Schwann cell endosome CGRP signals elicit periorbital mechanical allodynia in mice
De Logu, Francesco, Nassini, Romina, Hegron, Alan, Landini, Lorenzo, Jensen, Dane D, Latorre, Rocco, Ding, Julia, Marini, Matilde, Souza Monteiro de Araujo, Daniel, Ramírez-Garcia, Paulina, Whittaker, Michael, Retamal, Jeffri, Titiz, Mustafa, Innocenti, Alessandro, Davis, Thomas P, Veldhuis, Nicholas, Schmidt, Brian L, Bunnett, Nigel W, Geppetti, Pierangelo
Published in Nature communications (03.02.2022)
Published in Nature communications (03.02.2022)
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Endosomal signaling of delta opioid receptors is an endogenous mechanism and therapeutic target for relief from inflammatory pain
Jimenez-Vargas, Nestor N., Gong, Jing, Wisdom, Matthew J., Jensen, Dane D., Latorre, Rocco, Hegron, Alan, Teng, Shavonne, DiCello, Jesse J., Rajasekhar, Pradeep, Veldhuis, Nicholas A., Carbone, Simona E., Yu, Yang, Lopez-Lopez, Cintya, Jaramillo-Polanco, Josue, Canals, Meritxell, Reed, David E., Lomax, Alan E., Schmidt, Brian L., Leong, Kam W., Vanner, Stephen J., Halls, Michelle L., Bunnett, Nigel W., Poole, Daniel P.
Published in Proceedings of the National Academy of Sciences - PNAS (30.06.2020)
Published in Proceedings of the National Academy of Sciences - PNAS (30.06.2020)
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Opioid-Induced Pronociceptive Signaling in the Gastrointestinal Tract Is Mediated by Delta-Opioid Receptor Signaling
Jaramillo-Polanco, Josue, Lopez-Lopez, Cintya, Yu, Yang, Neary, Emma, Hegron, Alan, Canals, Meritxell, Bunnett, Nigel W, Reed, David E, Lomax, Alan E, Vanner, Stephen J
Published in The Journal of neuroscience (20.04.2022)
Published in The Journal of neuroscience (20.04.2022)
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Journal Article
Melatonin receptors limit dopamine reuptake by regulating dopamine transporter cell-surface exposure
Benleulmi-Chaachoua, Abla, Hegron, Alan, Le Boulch, Marine, Karamitri, Angeliki, Wierzbicka, Marta, Wong, Victoria, Stagljar, Igor, Delagrange, Philippe, Ahmad, Raise, Jockers, Ralf
Published in Cellular and molecular life sciences : CMLS (01.12.2018)
Published in Cellular and molecular life sciences : CMLS (01.12.2018)
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Therapeutic antagonism of the neurokinin 1 receptor in endosomes provides sustained pain relief
Hegron, Alan, Peach, Chloe J, Tonello, Raquel, Seemann, Philipp, Teng, Shavonne, Latorre, Rocco, Huebner, Harald, Weikert, Dorothee, Rientjes, Jeanette, Veldhuis, Nicholas A, Poole, Daniel P, Jensen, Dane D, Thomsen, Alex R B, Schmidt, Brian L, Imlach, Wendy L, Gmeiner, Peter, Bunnett, Nigel W
Published in Proceedings of the National Academy of Sciences - PNAS (30.05.2023)
Published in Proceedings of the National Academy of Sciences - PNAS (30.05.2023)
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Mice expressing fluorescent PAR2 reveal that endocytosis mediates colonic inflammation and pain
Latorre, Rocco, Hegron, Alan, Peach, Chloe J, Teng, Shavonne, Tonello, Raquel, Retamal, Jeffri S, Klein-Cloud, Rafael, Bok, Diana, Jensen, Dane D, Gottesman-Katz, Lena, Rientjes, Jeanette, Veldhuis, Nicholas A, Poole, Daniel P, Schmidt, Brian L, Pothoulakis, Charalabos H, Rankin, Carl, Xie, Ying, Koon, Wai, Bunnett, Nigel W
