Inhibiting Acetylcholinesterase to Activate Pleiotropic Prodrugs with Therapeutic Interest in Alzheimer's Disease
Toublet, François-Xavier, Lecoutey, Cédric, Lalut, Julien, Hatat, Bérénice, Davis, Audrey, Since, Marc, Corvaisier, Sophie, Freret, Thomas, Sopkova de Oliveira Santos, Jana, Claeysen, Sylvie, Boulouard, Michel, Dallemagne, Patrick, Rochais, Christophe
Published in Molecules (Basel, Switzerland) (31.07.2019)
Published in Molecules (Basel, Switzerland) (31.07.2019)
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Journal Article
Pleiotropic prodrugs: Design of a dual butyrylcholinesterase inhibitor and 5-HT6 receptor antagonist with therapeutic interest in Alzheimer’s disease
Toublet, François-Xavier, Lalut, Julien, Hatat, Bérénice, Lecoutey, Cédric, Davis, Audrey, Since, Marc, Corvaisier, Sophie, Freret, Thomas, Sopková-de Oliveira Santos, Jana, Claeysen, Sylvie, Boulouard, Michel, Dallemagne, Patrick, Rochais, Christophe
Published in European journal of medicinal chemistry (15.01.2021)
Published in European journal of medicinal chemistry (15.01.2021)
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A Novel in vivo Anti-amnesic Agent, Specially Designed to Express Both Acetylcholinesterase (AChE) Inhibitory, Serotonergic Subtype 4 Receptor (5-HT 4 R) Agonist and Serotonergic Subtype 6 Receptor (5-HT 6 R) Inverse Agonist Activities, With a Potential Interest Against Alzheimer's Disease
Hatat, Bérénice, Yahiaoui, Samir, Lecoutey, Cédric, Davis, Audrey, Freret, Thomas, Boulouard, Michel, Claeysen, Sylvie, Rochais, Christophe, Dallemagne, Patrick
Published in Frontiers in aging neuroscience (19.06.2019)
Published in Frontiers in aging neuroscience (19.06.2019)
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Journal Article
Vertigoheel improves central vestibular compensation after unilateral peripheral vestibulopathy in rats
Hatat, Bérénice, Boularand, Romain, Bringuier, Claire, Chanut, Nicolas, Besnard, Stéphane, Mueller, Andrea M., Weyer, Kathrin, Seilheimer, Bernd, Tighilet, Brahim, Chabbert, Christian
Published in Frontiers in neurology (23.09.2022)
Published in Frontiers in neurology (23.09.2022)
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Journal Article
Effect of Fluoxetine and Acacetin on Central Vestibular Compensation in an Animal Model of Unilateral Peripheral Vestibulopathy
Hatat, Bérénice, Boularand, Romain, Bringuier, Claire, Chanut, Nicolas, Chabbert, Christian, Tighilet, Brahim
Published in Biomedicines (27.08.2022)
Published in Biomedicines (27.08.2022)
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Journal Article
Novel multi target-directed ligands targeting 5-HT4 receptors with in cellulo antioxidant properties as promising leads in Alzheimer's disease
Lanthier, Caroline, Payan, Hugo, Liparulo, Irene, Hatat, Bérénice, Lecoutey, Cédric, Since, Marc, Davis, Audrey, Bergamini, Christian, Claeysen, Sylvie, Dallemagne, Patrick, Bolognesi, Maria-Laura, Rochais, Christophe
Published in European journal of medicinal chemistry (15.11.2019)
Published in European journal of medicinal chemistry (15.11.2019)
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Journal Article
Vertigoheel improves central vestibular compensation after unilateral peripheral vestibulopathy in rats
Hatat, Bérénice, Boularand, Romain, Bringuier, Claire, Chanut, Nicolas, Besnard, Stéphane, Mueller, Andrea, Weyer, Kathrin, Seilheimer, Bernd, Tighilet, Brahim, Chabbert, Christian
Published in Frontiers in neurology (2022)
Published in Frontiers in neurology (2022)
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Journal Article
Effect of Fluoxetine and Acacetin on Central Vestibular Compensation in an Animal Model of Unilateral Peripheral Vestibulopathy
Hatat, Bérénice, Boularand, Romain, Bringuier, Claire, Chanut, Nicolas, Chabbert, Christian, Tighilet, Brahim
Published in Biomedicines (27.08.2022)
Published in Biomedicines (27.08.2022)
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Journal Article
Pleiotropic prodrugs: Design of a dual butyrylcholinesterase inhibitor and 5-HT 6 receptor antagonist with therapeutic interest in Alzheimer's disease
Toublet, François-Xavier, Lalut, Julien, Hatat, Bérénice, Lecoutey, Cédric, Davis, Audrey, Since, Marc, Corvaisier, Sophie, Freret, Thomas, Sopková-de Oliveira Santos, Jana, Claeysen, Sylvie, Boulouard, Michel, Dallemagne, Patrick, Rochais, Christophe
Published in European journal of medicinal chemistry (15.01.2021)
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Published in European journal of medicinal chemistry (15.01.2021)
Journal Article
Novel multi target-directed ligands targeting 5-HT 4 receptors with in cellulo antioxidant properties as promising leads in Alzheimer's disease
Lanthier, Caroline, Payan, Hugo, Liparulo, Irene, Hatat, Bérénice, Lecoutey, Cédric, Since, Marc, Davis, Audrey, Bergamini, Christian, Claeysen, Sylvie, Dallemagne, Patrick, Bolognesi, Maria-Laura, Rochais, Christophe
Published in European journal of medicinal chemistry (06.08.2019)
Get full text
Published in European journal of medicinal chemistry (06.08.2019)
Journal Article