Discovery of novel CDK8 inhibitors using multiple crystal structures in docking-based virtual screening
Wang, Taijin, Yang, Zhuang, Zhang, Yongguang, Yan, Wei, Wang, Fang, He, Linhong, Zhou, Yuanyuan, Chen, Lijuan
Published in European journal of medicinal chemistry (31.03.2017)
Published in European journal of medicinal chemistry (31.03.2017)
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Journal Article
Comparison of counter-current chromatography and preparative high performance liquid chromatography applied to separating minor impurities in drug preparations
Li, Shucai, Wang, Wenwen, Tang, Huan, Chen, Kai, Yang, Jianhong, He, Linhong, Ye, Haoyu, Peng, Aihua, Chen, Lijuan
Published in Journal of Chromatography A (30.05.2014)
Published in Journal of Chromatography A (30.05.2014)
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Synthesis and Biological Evaluation of 3-Methyl-5-phenylthieno[2,3-d]pyrimidine-2,4(1H,3H)-dione Derivatives for the Treatment of Diet-Induced Obesity
Sang, Yun, Pei, Heyin, Ma, Liang, Huang, Li, Xie, Caifeng, Chen, Jinying, Liang, Xiaolin, Ran, Yan, Wang, Guangcheng, Yang, Zhuang, Cao, Dong, He, Lin, Wu, Yuzhe, He, Linhong, Zhu, Jun, Lan, Jingbo, Chen, Lijuan
Published in Chemical & pharmaceutical bulletin (01.09.2014)
Published in Chemical & pharmaceutical bulletin (01.09.2014)
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Engineering highly efficient Li+ responsive nanochannels via host–guest interaction and photochemistry regulation
Li, Shuting, Li, Manting, Chen, Limin, Yang, Jianying, Wang, Zhao, Yang, Fan, He, Linhong, Li, Xinchun
Published in Journal of colloid and interface science (01.06.2022)
Published in Journal of colloid and interface science (01.06.2022)
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Journal Article
Development of novel nitric oxide production inhibitors based on the 7H-pyrrolo[2,3-d]pyrimidine scaffold
Zhang, Jie, Xie, Xin, Qin, Tingsheng, Yao, Hualiang, Ling, Zhen, Deng, Fengyuan, Yue, Xiaoyang, He, Linhong
Published in Molecular diversity (06.05.2024)
Published in Molecular diversity (06.05.2024)
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Discovery of (R)-5-(benzo[d][1,3]dioxol-5-yl)-7-((1-(vinylsulfonyl)pyrrolidin-2-yl)methyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine (B6) as a potent Bmx inhibitor for the treatment of NSCLC
He, Linhong, Li, Da, Zhang, Chufeng, Bai, Peng, Chen, Lijuan
Published in Bioorganic & medicinal chemistry letters (01.09.2017)
Published in Bioorganic & medicinal chemistry letters (01.09.2017)
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Journal Article
A novel filtering patch antenna with high selectivity and wide out‐of‐band suppression
Zhang, Zihui, Jiao, Yong‐Chang, Hui, Caitao, He, Linhong
Published in Microwave and optical technology letters (01.07.2024)
Published in Microwave and optical technology letters (01.07.2024)
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Journal Article
Design and synthesis of highly selective Janus kinase 3 covalent inhibitors for the treatment of rheumatoid arthritis
Yao, Hualiang, Zhang, Jie, Zheng, Qisheng, Zeng, Xianxia, Huang, Huaizheng, Ling, Zhen, Tang, Minghai, Chen, Zhiquan, Wang, Wenchu, He, Linhong
Published in Archiv der Pharmazie (Weinheim) (01.06.2024)
Published in Archiv der Pharmazie (Weinheim) (01.06.2024)
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Structure-based design, synthesis and in vitro antiproliferative effects studies of novel dual BRD4/HDAC inhibitors
Shao, Mingfeng, He, Linhong, Zheng, Li, Huang, Lingxiao, Zhou, Yuanyuan, Wang, Taijing, Chen, Yong, Shen, Mingsheng, Wang, Fang, Yang, Zhuang, Chen, Lijuan
