Alternative Farnsworth-Munsell Scoring Methodology for Testing Eyewear
Hennessy, Edward R.
Published in Proceedings of the Human Factors and Ergonomics Society Annual Meeting (01.11.2019)
Published in Proceedings of the Human Factors and Ergonomics Society Annual Meeting (01.11.2019)
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Journal Article
Discovery and Optimization of the First ATP Competitive Type-III c‑MET Inhibitor
Michaelides, Iacovos N., Collie, Gavin W., Börjesson, Ulf, Vasalou, Christina, Alkhatib, Omar, Barlind, Louise, Cheung, Tony, Dale, Ian L., Embrey, Kevin J., Hennessy, Edward J., Khurana, Puneet, Koh, Cheryl M., Lamb, Michelle L., Liu, Jianming, Moss, Thomas A., O’Neill, Daniel J., Phillips, Christopher, Shaw, Joseph, Snijder, Arjan, Storer, R. Ian, Stubbs, Christopher J., Han, Fujin, Li, Chengzhi, Qiao, Jingchuan, Sun, Dong-Qing, Wang, Jingwen, Wang, Peng, Yang, Wenzhen
Published in Journal of medicinal chemistry (13.07.2023)
Published in Journal of medicinal chemistry (13.07.2023)
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Journal Article
Discovery of a Novel Class of Dimeric Smac Mimetics as Potent IAP Antagonists Resulting in a Clinical Candidate for the Treatment of Cancer (AZD5582)
Hennessy, Edward J, Adam, Ammar, Aquila, Brian M, Castriotta, Lillian M, Cook, Donald, Hattersley, Maureen, Hird, Alexander W, Huntington, Christopher, Kamhi, Victor M, Laing, Naomi M, Li, Danyang, MacIntyre, Terry, Omer, Charles A, Oza, Vibha, Patterson, Troy, Repik, Galina, Rooney, Michael T, Saeh, Jamal C, Sha, Li, Vasbinder, Melissa M, Wang, Haiyun, Whitston, David
Published in Journal of medicinal chemistry (27.12.2013)
Published in Journal of medicinal chemistry (27.12.2013)
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Journal Article
Generating Selective Leads for Mer Kinase InhibitorsExample of a Comprehensive Lead-Generation Strategy
Nissink, J. Willem M, Bazzaz, Sana, Blackett, Carolyn, Clark, Matthew A, Collingwood, Olga, Disch, Jeremy S, Gikunju, Diana, Goldberg, Kristin, Guilinger, John P, Hardaker, Elizabeth, Hennessy, Edward J, Jetson, Rachael, Keefe, Anthony D, McCoull, William, McMurray, Lindsay, Olszewski, Allison, Overman, Ross, Pflug, Alexander, Preston, Marian, Rawlins, Philip B, Rivers, Emma, Schimpl, Marianne, Smith, Paul, Truman, Caroline, Underwood, Elizabeth, Warwicker, Juli, Winter-Holt, Jon, Woodcock, Simon, Zhang, Ying
Published in Journal of medicinal chemistry (25.03.2021)
Published in Journal of medicinal chemistry (25.03.2021)
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Journal Article
Optimization of an Imidazo[1,2‑a]pyridine Series to Afford Highly Selective Type I1/2 Dual Mer/Axl Kinase Inhibitors with In Vivo Efficacy
McCoull, William, Boyd, Scott, Brown, Martin R, Coen, Muireann, Collingwood, Olga, Davies, Nichola L, Doherty, Ann, Fairley, Gary, Goldberg, Kristin, Hardaker, Elizabeth, He, Guang, Hennessy, Edward J, Hopcroft, Philip, Hodgson, George, Jackson, Anne, Jiang, Xiefeng, Karmokar, Ankur, Lainé, Anne-Laure, Lindsay, Nicola, Mao, Yumeng, Markandu, Roshini, McMurray, Lindsay, McLean, Neville, Mooney, Lorraine, Musgrove, Helen, Nissink, J. Willem M, Pflug, Alexander, Reddy, Venkatesh Pilla, Rawlins, Philip B, Rivers, Emma, Schimpl, Marianne, Smith, Graham F, Tentarelli, Sharon, Travers, Jon, Troup, Robert I, Walton, Josephine, Wang, Cheng, Wilkinson, Stephen, Williamson, Beth, Winter-Holt, Jon, Yang, Dejian, Zheng, Yuting, Zhu, Qianxiu, Smith, Paul D
Published in Journal of medicinal chemistry (23.09.2021)
Published in Journal of medicinal chemistry (23.09.2021)
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Journal Article
Structural and Molecular Insight into Resistance Mechanisms of First Generation cMET Inhibitors
Collie, Gavin W, Koh, Cheryl M, O’Neill, Daniel J, Stubbs, Christopher J, Khurana, Puneet, Eddershaw, Alice, Snijder, Arjan, Mauritzson, Fredrik, Barlind, Louise, Dale, Ian L, Shaw, Joseph, Phillips, Christopher, Hennessy, Edward J, Cheung, Tony, Narvaez, Ana J
Published in ACS medicinal chemistry letters (12.09.2019)
Published in ACS medicinal chemistry letters (12.09.2019)
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Journal Article
Discovery of Potent KIFC1 Inhibitors Using a Method of Integrated High-Throughput Synthesis and Screening
Yang, Bin, Lamb, Michelle L, Zhang, Tao, Hennessy, Edward J, Grewal, Gurmit, Sha, Li, Zambrowski, Mark, Block, Michael H, Dowling, James E, Su, Nancy, Wu, Jiaquan, Deegan, Tracy, Mikule, Keith, Wang, Wenxian, Kaspera, Rüdiger, Chuaqui, Claudio, Chen, Huawei
Published in Journal of medicinal chemistry (11.12.2014)
