robustica: customizable robust independent component analysis
Anglada-Girotto, Miquel, Miravet-Verde, Samuel, Serrano, Luis, Head, Sarah A
Published in BMC bioinformatics (05.12.2022)
Published in BMC bioinformatics (05.12.2022)
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Silencing of SRRM4 suppresses microexon inclusion and promotes tumor growth across cancers
Head, Sarah A, Hernandez-Alias, Xavier, Yang, Jae-Seong, Ciampi, Ludovica, Beltran-Sastre, Violeta, Torres-Méndez, Antonio, Irimia, Manuel, Schaefer, Martin H, Serrano, Luis
Published in PLoS biology (23.02.2021)
Published in PLoS biology (23.02.2021)
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Antifungal drug itraconazole targets VDAC1 to modulate the AMPK/mTOR signaling axis in endothelial cells
Head, Sarah A., Shi, Wei, Zhao, Liang, Gorshkov, Kirill, Pasunooti, Kalyan, Chen, Yue, Deng, Zhiyou, Li, Ruo-jing, Shim, Joong Sup, Tan, Wenzhi, Hartung, Thomas, Zhang, Jin, Zhao, Yingming, Colombini, Marco, Liu, Jun O.
Published in Proceedings of the National Academy of Sciences - PNAS (29.12.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (29.12.2015)
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Pharmacological blockade of cholesterol trafficking by cepharanthine in endothelial cells suppresses angiogenesis and tumor growth
Lyu, Junfang, Yang, Eun Ju, Head, Sarah A., Ai, Nana, Zhang, Baoyuan, Wu, Changjie, Li, Ruo-Jing, Liu, Yifan, Yang, Chen, Dang, Yongjun, Kwon, Ho Jeong, Ge, Wei, Liu, Jun O., Shim, Joong Sup
Published in Cancer letters (28.11.2017)
Published in Cancer letters (28.11.2017)
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Simultaneous Targeting of NPC1 and VDAC1 by Itraconazole Leads to Synergistic Inhibition of mTOR Signaling and Angiogenesis
Head, Sarah A, Shi, Wei Q, Yang, Eun Ju, Nacev, Benjamin A, Hong, Sam Y, Pasunooti, Kalyan K, Li, Ruo-Jing, Shim, Joong Sup, Liu, Jun O
Published in ACS chemical biology (20.01.2017)
Published in ACS chemical biology (20.01.2017)
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Modulation of the Endomembrane System by the Anticancer Natural Product Superstolide/ZJ-101
Sanchez, Phillip R, Head, Sarah A, Qian, Shan, Qiu, Haibo, Roy, Avishek, Jin, Zhendong, Zheng, Wei, Liu, Jun O
Published in International journal of molecular sciences (31.05.2023)
Published in International journal of molecular sciences (31.05.2023)
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Comparison of dose selection based on target engagement versus inhibition of receptor–ligand interaction for checkpoint inhibitors
Head, Sarah A., Johnson, Carter, Sarkar, Saheli, Matteson, Andrew, Marcantonio, Diana H., Hua, Fei, Burke, John M., Apgar, Joshua F., Flowers, David
Published in CPT: pharmacometrics and systems pharmacology (01.06.2024)
Published in CPT: pharmacometrics and systems pharmacology (01.06.2024)
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Divergence of Antiangiogenic Activity and Hepatotoxicity of Different Stereoisomers of Itraconazole
Shim, Joong Sup, Li, Ruo-Jing, Bumpus, Namandje N, Head, Sarah A, Kumar Pasunooti, Kalyan, Yang, Eun Ju, Lv, Junfang, Shi, Wei, Liu, Jun O
Published in Clinical cancer research (01.06.2016)
Published in Clinical cancer research (01.06.2016)
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Insights into the structure–activity relationship of the anticancer compound ZJ-101: A role played by the amide moiety
Qiu, Haibo, Qian, Shan, Head, Sarah A., Sanchez, Phillip R., Liu, Jun O., Jin, Zhendong
Published in Bioorganic & medicinal chemistry letters (01.06.2024)
Published in Bioorganic & medicinal chemistry letters (01.06.2024)
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Synthesis and biological evaluation of biotinylated ZJ-101
Qian, Shan, Head, Sarah A., Sanchez, Phillip R., Liu, Jun O., Jin, Zhendong
Published in Bioorganic & medicinal chemistry letters (15.07.2023)
Published in Bioorganic & medicinal chemistry letters (15.07.2023)
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Targeted Delivery and Sustained Antitumor Activity of Triptolide through Glucose Conjugation
He, Qing-Li, Minn, Il, Wang, Qiaoling, Xu, Peng, Head, Sarah A., Datan, Emmanuel, Yu, Biao, Pomper, Martin G., Liu, Jun O.
