Distinct effects of the antiestrogen Faslodex on the stability of estrogen receptors-alpha and -beta in the breast cancer cell line MCF-7
Peekhaus, NT, Chang, T, Hayes, EC, Wilkinson, HA, Mitra, SW, Schaeffer, JM, Rohrer, SP
Published in Journal of molecular endocrinology (01.06.2004)
Published in Journal of molecular endocrinology (01.06.2004)
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Rapid Identification of Subtype-Selective Agonists of the Somatostatin Receptor Through Combinatorial Chemistry
Rohrer, Susan P., Birzin, Elizabeth T., Mosley, Ralph T., Berk, Scott C., Hutchins, Steven M., Shen, Dong-Ming, Xiong, Yusheng, Hayes, Edward C., Parmar, Rupa M., Foor, Forrest, Mitra, Sudha W., Degrado, Sylvia J., Shu, Min, Klopp, John M., Cai, Sheng-Jian, Blake, Allan, Wanda W. S. Chan, Pasternak, Alex, Yang, Lihu, Patchett, Arthur A., Smith, Roy G., Chapman, Kevin T., Schaeffer, James M.
Published in Science (American Association for the Advancement of Science) (23.10.1998)
Published in Science (American Association for the Advancement of Science) (23.10.1998)
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TriCalm(®) hydrogel is significantly superior to 2% diphenhydramine and 1% hydrocortisone in reducing the peak intensity, duration, and overall magnitude of cowhage-induced itch
Papoiu, Alexandru Dp, Chaudhry, Hunza, Hayes, Erin C, Chan, Yiong-Huak, Herbst, Kenneth D
Published in Clinical, cosmetic and investigational dermatology (01.01.2015)
Published in Clinical, cosmetic and investigational dermatology (01.01.2015)
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Estrogen receptor ligands. Part 9: Dihydrobenzoxathiin SERAMs with alkyl substituted pyrrolidine side chains and linkers
Blizzard, Timothy A., DiNinno, Frank, Morgan, Jerry D., Chen, Helen Y., Wu, Jane Y., Kim, Seongkon, Chan, Wanda, Birzin, Elizabeth T., Yang, Yi Tien, Pai, Lee-Yuh, Fitzgerald, Paula M.D., Sharma, Nandini, Li, Ying, Zhang, Zhoupeng, Hayes, Edward C., DaSilva, Carolyn A., Tang, Wei, Rohrer, Susan P., Schaeffer, James M., Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (03.01.2005)
Published in Bioorganic & medicinal chemistry letters (03.01.2005)
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The discovery of tetrahydrofluorenones as a new class of estrogen receptor β-subtype selective ligands
Wilkening, R.R., Ratcliffe, R.W., Tynebor, E.C., Wildonger, K.J., Fried, A.K., Hammond, M.L., Mosley, R.T., Fitzgerald, P.M.D., Sharma, N., McKeever, B.M., Nilsson, S., Carlquist, M., Thorsell, A., Locco, L., Katz, R., Frisch, K., Birzin, E.T., Wilkinson, H.A., Mitra, S., Cai, S., Hayes, E.C., Schaeffer, J.M., Rohrer, S.P.
Published in Bioorganic & medicinal chemistry letters (01.07.2006)
Published in Bioorganic & medicinal chemistry letters (01.07.2006)
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Estrogen receptor ligands. Part 10: Chromanes: old scaffolds for new SERAMs
Tan, Qiang, Blizzard, Timothy A., Morgan, Jerry D., Birzin, Elizabeth T., Chan, Wanda, Yang, Yi Tien, Pai, Lee-Yuh, Hayes, Edward C., DaSilva, Carolyn A., Warrier, Sudha, Yudkovitz, Joel, Wilkinson, Hilary A., Sharma, Nandini, Fitzgerald, Paula M.D., Li, Susan, Colwell, Lawrence, Fisher, John E., Adamski, Sharon, Reszka, Alfred A., Kimmel, Donald, DiNinno, Frank, Rohrer, Susan P., Freedman, Leonard P., Schaeffer, James M., Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (15.03.2005)
Published in Bioorganic & medicinal chemistry letters (15.03.2005)
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Synthesis and Biological Activities of Potent Peptidomimetics Selective for Somatostatin Receptor Subtype 2
Yang, Lihu, Berk, Scott C., Rohrer, Susan P., Mosley, Ralph T., Guo, Liangqin, Underwood, Dennis J., Arison, Byron H., Birzin, Elizabeth T., Hayes, Edward C., Mitra, Sudha W., Parmar, Rupa M., Cheng, Kang, Wu, Tsuei-Ju, Butler, Bridgette S., Foor, Forrest, Pasternak, Alexander, Pan, Yanping, Silva, Maria, Freidinger, Roger M., Smith, Roy G., Chapman, Kevin, Schaeffer, James M., Patchett, Arthur A.