Published in Journal of medicinal chemistry (11.12.2014)
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Journal Article
Identification and Optimization of Benzimidazole Sulfonamides as Orally Bioavailable Sphingosine 1‑Phosphate Receptor 1 Antagonists with in Vivo Activity
Hennessy, Edward J., Oza, Vibha, Adam, Ammar, Byth, Kate, Castriotta, Lillian, Grewal, Gurmit, Hamilton, Geraldine A., Kamhi, Victor M., Lewis, Paula, Li, Danyang, Lyne, Paul, Öster, Linda, Rooney, Michael T., Saeh, Jamal C., Sha, Li, Su, Qibin, Wen, Shengua, Xue, Yafeng, Yang, Bin
Published in Journal of medicinal chemistry (10.09.2015)
Published in Journal of medicinal chemistry (10.09.2015)
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Journal Article
Optimization of Highly Kinase Selective Bis-anilino Pyrimidine PAK1 Inhibitors
McCoull, William, Hennessy, Edward J, Blades, Kevin, Chuaqui, Claudio, Dowling, James E, Ferguson, Andrew D, Goldberg, Frederick W, Howe, Nicholas, Jones, Christopher R, Kemmitt, Paul D, Lamont, Gillian, Varnes, Jeffrey G, Ward, Richard A, Yang, Bin
Published in ACS medicinal chemistry letters (08.12.2016)
Published in ACS medicinal chemistry letters (08.12.2016)
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Journal Article
Discovery of heterocyclic sulfonamides as sphingosine 1-phosphate receptor 1 (S1P1) antagonists
Hennessy, Edward J., Grewal, Gurmit, Byth, Kate, Kamhi, Victor M., Li, Danyang, Lyne, Paul, Oza, Vibha, Ronco, Lucienne, Rooney, Michael T., Saeh, Jamal C., Su, Qibin
Published in Bioorganic & medicinal chemistry letters (15.05.2015)
Published in Bioorganic & medicinal chemistry letters (15.05.2015)
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Journal Article
Discovery of aminopiperidine-based Smac mimetics as IAP antagonists
Hennessy, Edward J., Saeh, Jamal C., Sha, Li, MacIntyre, Terry, Wang, Haiyun, Larsen, Nicholas A., Aquila, Brian M., Ferguson, Andrew D., Laing, Naomi M., Omer, Charles A.
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
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Journal Article
Structure-based design and synthesis of tricyclic IAP (Inhibitors of Apoptosis Proteins) inhibitors
Hird, Alexander W., Aquila, Brian M., Block, Michael H., Hennessy, Edward J., Kamhi, Victor M., Omer, Charles A., Laing, Naomi M., Saeh, Jamal C., Sha, Li, Yang, Bin
Published in Bioorganic & medicinal chemistry letters (01.04.2014)
Published in Bioorganic & medicinal chemistry letters (01.04.2014)
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Journal Article
Direct and selective elimination of specific prions and amyloids by 4,5-dianilinophthalimide and analogs
Wang, Huan, Duennwald, Martin L, Roberts, Blake E, Rozeboom, Leslie M, Zhang, Yingxin L, Steele, Andrew D, Krishnan, Rajaraman, Su, Linhui Julie, Griffin, Drees, Mukhopadhyay, Samrat, Hennessy, Edward J, Weigele, Peter, Blanchard, Barbara J, King, Jonathan, Deniz, Ashok A, Buchwald, Stephen L, Ingram, Vernon M, Lindquist, Susan, Shorter, James
Published in Proceedings of the National Academy of Sciences - PNAS (20.05.2008)
Published in Proceedings of the National Academy of Sciences - PNAS (20.05.2008)
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Journal Article
Utilization of Structure-Based Design to Identify Novel, Irreversible Inhibitors of EGFR Harboring the T790M Mutation
Hennessy, Edward J, Chuaqui, Claudio, Ashton, Susan, Colclough, Nicola, Cross, Darren A. E, Debreczeni, Judit É, Eberlein, Cath, Gingipalli, Lakshmaiah, Klinowska, Teresa C. M, Orme, Jonathan P, Sha, Li, Wu, Xiaoyun
Published in ACS medicinal chemistry letters (12.05.2016)
Published in ACS medicinal chemistry letters (12.05.2016)
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Journal Article
Preparation of highly functionalized 1,5-disubstituted tetrazoles via palladium-catalyzed Suzuki coupling
Hennessy, Edward J., Cornebise, Mark, Gingipalli, Lakshmaiah, Grebe, Tyler, Hande, Sudhir, Hoesch, Valerie, Huynh, Hoan, Throner, Scott, Varnes, Jeffrey, Wu, Ye
Published in Tetrahedron letters (26.04.2017)
Published in Tetrahedron letters (26.04.2017)
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Journal Article
Evaluating the Effects of Clothing and Individual Equipment on Marksmanship Performance Using a Novel Five Target Methodology
McNamara, Jay A., Choi, Hyeg Joo, Brown, Stephanie A.T., Hennessy, Edward R., Mitchell, K. Blake
Published in Proceedings of the Human Factors and Ergonomics Society Annual Meeting (01.09.2016)
Published in Proceedings of the Human Factors and Ergonomics Society Annual Meeting (01.09.2016)
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Journal Article