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Hašková, Pavlína, Applová, Lenka, Jansová, Hana, Homola, Pavel, Franz, Katherine J, Vávrová, Kateřina, Roh, Jaroslav, Šimůnek, Tomáš
Published in Scientific reports (13.06.2022)
Published in Scientific reports (13.06.2022)
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Aroylhydrazone iron chelators: Tuning antioxidant and antiproliferative properties by hydrazide modifications
Hrušková, Kateřina, Potůčková, Eliška, Hergeselová, Tereza, Liptáková, Lucie, Hašková, Pavlína, Mingas, Panagiotis, Kovaříková, Petra, Šimůnek, Tomáš, Vávrová, Kateřina
Published in European journal of medicinal chemistry (14.09.2016)
Published in European journal of medicinal chemistry (14.09.2016)
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Structure–Activity Relationships of Nitro-Substituted Aroylhydrazone Iron Chelators with Antioxidant and Antiproliferative Activities
Hruskova, Katerina, Potuckova, Eliska, Opalka, Lukas, Hergeselova, Tereza, Haskova, Pavlina, Kovarikova, Petra, Simunek, Tomas, Vavrova, Katerina
Published in Chemical research in toxicology (18.06.2018)
Published in Chemical research in toxicology (18.06.2018)
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Structure-activity relationships of novel salicylaldehyde isonicotinoyl hydrazone (SIH) analogs: iron chelation, anti-oxidant and cytotoxic properties
Potůčková, Eliška, Hrušková, Kateřina, Bureš, Jan, Kovaříková, Petra, Špirková, Iva A, Pravdíková, Kateřina, Kolbabová, Lucie, Hergeselová, Tereza, Hašková, Pavlína, Jansová, Hana, Macháček, Miloslav, Jirkovská, Anna, Richardson, Vera, Lane, Darius J R, Kalinowski, Danuta S, Richardson, Des R, Vávrová, Kateřina, Šimůnek, Tomáš
Published in PloS one (13.11.2014)
Published in PloS one (13.11.2014)
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Chronic anthracycline cardiotoxicity: molecular and functional analysis with focus on nuclear factor erythroid 2-related factor 2 and mitochondrial biogenesis pathways
Jirkovsky, Eduard, Popelová, Olga, Kriváková-Stanková, Pavla, Vávrová, Anna, Hroch, Milos, Hasková, Pavlína, Brcáková-Dolezelová, Eva, Micuda, Stanislav, Adamcová, Michaela, Simůnek, Tomás, Cervinková, Zuzana, Gersl, Vladimír, Sterba, Martin
Published in The Journal of pharmacology and experimental therapeutics (01.11.2012)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2012)
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In Vitro Characterization of the Pharmacological Properties of the Anti-Cancer Chelator, Bp4eT, and Its Phase I Metabolites
Potůčková, Eliška, Roh, Jaroslav, Macháček, Miloslav, Sahni, Sumit, Stariat, Ján, Šesták, Vít, Jansová, Hana, Hašková, Pavlína, Jirkovská, Anna, Vávrová, Kateřina, Kovaříková, Petra, Kalinowski, Danuta S, Richardson, Des R, Šimůnek, Tomáš
Published in PloS one (13.10.2015)
Published in PloS one (13.10.2015)
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Comparison of various iron chelators and prochelators as protective agents against cardiomyocyte oxidative injury
Jansová, Hana, Macháček, Miloslav, Wang, Qin, Hašková, Pavlína, Jirkovská, Anna, Potůčková, Eliška, Kielar, Filip, Franz, Katherine J., Šimůnek, Tomáš
Published in Free radical biology & medicine (01.09.2014)
Published in Free radical biology & medicine (01.09.2014)
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Cardioprotective effects of iron chelator HAPI and ROS-activated boronate prochelator BHAPI against catecholamine-induced oxidative cellular injury
Hašková, Pavlína, Jansová, Hana, Bureš, Jan, Macháček, Miloslav, Jirkovská, Anna, Franz, Katherine J, Kovaříková, Petra, Šimůnek, Tomáš, Dr
Published in Toxicology (Amsterdam) (14.09.2016)
Published in Toxicology (Amsterdam) (14.09.2016)
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Iron chelation with salicylaldehyde isonicotinoyl hydrazone protects against catecholamine autoxidation and cardiotoxicity
Haskova, Pavlina, Kovarikova, Petra, Koubkova, Lucie, Vavrova, Anna, Mackova, Eliska, Simunek, Tomas
Published in Free radical biology & medicine (15.02.2011)
Published in Free radical biology & medicine (15.02.2011)
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Characterization of cytoprotective and toxic properties of iron chelator SIH, prochelator BSIH and their degradation products
Jansová, Hana, Bureš, Jan, Macháček, Miloslav, Hašková, Pavlína, Jirkovská, Anna, Roh, Jaroslav, Wang, Qin, Franz, Katherine J, Kovaříková, Petra, Šimůnek, Tomáš
