Design of a Supersoft Topical JAK Inhibitor, Which Is Effective in Human Skin but Rapidly Deactivated in Blood
Thoma, Gebhard, Decoret, Odile, Vangrevelinghe, Eric, Trunzer, Markus, Decker, Andrea, Orjuela Leon, Anette, Beerli, Christian, Bruno, Sandro, Hauchard, Alice, Paulat, Guido, Zerwes, Hans-Guenter, Hacini-Rachinel, Feriel
Published in Journal of medicinal chemistry (09.11.2023)
Published in Journal of medicinal chemistry (09.11.2023)
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Journal Article
Discovery and Characterization of the Topical Soft JAK Inhibitor CEE321 for Atopic Dermatitis
Thoma, Gebhard, Duthaler, Rudolf O., Waelchli, Rudolf, Hauchard, Alice, Bruno, Sandro, Strittmatter-Keller, Ulrike, Orjuela Leon, Anette, Viebrock, Sabine, Aichholz, Reiner, Beltz, Karen, Grove, Kerri, Hoque, Shaila, Rudewicz, Patrick J., Zerwes, Hans-Guenter
Published in Journal of medicinal chemistry (09.02.2023)
Published in Journal of medicinal chemistry (09.02.2023)
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Adriforant is a functional antagonist of histamine receptor 4 and attenuates itch and skin inflammation in mice
Uluckan, Özge, Bruno, Sandro, Wang, Yichen, Wack, Nathalie, Wilzopolski, Jenny, Goetschy, Jean-Francois, Delucis-Bronn, Corinne, Urban, Beatrice, Fehlmann, Dominique, Stark, Holger, Hauchard, Alice, Roussel, Elsa, Kempf, Dominique, Kaupmann, Klemens, Raulf, Friedrich, Bäumer, Wolfgang, Röhn, Till A., Zerwes, Hans Günter
Published in European journal of pharmacology (15.04.2023)
Published in European journal of pharmacology (15.04.2023)
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Modelling atopic dermatitis in healthy human skin for the characterization of topical compounds
Hacini‐Rachinel, Feriel, Hauchard, Alice, Bruno, Sandro, Paulat, Guido, Cojean, Celine, Loesle, Perrine, Schneider, Martin Alexander, Bourne, Marta, Elain, Gaelle, Roth, Lukas, Urban, Beatrice, Viebrock, Sabine, Leon, Anette Orjuela, Roehn, Till A., Loesche, Christian, Werfel, Thomas, Thoma, Gebhard, Zerwes, Hans‐Günter
Published in Experimental dermatology (01.05.2024)
Published in Experimental dermatology (01.05.2024)
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