3-(7-Azaindolyl)-4-arylmaleimides as potent, selective inhibitors of glycogen synthase kinase-3
Zhang, Han-Cheng, Ye, Hong, Conway, Bruce R., Derian, Claudia K., Addo, Michael F., Kuo, Gee-Hong, Hecker, Leonard R., Croll, Diane R., Li, Jian, Westover, Lori, Xu, Jun Z., Look, Richard, Demarest, Keith T., Andrade-Gordon, Patricia, Damiano, Bruce P., Maryanoff, Bruce E.
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Novel Indolylindazolylmaleimides as Inhibitors of Protein Kinase C-β: Synthesis, Biological Activity, and Cardiovascular Safety
Zhang, Han-Cheng, Derian, Claudia K, McComsey, David F, White, Kimberly B, Ye, Hong, Hecker, Leonard R, Li, Jian, Addo, Michael F, Croll, Diane, Eckardt, Annette J, Smith, Charles E, Li, Quan, Cheung, Wai-Man, Conway, Bruce R, Emanuel, Stuart, Demarest, Keith T, Andrade-Gordon, Patricia, Damiano, Bruce P, Maryanoff, Bruce E
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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In-depth study of tripeptide-based alpha-ketoheterocycles as inhibitors of thrombin. Effective utilization of the S-1 ' subsite and its implications to structure-based drug design
Costanzo, MJ, Almond, HR, Hecker, LR, Schott, MR, Yabut, SC, Zhang, HC, Andrade-Gordon, P, Corcoran, TW, Giardino, EC, Kauffman, JA, Lewis, JM, de Garavilla, L, Haertlein, BJ, Maryanoff, BE
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Potent, Orally Active GPIIb/IIIa Antagonists Containing a Nipecotic Acid Subunit. Structure−Activity Studies Leading to the Discovery of RWJ-53308
Hoekstra, William J, Maryanoff, Bruce E, Damiano, Bruce P, Andrade-Gordon, Patricia, Cohen, Judith H, Costanzo, Michael J, Haertlein, Barbara J, Hecker, Leonard R, Hulshizer, Becky L, Kauffman, Jack A, Keane, Patricia, McComsey, David F, Mitchell, John A, Scott, Lorraine, Shah, Rekha D, Yabut, Stephen C
Published in Journal of medicinal chemistry (16.12.1999)
Published in Journal of medicinal chemistry (16.12.1999)
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Synthesis, resolution, and absolute configuration of novel tricyclic benzodiazepines
Matthews, Jay M., Dyatkin, Alexey B., Evangelisto, Mary, Gauthier, Diane A., Hecker, Leonard R., Hoekstra, William J., Liu, Fuqiang, Poulter, Brenda L., Sorgi, Kirk L., Maryanoff, Bruce E.
Published in Tetrahedron: asymmetry (19.04.2004)
Published in Tetrahedron: asymmetry (19.04.2004)
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Synthesis and biological evaluation of novel indoloazepine derivatives as non-peptide vasopressin V2 receptor antagonists
Matthews, Jay M, Greco, Michael N, Hecker, Leonard R, Hoekstra, William J, Andrade-Gordon, Patricia, Garavilla, Lawrence de, Demarest, Keith T, Ericson, Eric, Gunnet, Joseph W, Hageman, William, Look, Richard, Moore, John B, Maryanoff, Bruce E
Published in Bioorganic & medicinal chemistry letters (24.02.2003)
Published in Bioorganic & medicinal chemistry letters (24.02.2003)
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Potent nonpeptide vasopressin receptor antagonists based on oxazino- and thiazinobenzodiazepine templates
Matthews, Jay M., Hoekstra, William J., Dyatkin, Alexey B., Hecker, Leonard R., Hlasta, Dennis J., Poulter, Brenda L., Andrade-Gordon, Patricia, de Garavilla, Lawrence, Demarest, Keith T., Ericson, Eric, Gunnet, Joseph W., Hageman, William, Look, Richard, Moore, John B., Reynolds, Charles H., Maryanoff, Bruce E.
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
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Potent thrombin inhibitors that probe the S-1' subsite: Tripeptide transition state analogues based on a heterocycle-activated carbonyl group
Costanzo, MJ, Maryanoff, BE, Hecker, LR, Schott, MR, Yabut, SC, Zhang, HC, AndradeGordon, P, Kauffman, JA, Lewis, JM, Krishnan, R, Tulinsky, A
Published in Journal of medicinal chemistry (02.08.1996)
Published in Journal of medicinal chemistry (02.08.1996)
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An Expedient Method for Resolution of 3-Amino-3-(3‘-pyridyl)propionic Acid and Related Compounds
Boesch, Heinz, Cesco-Cancian, Sergio, Hecker, Leonard R, Hoekstra, William J, Justus, Michael, Maryanoff, Cynthia A, Scott, Lorraine, Shah, Rekha D, Solms, Guenter, Sorgi, Kirk L, Stefanick, Stephen M, Thurnheer, Urs, Villani, Frank J, Walker, Donald G
Published in Organic process research & development (01.01.2001)
Published in Organic process research & development (01.01.2001)
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Novel thrombin inhibitors that are based on a macrocyclic tripeptide motif
Greco, Michael N., Powell, Eugene T., Hecker, Leonard R., Andrade-Gordon, Patricia, Kauffman, Jack A., Lewis, Joan M., Ganesh, Venkatapathy, Tulinsky, Alexander, Maryanoff, Bruce E.
Published in Bioorganic & medicinal chemistry letters (17.12.1996)
Published in Bioorganic & medicinal chemistry letters (17.12.1996)
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IMPROVED PROCEDURES FOR THE PREPARATION OF CYCLOALKYLTHIOUREAS, ARYLALKYLTHIOUREAS, AND ARYLTHIOUREAS
RASMUSSEN, CR, VILLANI, FJ, WEANER, LE, REYNOLDS, BE, HOOD, AR, HECKER, LR, NORTEY, SO, HANSLIN, A, COSTANZO, MJ, POWELL, ET, MOLINARI, AJ
Published in Synthesis (Stuttgart) (01.06.1988)
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Published in Synthesis (Stuttgart) (01.06.1988)
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A VERSATILE SYNTHESIS OF NOVEL N,N,N'-TRISUBSTITUTED GUANIDINES
RASMUSSEN, CR, VILLANI, FJ, REYNOLDS, BE, PLAMPIN, JN, HOOD, AR, HECKER, LR, NORTEY, SO, HANSLIN, A, COSTANZO, MJ, HOWSE, RM, MOLINARI, AJ
Published in Synthesis (Stuttgart) (1988)
Published in Synthesis (Stuttgart) (1988)
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