Moderation of iodoacetate-induced experimental osteoarthritis in rats by matrix metalloproteinase inhibitors
Janusz, M.J., Hookfin, E.B., Heitmeyer, S.A., Woessner, J.F., Freemont, A.J., Hoyland, J.A., Brown, K.K., Hsieh, L.C., Almstead, N.G., De, B., Natchus, M.G., Pikul, S., Taiwo, Y.O.
Published in Osteoarthritis and cartilage (01.11.2001)
Published in Osteoarthritis and cartilage (01.11.2001)
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Detection of aggrecanase- and MMP-generated catabolic neoepitopes in the rat iodoacetate model of cartilage degeneration
Janusz, M.J., Little, C.B., King, L.E., Hookfin, E.B., Brown, K.K., Heitmeyer, S.A., Caterson, B., Poole, A.R., Taiwo, Y.O.
Published in Osteoarthritis and cartilage (01.09.2004)
Published in Osteoarthritis and cartilage (01.09.2004)
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Journal Article
Development of New Hydroxamate Matrix Metalloproteinase Inhibitors Derived from Functionalized 4-Aminoprolines
Natchus, Michael G, Bookland, Roger G, De, Biswanath, Almstead, Neil G, Pikul, Stanislaw, Janusz, Michael J, Heitmeyer, Sandra A, Hookfin, Erin B, Hsieh, Lily C, Dowty, Martin E, Dietsch, Charles R, Patel, Vikram S, Garver, Susan M, Gu, Fei, Pokross, Matthew E, Mieling, Glen E, Baker, Timothy R, Foltz, David J, Peng, Sean X, Bornes, David M, Strojnowski, Michael J, Taiwo, Yetunde O
Published in Journal of medicinal chemistry (28.12.2000)
Published in Journal of medicinal chemistry (28.12.2000)
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Journal Article
Induction of osteoarthritis in the rat by surgical tear of the meniscus: Inhibition of joint damage by a matrix metalloproteinase inhibitor
Janusz, M.J., Bendele, A.M., Brown, K.K., Taiwo, Y.O., Hsieh, L., Heitmeyer, S.A.
Published in Osteoarthritis and cartilage (01.10.2002)
Published in Osteoarthritis and cartilage (01.10.2002)
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Journal Article
Comparison of the pharmacology of hydroxamate- and carboxylate-based matrix metalloproteinase inhibitors (MMPIs) for the treatment of osteoarthritis
Janusz, M J, Hookfin, E B, Brown, K K, Hsieh, L C, Heitmeyer, S A, Taiwo, Y O, Natchus, M G, Pikul, S, Almstead, N G, De, B, Peng, S X, Baker, T R, Patel, V
Published in Inflammation research (01.02.2006)
Published in Inflammation research (01.02.2006)
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Development of Orally Bioavailable Bicyclic Pyrazolones as Inhibitors of Tumor Necrosis Factor-α Production
Clark, Michael P, Laughlin, Steven K, Laufersweiler, Matthew J, Bookland, Roger G, Brugel, Todd A, Golebiowski, Adam, Sabat, Mark P, Townes, Jennifer A, VanRens, John C, Djung, Jane F, Natchus, Michael G, De, Biswanath, Hsieh, Lily C, Xu, Susan C, Walter, Rick L, Mekel, Marlene J, Heitmeyer, Sandra A, Brown, Kimberly K, Juergens, Karen, Taiwo, Yetunde O, Janusz, Michael J
Published in Journal of medicinal chemistry (20.05.2004)
Published in Journal of medicinal chemistry (20.05.2004)
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The development of novel inhibitors of tumor necrosis factor-α (TNF-α) production based on substituted [5,5]-bicyclic pyrazolones
Laufersweiler, Matthew J, Brugel, Todd A, Clark, Michael P, Golebiowski, Adam, Bookland, Roger G, Laughlin, Steven K, Sabat, Mark P, Townes, Jennifer A, VanRens, John C, De, Biswanath, Hsieh, Lily C, Heitmeyer, Sandra A, Juergens, Karen, Brown, Kimberly K, Mekel, Marlene J, Walter, Richard L, Janusz, Michael J
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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Method and device for producing, filling, and closing bags, and a bag
KOEHN UWE, VOSS HANS-LUDWIG, WOCKENFUSS GERD, GROSSE-HEITMEYER RUEDIGER, HAWIGHORST THOMAS
Year of Publication 16.07.2014
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Year of Publication 16.07.2014
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