Development of a Novel Lead that Targets M. tuberculosis Polyketide Synthase 13
Aggarwal, Anup, Parai, Maloy K., Shetty, Nishant, Wallis, Deeann, Woolhiser, Lisa, Hastings, Courtney, Dutta, Noton K., Galaviz, Stacy, Dhakal, Ramesh C., Shrestha, Rupesh, Wakabayashi, Shoko, Walpole, Chris, Matthews, David, Floyd, David, Scullion, Paul, Riley, Jennifer, Epemolu, Ola, Norval, Suzanne, Snavely, Thomas, Robertson, Gregory T., Rubin, Eric J., Ioerger, Thomas R., Sirgel, Frik A., van der Merwe, Ruben, van Helden, Paul D., Keller, Peter, Böttger, Erik C., Karakousis, Petros C., Lenaerts, Anne J., Sacchettini, James C.
Published in Cell (13.07.2017)
Published in Cell (13.07.2017)
Get full text
Journal Article
Comparative Analysis of Pharmacodynamics in the C3HeB/FeJ Mouse Tuberculosis Model for DprE1 Inhibitors TBA-7371, PBTZ169, and OPC-167832
Robertson, Gregory T, Ramey, Michelle E, Massoudi, Lisa M, Carter, Claire L, Zimmerman, Matt, Kaya, Firat, Graham, Barbara G, Gruppo, Veronica, Hastings, Courtney, Woolhiser, Lisa K, Scott, Dashick W L, Asay, Bryce C, Eshun-Wilson, Franceen, Maidj, Ekaterina, Podell, Brendan K, Vásquez, Joshua J, Lyons, Mike A, Dartois, Véronique, Lenaerts, Anne J
Published in Antimicrobial agents and chemotherapy (18.10.2021)
Published in Antimicrobial agents and chemotherapy (18.10.2021)
Get full text
Journal Article
Pyrazolo[1,5‑a]pyridine Inhibitor of the Respiratory Cytochrome bcc Complex for the Treatment of Drug-Resistant Tuberculosis
Lu, Xiaoyun, Williams, Zoe, Hards, Kiel, Tang, Jian, Cheung, Chen-Yi, Aung, Htin Lin, Wang, Bangxing, Liu, Zhiyong, Hu, Xianglong, Lenaerts, Anne, Woolhiser, Lisa, Hastings, Courtney, Zhang, Xiantao, Wang, Zhe, Rhee, Kyu, Ding, Ke, Zhang, Tianyu, Cook, Gregory M
Published in ACS infectious diseases (08.02.2019)
Published in ACS infectious diseases (08.02.2019)
Get full text
Journal Article
Spectinamides are effective partner agents for the treatment of tuberculosis in multiple mouse infection models
Robertson, Gregory T, Scherman, Michael S, Bruhn, David F, Liu, Jiuyu, Hastings, Courtney, McNeil, Michael R, Butler, Michelle M, Bowlin, Terry L, Lee, Robin B, Lee, Richard E, Lenaerts, Anne J
Published in Journal of antimicrobial chemotherapy (01.03.2017)
Published in Journal of antimicrobial chemotherapy (01.03.2017)
Get full text
Journal Article
Enzyme-Like Catalysis of the Nazarov Cyclization by Supramolecular Encapsulation
Hastings, Courtney, Pluth, Michael, Bergman, Robert, Raymond, Kenneth
Published in Journal of the American Chemical Society (29.03.2010)
Published in Journal of the American Chemical Society (29.03.2010)
Get full text
Journal Article
Discovery of a cofactor-independent inhibitor of Mycobacterium tuberculosis InhA
Xia, Yi, Zhou, Yasheen, Carter, David S, McNeil, Matthew B, Choi, Wai, Halladay, Jason, Berry, Pamela W, Mao, Weimin, Hernandez, Vincent, O'Malley, Theresa, Korkegian, Aaron, Sunde, Bjorn, Flint, Lindsay, Woolhiser, Lisa K, Scherman, Michael S, Gruppo, Veronica, Hastings, Courtney, Robertson, Gregory T, Ioerger, Thomas R, Sacchettini, Jim, Tonge, Peter J, Lenaerts, Anne J, Parish, Tanya, Alley, Mrk
Published in Life science alliance (01.06.2018)
Published in Life science alliance (01.06.2018)
Get full text
Journal Article
Spectinamide MBX-4888A exhibits favorable lesion and tissue distribution and promotes treatment shortening in advanced murine models of tuberculosis
Bauman, Allison A, Sarathy, Jansy P, Kaya, Firat, Massoudi, Lisa M, Scherman, Michael S, Hastings, Courtney, Liu, Jiuyu, Xie, Min, Brooks, Elizabeth J, Ramey, Michelle E, Jones, Isabelle L, Benedict, Noalani D, Maclaughlin, Madelyn R, Miller-Dawson, Jake A, Waidyarachchi, Samanthi L, Butler, Michelle M, Bowlin, Terry L, Zimmerman, Matthew D, Lenaerts, Anne J, Meibohm, Bernd, Gonzalez-Juarrero, Mercedes, Lyons, Michael A, Dartois, Véronique, Lee, Richard E, Robertson, Gregory T
Published in bioRxiv (13.05.2024)
Published in bioRxiv (13.05.2024)
Get full text
Journal Article
Spectinamide MBX-4888A exhibits favorable lesion and tissue distribution and promotes treatment shortening in advanced murine models of tuberculosis
Bauman, Allison A, Sarathy, Jansy P, Kaya, Firat, Massoudi, Lisa M, Scherman, Michael S, Hastings, Courtney, Liu, Jiuyu, Xie, Min, Brooks, Elizabeth J, Ramey, Michelle E, Jones, Isabelle L, Benedict, Noalani D, Maclaughlin, Madelyn R, Miller-Dawson, Jake A, Waidyarachchi, Samanthi L, Butler, Michelle M, Bowlin, Terry L, Zimmerman, Matthew D, Lenaerts, Anne J, Meibohm, Bernd, Gonzalez-Juarrero, Mercedes, Lyons, Michael A, Dartois, Véronique, Lee, Richard E, Robertson, Gregory T
Published in bioRxiv : the preprint server for biology (13.05.2024)
Get more information
Published in bioRxiv : the preprint server for biology (13.05.2024)
Journal Article
ChemInform Abstract: Simultaneously Bound Guests and Chiral Recognition: A Chiral Self-Assembled Supramolecular Host Encapsulates Hydrophobic Guests
Hastings, Courtney J., Pluth, Michael D., Biros, Shannon M., Bergman, Robert G., Raymond, Kenneth N.
Published in ChemInform (04.11.2008)
Published in ChemInform (04.11.2008)
Get full text
Journal Article