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Rosing, H., Hillebrand, M. J. X., Jimeno, J. M., Gómez, A., Floriano, P., Faircloth, G., Henrar, R. E. C., Vermorken, J. B., Cvitkovic, E., Bult, A., Beijnen, J. H.
Published in Journal of mass spectrometry. (01.11.1998)
Published in Journal of mass spectrometry. (01.11.1998)
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A clinical pharmacokinetics study of carzelesin given by short-term intravenous infusion in a phase I study
VAN TELLINGEN, O, PUNT, C. J. A, AWADA, A, WAGENER, D. J. T, PICCART, M. J, GROOT, Y, SCHAAF, L. J, HENRAR, R. E. C, NOOIJEN, W. J, BEIJNEN, J. H
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Published in Cancer chemotherapy and pharmacology (1998)
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Pharmaceutical development of a parenteral lyophilized formulation of the investigational antitumor neuropeptide antagonist [Arg6, D-Trp7,9, MePhe8]-substance P {6-11}
JONKMAN-DE VRIES, J. D, ROSING, H, TALSMA, H, HENRAR, R. E. C, KETTENES-VAN DEN BOSCH, J. J, BULT, A, BEIJNEN, J. H
Published in Investigational new drugs (01.01.1998)
Published in Investigational new drugs (01.01.1998)
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In vitro biocompatibility studies with the experimental anticancer agent BIBX1382BS
Nuijen, B., Bouma, M., Henrar, R.E.C., Brauns, U., Bette, P., Bult, A., Beijnen, J.H.
Published in International journal of pharmaceutics (25.01.2000)
Published in International journal of pharmaceutics (25.01.2000)
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Comparative pharmacology of the novel cyclopropylpyrroloindole-prodrug carzelesin in mice, rats, and humans
VAN TELLINGEN, O, NOOIJEN, W. J, SCHAAF, L. J, VAN DER VALK, M, VAN ASPEREN, J, HENRAR, R. E. C, BEIJNEN, J. H
Published in Cancer research (Chicago, Ill.) (01.06.1998)
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Published in Cancer research (Chicago, Ill.) (01.06.1998)
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Purity determinations in the bulk drug of the novel indoloquinone antitumor agent EO9
Jonkman-de Vries, J D, Kettenes-van den Bosch, J J, Henrar, R E, Bult, A, Beijnen, J H
Published in Investigational new drugs (01.01.1996)
Published in Investigational new drugs (01.01.1996)
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Pharmaceutical development of a parenteral formulation of the novel anti-tumor agent carzelesin (U-80,244)
Jonkman-de Vries, J D, de Graaff-Teulen, M J, Henrar, R E, Kettenes-van den Bosch, J J, Bult, A, Beijnen, J H
Published in Investigational new drugs (01.12.1994)
Published in Investigational new drugs (01.12.1994)
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Preclinical antitumour activity and animal toxicology studies of rhizoxin, a novel tubulin-interacting agent
HENDRIKS, H. R, PLOWMAN, J, BERGER, D. P, PAULL, K. D, FIEBIG, H. H, FODSTAD, Ø, DREEF-VAN DER MEULEN, H. C, HENRAR, R. E. C, PINEDO, H. M, SCHWARTSMANN, G
Published in Annals of oncology (01.11.1992)
Published in Annals of oncology (01.11.1992)
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Analysis of Ecteinascidin 743, a new potent marine-derived anticancer drug, in human plasma by high-performance liquid chromatography in combination with solid-phase extraction
Rosing, H, Hillebrand, M.J.X, Jimeno, J.M, Gómez, A, Floriano, P, Faircloth, G, Cameron, L, Henrar, R.E.C, Vermorken, J.B, Bult, A, Beijnen, J.H
Published in Journal of chromatography. B, Biomedical sciences and applications (12.06.1998)
Published in Journal of chromatography. B, Biomedical sciences and applications (12.06.1998)
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Bioanalysis of thiocoraline, a new marine antitumoral depsipeptide, in plasma by high-performance liquid chromatography and fluorescence detection