Published in Angewandte Chemie (International ed.) (19.09.2016)
Published in Angewandte Chemie (International ed.) (19.09.2016)
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ProteinFishing: a protein complex generator within the ModelX toolsuite
Cianferoni, Damiano, Radusky, Leandro G, Head, Sarah A, Serrano, Luis, Delgado, Javier
Published in Bioinformatics (15.08.2020)
Published in Bioinformatics (15.08.2020)
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Novel Tetrazole-Containing Analogues of Itraconazole as Potent Antiangiogenic Agents with Reduced Cytochrome P450 3A4 Inhibition
Li, Yingjun, Pasunooti, Kalyan Kumar, Li, Ruo-Jing, Liu, Wukun, Head, Sarah A, Shi, Wei Q, Liu, Jun O
Published in Journal of medicinal chemistry (27.12.2018)
Published in Journal of medicinal chemistry (27.12.2018)
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Specialization of the photoreceptor transcriptome by Srrm3 -dependent microexons is required for outer segment maintenance and vision
Ciampi, Ludovica, Mantica, Federica, López-Blanch, Laura, Permanyer, Jon, Rodriguez-Marín, Cristina, Zang, Jingjing, Cianferoni, Damiano, Jiménez-Delgado, Senda, Bonnal, Sophie, Miravet-Verde, Samuel, Ruprecht, Verena, Neuhauss, Stephan C F, Banfi, Sandro, Carrella, Sabrina, Serrano, Luis, Head, Sarah A, Irimia, Manuel
Published in Proceedings of the National Academy of Sciences - PNAS (19.07.2022)
Published in Proceedings of the National Academy of Sciences - PNAS (19.07.2022)
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Itraconazole Inhibits Enterovirus Replication by Targeting the Oxysterol-Binding Protein
Strating, Jeroen R.P.M., van der Linden, Lonneke, Albulescu, Lucian, Bigay, Joëlle, Arita, Minetaro, Delang, Leen, Leyssen, Pieter, van der Schaar, Hilde M., Lanke, Kjerstin H.W., Thibaut, Hendrik Jan, Ulferts, Rachel, Drin, Guillaume, Schlinck, Nina, Wubbolts, Richard W., Sever, Navdar, Head, Sarah A., Liu, Jun O., Beachy, Philip A., De Matteis, Maria A., Shair, Matthew D., Olkkonen, Vesa M., Neyts, Johan, van Kuppeveld, Frank J.M.
Published in Cell reports (Cambridge) (03.02.2015)
Published in Cell reports (Cambridge) (03.02.2015)
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Inhibition of angiogenesis by selective estrogen receptor modulators through blockade of cholesterol trafficking rather than estrogen receptor antagonism
Shim, Joong Sup, Li, Ruo-Jing, Lv, Junfang, Head, Sarah A, Yang, Eun Ju, Liu, Jun O
Published in Cancer letters (28.06.2015)
Published in Cancer letters (28.06.2015)
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Insights into the structure–activity relationship of the anticancer compound ZJ-101, a derivative of marine natural product superstolide A: A role played by the lactone moiety
Qiu, Haibo, Qian, Shan, Head, Sarah A., Liu, Jun O., Jin, Zhendong
Published in Bioorganic & medicinal chemistry letters (01.10.2016)
Published in Bioorganic & medicinal chemistry letters (01.10.2016)
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Structure-activity relationship study of itraconazole, a broad-range inhibitor of picornavirus replication that targets oxysterol-binding protein (OSBP)
Bauer, Lisa, Ferla, Salvatore, Head, Sarah A., Bhat, Shridhar, Pasunooti, Kalyan K., Shi, Wei Q., Albulescu, Lucian, Liu, Jun O., Brancale, Andrea, van Kuppeveld, Frank J.M., Strating, Jeroen R.P.M.
Published in Antiviral research (01.08.2018)
Published in Antiviral research (01.08.2018)
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Astemizole Inhibits mTOR Signaling and Angiogenesis by Blocking Cholesterol Trafficking
Lyu, Junfang, Yang, Eun Ju, Head, Sarah A, Ai, Nana, Zhang, Baoyuan, Wu, Changjie, Li, Ruo-Jing, Liu, Yifan, Chakravarty, Harapriya, Zhang, Shaolin, Tam, Kin Yip, Dang, Yongjun, Kwon, Ho Jeong, Ge, Wei, Liu, Jun O, Shim, Joong Sup
Published in International journal of biological sciences (01.01.2018)
Published in International journal of biological sciences (01.01.2018)
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