschke, Amy, Loch, James T, McKenzie, Andrew R, Pradeepan, Selvi, Prasad, Swati, Martínez-Botella, Gabriel
Published in ACS chemical biology (16.11.2012)
Published in ACS chemical biology (16.11.2012)
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The Origin of endo Stereoselectivity in the Hetero-Diels-Alder Reactions of Aldehydes with ortho-Xylylenes: CH-π, π-π, and Steric Effects on Stereoselectivity
Ujaque, Gregori, Lee, Patrick S., Houk, K. N., Hentemann, Martin F., Danishefsky, Samuel J.
Published in Chemistry : a European journal (02.08.2002)
Published in Chemistry : a European journal (02.08.2002)
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Concise Stereoselective Routes to Advanced Intermediates Related to Natural and Unnatural Pinnaic Acid This work was supported by the National Institutes of Health (Grant Numbers: CA28824). Postdoctoral Fellowship support is gratefully acknowledged by M.W.C. (U.S. Army BCRP, DAMD17-98-1-8154), M.F.H. (5T32 CA62948-05), and D.T. (Schering Research Foundation, Berlin). We thank Dr. George Sukenick of the MSKCC NMR Core Facility for NMR and mass spectral analyses
Carson, Matthew W., Kim, Guncheol, Hentemann, Martin F., Trauner, Dirk, Danishefsky, Samuel J.
Published in Angewandte Chemie International Edition (03.12.2001)
Published in Angewandte Chemie International Edition (03.12.2001)
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PYRIMIDYL CYCLOPENTANES AS AKT PROTEIN KINASE INHIBITORS
HENTEMANN MARTIN F, SCHLACHTER STEPHEN T, XIAO DENGMING, LIANG JUN, GRAHAM JAMES M, BLAKE JAMES F, SPENCER KEITH L, BENCSIK JOSEF, MITCHELL IAN S, XU RUI, SAFINA BRIAN S, WELCH MIKE, KALLAN NICHOLAS C
Year of Publication 04.08.2015
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Year of Publication 04.08.2015
Patent
5H-CYCLOPENTA[d]PYRIMIDINE AS AKT PROTEIN KINASE INHIBITOR
HENTEMANN MARTIN F, ANNA BANKA, BENCSIK JOSEF R, JAMES F BLAKE, LIANG JUN, STEPHEN T SCHLACHTER, RUI XU, IAN S MITCHELL, ELI M WALLACE, TONY P TANG, KALLEN NICHOLAS C
Year of Publication 15.01.2015
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Year of Publication 15.01.2015
Patent
PYRIMIDYL CYCLOPENTANES AS AKT PROTEIN KINASE INHIBITORS
HENTEMANN MARTIN F, SCHLACHTER STEPHEN T, XIAO DENGMING, LIANG JUN, GRAHAM JAMES M, BLAKE JAMES F, SPENCER KEITH L, BENCSIK JOSEF, MITCHELL IAN S, XU RUI, SAFINA BRIAN S, WELCH MIKE, KALLAN NICHOLAS C
Year of Publication 30.04.2010
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Year of Publication 30.04.2010
Patent
Synthesis and oxidation reactions of cycloheptatrienyl sulfones
Tong, Zhiwei, Chen, Yuzhong, Hentemann, Martin F, Fuchs, Philip L
Published in Tetrahedron letters (07.10.2000)
Published in Tetrahedron letters (07.10.2000)
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SULFONE SUBSTITUTED 2,3-DIHYDROIMIDAZO Ý1,2-C¨QUINAZOLINE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES WITH ANGIOGENESIS
HENTEMANN, Martin, F, SCOTT, William, REDMAN, Aniko, JOHNSON, Jeffrey, WOOD, Jill, GUERNON, Leatte, BULLION, Ann-marie
Year of Publication 18.01.2017
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Year of Publication 18.01.2017
Patent
Thermal Intermolecular Hetero Diels-Alder Cycloadditions of Aldehydes and Imines via o-Quinone Dimethides
Hentemann, Martin F., Allen, John G., Danishefsky, Samuel J.
Published in Angewandte Chemie (02.06.2000)
Published in Angewandte Chemie (02.06.2000)
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