Sparidans, Rolf W, Henrar, Roland E.C, Jimeno, José M, Faircloth, Glynn, Floriano, Pablo, Beijnen, Jos H
Published in Journal of chromatography. B, Biomedical sciences and applications (16.04.1999)
Published in Journal of chromatography. B, Biomedical sciences and applications (16.04.1999)
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Bioanalysis of aplidine, a new marine antitumoral depsipeptide, in plasma by high-performance liquid chromatography after derivatization with trans-4′-hydrazino-2-stilbazole
Sparidans, Rolf W, Kettenes-van den Bosch, J.Jantien, van Tellingen, Olaf, Nuyen, Bastiaan, Henrar, Roland E.C, Jimeno, José M, Faircloth, Glynn, Floriano, Pablo, Rinehart, Kenneth L, Beijnen, Jos H
Published in Journal of chromatography. B, Biomedical sciences and applications (11.06.1999)
Published in Journal of chromatography. B, Biomedical sciences and applications (11.06.1999)
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Fully automated high-performance liquid chromatographic method for the determination of carzelesin (U-80,244) and metabolites (U-76,073 and U-76,074) in human plasma
van Tellingen, Olaf, Pels, Esther M., Henrar, Roland E.C., Schaaf, Lawrence J., Padbury, Guy E., Beijnen, Jos H., Nooijen, Willem J.
Published in Journal of chromatography (14.01.1994)
Published in Journal of chromatography (14.01.1994)
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EO9: A novel bioreductive alkylating indoloquinone with preferential solid tumour activity and lack of bone marrow toxicity in preclinical models
Hendriks, H.R., Pizao, P.E., Berger, D.P., Kooistra, K.L., Bibby, M.C., Boven, E., Dreef-van der Meulen, H.C., Henrar, R.E.C., Fiebig, H.H., Double, J.A., Hornstra, H.W., Pinedo, H.M., Workman, P., Schwartsmann, G.
Published in European journal of cancer (1990) (1993)
Published in European journal of cancer (1990) (1993)
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Compatibility and stability of aplidine, a novel marine-derived depsipeptide antitumor agent, in infusion devices, and its hemolytic and precipitation potential upon i.v. administration
Nuijen, B, Bouma, M, Henrar, R E, Manada, C, Bult, A, Beijnen, J H
Published in Anti-cancer drugs (01.11.1999)
Published in Anti-cancer drugs (01.11.1999)
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Pharmaceutical development of a parenteral lyophilized formulation of the novel antitumor agent aplidine
Nuijen, B, Bouma, M, Henrar, R E, Floriano, P, Jimeno, J M, Talsma, H, Kettenes-van den Bosch, J J, Heck, A J, Bult, A, Beijnen, J H
Published in PDA journal of pharmaceutical science and technology (01.05.2000)
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Published in PDA journal of pharmaceutical science and technology (01.05.2000)
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Revisions of general guidelines for the preclinical toxicology of new cytotoxic anticancer agents in Europe. The Cancer Research Campaign (CRC) Phase I/II Clinical Trials Committee and the European Organization for Research and Treatment of Cancer (EORTC) New Drug Development Office
Burtles, S S, Newell, D R, Henrar, R E, Connors, T A
Published in European journal of cancer (1990) (1995)
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Published in European journal of cancer (1990) (1995)
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Original article: Preclinical antitumour activity and animal toxicology studies of rhizoxin, a novel tubulin-interacting agent
Hendriks, H.R., Plowman, J., Berger, D. P., Paull, K. D., Fiebig, H. H., Fodstad, Ø., Meulen, H. C. Dreef-van der, Henrar, R. E. C., Pinedo, H. M., Schwartsman, G.
Published in Annals of oncology (01.11.1992)
Published in Annals of oncology (01.11.1992)
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