Published in Bioorganic & medicinal chemistry letters (01.09.2017)
Published in Bioorganic & medicinal chemistry letters (01.09.2017)
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Structural exploration, synthesis and pharmacological evaluation of novel 5-benzylidenethiazolidine-2,4-dione derivatives as iNOS inhibitors against inflammatory diseases
Ma, Liang, Pei, Heying, Lei, Lei, He, Linhong, Chen, Jinying, Liang, Xiaolin, Peng, Aihua, Ye, Haoyu, Xiang, Mingli, Chen, Lijuan
Published in European journal of medicinal chemistry (06.03.2015)
Published in European journal of medicinal chemistry (06.03.2015)
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Journal Article
Design, synthesis and biological evaluation of 4-anilinoquinoline derivatives as novel potent tubulin depolymerization agents
Zhou, Yuanyuan, Yan, Wei, Cao, Dong, Shao, Mingfeng, Li, Dan, Wang, Fang, Yang, Zhuang, Chen, Yong, He, Linhong, Wang, Taijin, Shen, Mingsheng, Chen, Lijuan
Published in European journal of medicinal chemistry (29.09.2017)
Published in European journal of medicinal chemistry (29.09.2017)
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Journal Article
Design, synthesis and biological evaluation of 7H-pyrrolo[2,3-d]pyrimidin-4-amine derivatives as selective Btk inhibitors with improved pharmacokinetic properties for the treatment of rheumatoid arthritis
He, Linhong, Pei, Heying, Zhang, Chufeng, Shao, Mingfeng, Li, Dan, Tang, Mingli, Wang, Taijing, Chen, Xiaoxin, Xiang, Mingli, Chen, Lijuan
Published in European journal of medicinal chemistry (10.02.2018)
Published in European journal of medicinal chemistry (10.02.2018)
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Journal Article
Structural optimizations on the 7H-pyrrolo[2,3-d]pyrimidine scaffold to develop highly selective, safe and potent JAK3 inhibitors for the treatment of Rheumatoid arthritis
He, Linhong, Zhang, Jie, Ling, Zhen, Zeng, Xianxia, Yao, Hualiang, Tang, Minghai, Huang, Huaizheng, Xie, Xin, Qin, Tinsheng, Feng, Xianjing, Chen, Zhiquan, Deng, Fengyuan, Yue, Xiaoyang
Published in Bioorganic chemistry (01.08.2024)
Published in Bioorganic chemistry (01.08.2024)
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Journal Article
Structural optimizations on the 7H-pyrrolo2,3-dpyrimidine scaffold to develop highly selective, safe and potent JAK3 inhibitors for the treatment of Rheumatoid arthritis
He, Linhong, Zhang, Jie, Ling, Zhen, Zeng, Xianxia, Yao, Hualiang, Tang, Minghai, Huang, Huaizheng, Xie, Xin, Qin, Tinsheng, Feng, Xianjing, Chen, Zhiquan, Deng, Fengyuan, Yue, Xiaoyang
Published in Bioorganic chemistry (01.08.2024)
Published in Bioorganic chemistry (01.08.2024)
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Journal Article
Discovery of 5-methyl-2-(4-((4-(methylsulfonyl)benzyl)oxy)phenyl)-4-(piperazin-1-yl)pyrimidine derivatives as novel GRP119 agonists for the treatment of diabetes and obesity
Chen, Jinying, Sang, Zitai, Li, Lu, He, Linhong, Ma, Liang
Published in Molecular diversity (01.08.2017)
Published in Molecular diversity (01.08.2017)
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Journal Article
Discovery of a highly selective JAK3 inhibitor for the treatment of rheumatoid arthritis
Pei, Heying, He, Linhong, Shao, Mingfeng, Yang, Zhuang, Ran, Yan, Li, Dan, Zhou, Yuanyuan, Tang, Minghai, Wang, Taijin, Gong, Yanqiu, Chen, Xiaoxin, Yang, Shengyong, Xiang, Mingli, Chen, Lijuan
Published in Scientific reports (27.03.2018)
Published in Scientific reports (27.03.2018)
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