Published in Proceedings of the National Academy of Sciences - PNAS (08.02.2022)
Published in Proceedings of the National Academy of Sciences - PNAS (08.02.2022)
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Journal Article
Mice expressing fluorescent PAR 2 reveal that endocytosis mediates colonic inflammation and pain
Latorre, Rocco, Hegron, Alan, Peach, Chloe J, Teng, Shavonne, Tonello, Raquel, Retamal, Jeffri S, Klein-Cloud, Rafael, Bok, Diana, Jensen, Dane D, Gottesman-Katz, Lena, Rientjes, Jeanette, Veldhuis, Nicholas A, Poole, Daniel P, Schmidt, Brian L, Pothoulakis, Charalabos H, Rankin, Carl, Xie, Ying, Koon, Hon Wai, Bunnett, Nigel W
Published in Proceedings of the National Academy of Sciences - PNAS (08.02.2022)
Published in Proceedings of the National Academy of Sciences - PNAS (08.02.2022)
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Journal Article
Human GLP1R variants affecting GLP1R cell surface expression are associated with impaired glucose control and increased adiposity
Gao, Wenwen, Liu, Lei, Huh, Eunna, Gbahou, Florence, Cecon, Erika, Oshima, Masaya, Houzé, Ludivine, Katsonis, Panagiotis, Hegron, Alan, Fan, Zhiran, Hou, Guofei, Charpentier, Guillaume, Boissel, Mathilde, Derhourhi, Mehdi, Marre, Michel, Balkau, Beverley, Froguel, Philippe, Scharfmann, Raphael, Lichtarge, Olivier, Dam, Julie, Bonnefond, Amélie, Liu, Jianfeng, Jockers, Ralf
Published in Nature metabolism (01.10.2023)
Published in Nature metabolism (01.10.2023)
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Type 2 diabetes-associated variants of the MT 2 melatonin receptor affect distinct modes of signaling
Karamitri, Angeliki, Plouffe, Bianca, Bonnefond, Amélie, Chen, Min, Gallion, Jonathan, Guillaume, Jean-Luc, Hegron, Alan, Boissel, Mathilde, Canouil, Mickaël, Langenberg, Claudia, Wareham, Nicholas J, Le Gouill, Christian, Lukasheva, Viktoria, Lichtarge, Olivier, Froguel, Philippe, Bouvier, Michel, Jockers, Ralf
Published in Science signaling (28.08.2018)
Published in Science signaling (28.08.2018)
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Identification of Key Regions Mediating Human Melatonin Type 1 Receptor Functional Selectivity Revealed by Natural Variants
Hegron, Alan, Huh, Eunna, Deupi, Xavier, Sokrat, Badr, Gao, Wenwen, Le Gouill, Christian, Canouil, Mickaël, Boissel, Mathilde, Charpentier, Guillaume, Roussel, Ronan, Balkau, Beverley, Froguel, Philippe, Plouffe, Bianca, Bonnefond, Amélie, Lichtarge, Olivier, Jockers, Ralf, Bouvier, Michel
Published in ACS pharmacology & translational science (01.09.2021)
Published in ACS pharmacology & translational science (01.09.2021)
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Journal Article
Identification of Key Regions Mediating Human Melatonin Type 1 Receptor Functional Selectivity Revealed by Natural Variants
Hegron, Alan, Huh, Eunna, Deupi, Xavier, Sokrat, Badr, Gao, Wenwen, Le Gouill, Christian, Canouil, Mickaël, Boissel, Mathilde, Charpentier, Guillaume, Roussel, Ronan, Balkau, Beverley, Froguel, Philippe, Plouffe, Bianca, Bonnefond, Amélie, Lichtarge, Olivier, Jockers, Ralf, Bouvier, Michel
Published in ACS pharmacology & translational science (08.10.2021)
Published in ACS pharmacology & translational science (08.10.2021)
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