Published in Proceedings of the National Academy of Sciences - PNAS (01.09.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (01.09.1998)
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Estrogen receptor ligands. Part 13: Dihydrobenzoxathiin SERAMs with an optimized antagonist side chain
Blizzard, Timothy A., DiNinno, Frank, Chen, Helen Y., Kim, Seongkon, Wu, Jane Y., Chan, Wanda, Birzin, Elizabeth T., Yang, Yi Tien, Pai, Lee-Yuh, Hayes, Edward C., DaSilva, Carolyn A., Rohrer, Susan P., Schaeffer, James M., Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (01.09.2005)
Published in Bioorganic & medicinal chemistry letters (01.09.2005)
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Estrogen receptor ligands. Part 11: Synthesis and activity of isochromans and isothiochromans
Liu, Jian, Birzin, Elizabeth T., Chan, Wanda, Yang, Yi Tien, Pai, Lee-Yuh, DaSilva, Carolyn, Hayes, Edward C., Mosley, Ralph T., DiNinno, Frank, Rohrer, Susan P., Schaeffer, James M., Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
Published in Bioorganic & medicinal chemistry letters (01.02.2005)
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Estrogen receptor ligands. Part 7: Dihydrobenzoxathiin SERAMs with bicyclic amine side chains
Blizzard, Timothy A, DiNinno, Frank, Morgan, Jerry D, Chen, Helen Y, Wu, Jane Y, Gude, Candido, Kim, Seongkon, Chan, Wanda, Birzin, Elizabeth T, Tien Yang, Yi, Pai, Lee-Yuh, Zhang, Zhoupeng, Hayes, Edward C, DaSilva, Carolyn A, Tang, Wei, Rohrer, Susan P, Schaeffer, James M, Hammond, Milton L
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
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Estrogen receptor ligands. Part 14: Application of novel antagonist side chains to existing platforms
Blizzard, Timothy A., Morgan, Jerry D., Chan, Wanda, Birzin, Elizabeth T., Pai, Lee-Yuh, Hayes, Edward C., DaSilva, Carolyn A., Mosley, Ralph T., Yang, Yi Tien, Rohrer, Susan P., DiNinno, Frank, Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
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Estrogen receptor ligands. Part 8: Dihydrobenzoxathiin SERAMs with heteroatom-substituted side chains
Blizzard, Timothy A, DiNinno, Frank, Morgan, Jerry D, Wu, Jane Y, Chen, Helen Y, Kim, Seongkon, Chan, Wanda, Birzin, Elizabeth T, Yang, Yi Tien, Pai, Lee-Yuh, Zhang, Zhoupeng, Hayes, Edward C, DaSilva, Carolyn A, Tang, Wei, Rohrer, Susan P, Schaeffer, James M, Hammond, Milton L
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
Published in Bioorganic & medicinal chemistry letters (02.08.2004)
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Estrogen receptor ligands. Part 5: The SAR of dihydrobenzoxathiins containing modified basic side chains
QIANG TAN, BIRZIN, Elizabeth T, HAMMOND, Milton L, WANDA CHAN, YI TIEN YANG, PAI, Lee-Yuh, HAYES, Edward C, DASILVA, Carolyn A, DININNO, Frank, ROHRER, Susan P, SCHAEFFER, James M
Published in Bioorganic & medicinal chemistry letters (16.07.2004)
Published in Bioorganic & medicinal chemistry letters (16.07.2004)
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Estrogen receptor ligands. Part 6: Synthesis and binding affinity of dihydrobenzodithiins
QIANG TAN, BIRZIN, Elizabeth T, HAMMOND, Milton L, CHAN, Wanda, YI TIEN YANG, PAI, Lee-Yuh, HAYES, Edward C, DASILVA, Carolyn A, DININNO, Frank, ROHRER, Susan P, SCHAEFFER, James M
Published in Bioorganic & medicinal chemistry letters (16.07.2004)
Published in Bioorganic & medicinal chemistry letters (16.07.2004)
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Nonpeptidyl Somatostatin Agonists Demonstrate That sst2 and sst5 Inhibit Stimulated Growth Hormone Secretion from Rat Anterior Pituitary Cells
Parmar, R.M., Chan, W.W.-S., Dashkevicz, M., Hayes, E.C., Rohrer, S.P., Smith, R.G., Schaeffer, J.M., Blake, A.D.
Published in Biochemical and biophysical research communications (24.09.1999)
Published in Biochemical and biophysical research communications (24.09.1999)
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Peptide leukotriene release after antigen challenge in patients sensitive to ragweed
Creticos, P.S, Peters, S.P, Adkinson, N.F. Jr, Naclerio, R.M
Published in The New England journal of medicine (21.06.1984)
Published in The New England journal of medicine (21.06.1984)
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