Synthesis of N-Substituted 4-(4-Hydroxyphenyl)piperidines, 4-(4-Hydroxybenzyl)piperidines, and (±)-3-(4-Hydroxyphenyl)pyrrolidines: Selective Antagonists at the 1a/2B NMDA Receptor Subtype
Guzikowski, Anthony P, Tamiz, Amir P, Acosta-Burruel, Manuel, Hong-Bae, Soo, Cai, Sui Xiong, Hawkinson, Jon E, Keana, John F. W, Kesten, Suzanne R, Shipp, Christina T, Tran, Minhtam, Whittemore, Edward R, Woodward, Richard M, Wright, Jon L, Zhou, Zhang-Lin
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Published in Journal of medicinal chemistry (09.03.2000)
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Anxiolytic and anticonvulsant activity of a synthetic neuroactive steroid Co 3-0593
WIELAND, S, BELLUZZI, J, HAWKINSON, J. E, HOGENKAMP, D, UPASANI, R, STEIN, L, WOOD, P. L, GEE, K. W, LAN, N. C
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Published in Psychopharmacologia (01.11.1997)
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Synthesis and Structure−Activity Relationships of 1,2,3,4-Tetrahydroquinoline-2,3,4-trione 3-Oximes: Novel and Highly Potent Antagonists for NMDA Receptor Glycine Site
Cai, Sui Xiong, Zhou, Zhang-Lin, Huang, Jin-Cheng, Whittemore, Edward R, Egbuwoku, Zizi O, Lü, Yixin, Hawkinson, Jon E, Woodward, Richard M, Weber, Eckard, Keana, John F. W
Published in Journal of medicinal chemistry (16.08.1996)
Published in Journal of medicinal chemistry (16.08.1996)
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Structure−Activity Relationships of Alkyl- and Alkoxy-Substituted 1,4-Dihydroquinoxaline-2,3-diones: Potent and Systemically Active Antagonists for the Glycine Site of the NMDA Receptor
Cai, Sui Xiong, Kher, Sunil M, Zhou, Zhang-Lin, Ilyin, Victor, Espitia, Stephen A, Tran, Minhtam, Hawkinson, Jon E, Woodward, Richard M, Weber, Eckard, Keana, John F. W
Published in Journal of medicinal chemistry (28.02.1997)
Published in Journal of medicinal chemistry (28.02.1997)
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4-Hydroxy-1-[2-(4-hydroxyphenoxy)ethyl]-4-(4-methylbenzyl)piperidine: A Novel, Potent, and Selective NR1/2B NMDA Receptor Antagonist
Zhou, Zhang-Lin, Cai, Sui Xiong, Whittemore, Edward R, Konkoy, Christopher S, Espitia, Stephen A, Tran, Minhtam, Rock, David M, Coughenour, Linda L, Hawkinson, Jon E, Boxer, Peter A, Bigge, Christopher F, Wise, Lawrence D, Weber, Eckard, Woodward, Richard M, Keana, John F. W
Published in Journal of medicinal chemistry (29.07.1999)
Published in Journal of medicinal chemistry (29.07.1999)
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5-(N-Oxyaza)-7-substituted-1,4-dihydroquinoxaline-2,3-diones: Novel, Systemically Active and Broad Spectrum Antagonists for NMDA/glycine, AMPA, and Kainate Receptors
Cai, Sui Xiong, Huang, Jin-Cheng, Espitia, Stephen A, Tran, Minhtam, Ilyin, Victor I, Hawkinson, Jon E, Woodward, Richard M, Weber, Eckard, Keana, John F. W
Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
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Novel phosphoserine phosphatase inhibitors
Hawkinson, Jon E, Acosta-Burruel, Manuel, Ta, Nahn D, Wood, Paul L
Published in European journal of pharmacology (22.10.1997)
Published in European journal of pharmacology (22.10.1997)
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Subtype-Selective N-Methyl-d-aspartate Receptor Antagonists: Synthesis and Biological Evaluation of 1-(Arylalkynyl)-4-benzylpiperidines
Wright, Jon L, Gregory, Tracy F, Bigge, Christopher F, Boxer, Peter A, Serpa, Kevin, Meltzer, Leonard T, Wise, Lawrence D, Cai, Sui Xiong, Hawkinson, Jon E, Konkoy, Christopher S, Whittemore, Edward R, Woodward, Richard M, Zhou, Zhang-Lin
Published in Journal of medicinal chemistry (01.07.1999)
Published in Journal of medicinal chemistry (01.07.1999)
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Analogs of 3-Hydroxy-1H-1-benzazepine-2,5-dione: Structure−Activity Relationship at N-Methyl-d-aspartate Receptor Glycine Sites
Guzikowski, Anthony P, Cai, Sui Xiong, Espitia, Stephen A, Hawkinson, Jon E, Huettner, James E, Nogales, Daniel F, Tran, Minhtam, Woodward, Richard M, Weber, Eckard, Keana, John F. W
Published in Journal of medicinal chemistry (08.11.1996)
Published in Journal of medicinal chemistry (08.11.1996)
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Structure−Activity Relationships of 4-Hydroxy-3-nitroquinolin-2(1H)-ones as Novel Antagonists at the Glycine Site of N-Methyl-d-aspartate Receptors
Cai, Sui Xiong, Zhou, Zhang-Lin, Huang, Jin-Cheng, Whittemore, Edward R, Egbuwoku, Zizi O, Hawkinson, Jon E, Woodward, Richard M, Weber, Eckard, Keana, John F. W
Published in Journal of medicinal chemistry (08.11.1996)
Published in Journal of medicinal chemistry (08.11.1996)
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Selective actions of certain neuroactive pregnanediols at the gamma-aminobutyric acid type A receptor complex in rat brain
McCauley, L D, Liu, V, Chen, J S, Hawkinson, J E, Lan, N C, Gee, K W
Published in Molecular pharmacology (01.02.1995)
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Published in Molecular pharmacology (01.02.1995)
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Characterization of the anticonvulsant properties of ganaxolone (CCD 1042; 3alpha-hydroxy-3beta-methyl-5alpha-pregnan-20-one), a selective, high-affinity, steroid modulator of the gamma-aminobutyric acid(A) receptor
Carter, R B, Wood, P L, Wieland, S, Hawkinson, J E, Belelli, D, Lambert, J J, White, H S, Wolf, H H, Mirsadeghi, S, Tahir, S H, Bolger, M B, Lan, N C, Gee, K W
Published in The Journal of pharmacology and experimental therapeutics (01.03.1997)
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Published in The Journal of pharmacology and experimental therapeutics (01.03.1997)
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Correlation of neuroactive steroid modulation of [35S]t-butylbicyclophosphorothionate and [3H]flunitrazepam binding and gamma-aminobutyric acidA receptor function
Hawkinson, J E, Kimbrough, C L, Belelli, D, Lambert, J J, Purdy, R H, Lan, N C
Published in Molecular pharmacology (01.11.1994)
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Published in Molecular pharmacology (01.11.1994)
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Photoaffinity ligands for the [3H]TBOB binding site of the GABAA receptor
Hawkinson, J E, Goeldner, M P, Palmer, C J, Casida, J E
Published in Journal of receptor research (1991)
Published in Journal of receptor research (1991)
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