Published in Toxicology (Amsterdam) (28.03.2016)
Published in Toxicology (Amsterdam) (28.03.2016)
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Comparison of various iron chelators used in clinical practice as protecting agents against catecholamine-induced oxidative injury and cardiotoxicity
HASKOVA, Pavlina, KOUBKOVA, Lucie, VAVROVA, Anna, MACKOVA, Eliska, HRUSKOVA, Katefina, KOVARIKOVA, Petra, VAVROVA, Kateřina, SIMUNEK, Tomas
Published in Toxicology (Amsterdam) (18.11.2011)
Published in Toxicology (Amsterdam) (18.11.2011)
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Design, Synthesis, and Biological Evaluation of Isothiosemicarbazones with Antimycobacterial Activity
Novotná, Eva, Waisser, Karel, Kuneš, Jiří, Palát, Karel, Skálová, Lenka, Szotáková, Barbora, Buchta, Vladimír, Stolaříková, Jiřina, Ulmann, Vít, Pávová, Marcela, Weber, Jan, Komrsková, Jitka, Hašková, Pavlína, Vokřál, Ivan, Wsól, Vladimír
Published in Archiv der Pharmazie (Weinheim) (01.08.2017)
Published in Archiv der Pharmazie (Weinheim) (01.08.2017)
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Methyl and ethyl ketone analogs of salicylaldehyde isonicotinoyl hydrazone: Novel iron chelators with selective antiproliferative action
Macková, Eliška, Hrušková, Kateřina, Bendová, Petra, Vávrová, Anna, Jansová, Hana, Hašková, Pavlína, Kovaříková, Petra, Vávrová, Kateřina, Šimůnek, Tomáš
Published in Chemico-biological interactions (30.05.2012)
Published in Chemico-biological interactions (30.05.2012)
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The Novel Iron Chelator, 2-Pyridylcarboxaldehyde 2-Thiophenecarboxyl Hydrazone, Reduces Catecholamine-Mediated Myocardial Toxicity
Mladĕnka, Pr̆emysl, Kalinowski, Danuta S, Hašková, Pavlína, Bobrovová, Zuzana, Hrdina, Radomír, Šimůnek, Tomáš, Nachtigal, Petr, Semecký, Vladimír, Vávrová, Jaroslava, Holečková, Magdaléna, Palicka, Vladimir, Mazurová, Yvona, Jansson, Patric J, Richardson, Des R
Published in Chemical research in toxicology (01.01.2009)
Published in Chemical research in toxicology (01.01.2009)
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In vivo and in vitro assessment of the role of glutathione antioxidant system in anthracycline-induced cardiotoxicity
VAVROVA, Anna, POPELOVA, Olga, STERBA, Martin, JIRKOVSKY, Eduard, HASKOVA, Pavlina, MERTLIKOVA-KAISEROVA, Helena, GERSL, Vladimír, SIMUNEK, Tomáš
Published in Archives of toxicology (01.05.2011)
Published in Archives of toxicology (01.05.2011)
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Intravenous rutin in rat exacerbates isoprenaline-induced cardiotoxicity likely due to intracellular oxidative stress
Filipský, Tomáš, Říha, Michal, Hašková, Pavlína, Pilařová, Veronika, Nováková, Lucie, Semecký, Vladimír, Vávrová, Jaroslava, Holečková, Magdaléna, Palicka, Vladimir, Šimůnek, Tomáš, Hrdina, Radomír, Mladěnka, Přemysl
Published in Redox report : communications in free radical research (04.03.2017)
Published in Redox report : communications in free radical research (04.03.2017)
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HPLC-DAD and MS/MS analysis of novel drug candidates from the group of aromatic hydrazones revealing the presence of geometric isomers
KOVARIKOVA, Petra, VAVROVA, Katerina, TOMALOVA, Katerina, SCHÖNGUT, Michal, HRUSKOVA, Katerina, HALASOVA, Pavlina, KLIMES, Jiri
Published in Journal of pharmaceutical and biomedical analysis (29.09.2008)
Published in Journal of pharmaceutical and biomedical analysis (29.09.2008)
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Conference Proceeding
Protective Effects of D-Penicillamine on Catecholamine-Induced Myocardial Injury
Palicka, Vladimir, Šimůnek, Tomáš, Mladěnka, Přemysl, Homola, Pavel, Holečková, Magdalena, Vávrová, Jaroslava, Váňová, Kateřina, Filipský, Tomáš, Martin, Jan, Hašková, Pavlína, Říha, Michal, Vítek, Libor
Published in Oxidative medicine and cellular longevity (01.01.2016)
Published in Oxidative medicine and cellular longevity (01.01.2016)
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Direct administration of rutin does not protect against catecholamine cardiotoxicity
Mladěnka, Přemysl, Zatloukalová, Libuše, Šimůnek, Tomáš, Bobrovová, Zuzana, Semecký, Vladimír, Nachtigal, Petr, Hašková, Pavlína, Macková, Eliška, Vávrová, Jaroslava, Holečková, Magdaléna, Palicka, Vladimir, Hrdina, Radomír
Published in Toxicology (Amsterdam) (08.01.2009)
Published in Toxicology (Amsterdam) (08.01.2009)
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