Development of human cGAS-specific small-molecule inhibitors for repression of dsDNA-triggered interferon expression
Lama, Lodoe, Adura, Carolina, Xie, Wei, Tomita, Daisuke, Kamei, Taku, Kuryavyi, Vitaly, Gogakos, Tasos, Steinberg, Joshua I, Miller, Michael, Ramos-Espiritu, Lavoisier, Asano, Yasutomi, Hashizume, Shogo, Aida, Jumpei, Imaeda, Toshihiro, Okamoto, Rei, Jennings, Andy J, Michino, Mayako, Kuroita, Takanobu, Stamford, Andrew, Gao, Pu, Meinke, Peter, Glickman, J Fraser, Patel, Dinshaw J, Tuschl, Thomas
Published in Nature communications (21.05.2019)
Published in Nature communications (21.05.2019)
Get full text
Journal Article
Functional-Group-Tolerant Catalytic Migratory Oxidative Coupling of Nitrones
Hashizume, Shogo, Oisaki, Kounosuke, Kanai, Motomu
Published in Chemistry, an Asian journal (01.11.2012)
Published in Chemistry, an Asian journal (01.11.2012)
Get full text
Journal Article
Design and synthesis of 6-methylpyridin-2-one derivatives as novel and potent GluN2A positive allosteric modulators for the treatment of cognitive impairment
Yukawa, Takafumi, Yamashita, Tohru, Imaeda, Toshihiro, Kakei, Hiroyuki, Hashizume, Shogo, Nakamura, Minoru, Daini, Masaki, Okabe, Atsutoshi, Nakashima, Kosuke, Harada, Akina, Narita, Naohiro, Bettini, Ezio, Ugolini, Annarosa, Corsi, Mauro, Hasui, Tomoaki
Published in Bioorganic & medicinal chemistry (01.02.2023)
Published in Bioorganic & medicinal chemistry (01.02.2023)
Get full text
Journal Article
HETEROCYCLIC COMPOUNDS
TAKAMI KAZUAKI, NAKAMURA MINORU, MORIMOTO SHINJI, WANG CHUN XIANG, YAMAGUCHI FUMIE, MIKAMI SATOSHI, IMAEDA TOSHIHIRO, DAINI MASAKI, KAKEI HIROYUKI, HASUI TOMOAKI, YAMASHITA TORU, TAKASHIMA YUKIE, NAKAMURA SHINJI, HASHIZUME SHOGO
Year of Publication 02.12.2021
Get full text
Year of Publication 02.12.2021
Patent
1-((1H-PYRAZOL-4-YL)METHYL)-3-(PHENYL)-1,3-DIHYDRO-2H-IMIDAZOL-2-ONE DERIVATIVES AND RELATED COMPOUNDS AS GPR139 ANTAGONISTS FOR THE TREATMENT OF E.G. DEPRESSION
HASUI, Tomoaki, NAKAMURA, Shinji, TAKAMI, Kazuaki, TAKASHIMA, Sachie, YAMAGUCHI, Fumie, NAKAMURA, Minoru, DAINI, Masaki, YAMASHITA, Toru, IMAEDA, Toshihiro, MIKAMI, Satoshi, KAKEI, Hiroyuki, WANG, Chunxiang, HASHIZUME, Shogo, MORIMOTO, Shinji
Year of Publication 02.11.2023
Get full text
Year of Publication 02.11.2023
Patent
1-((1H-PYRAZOL-4-YL)METHYL)-3-(PHENYL)-1,3-DIHYDRO-2H-IMIDAZOL-2-ONE DERIVATIVES AND RELATED COMPOUNDS AS GPR139 ANTAGONISTS FOR THE TREATMENT OF E.G. DEPRESSION
HASUI, Tomoaki, NAKAMURA, Shinji, TAKAMI, Kazuaki, TAKASHIMA, Sachie, YAMAGUCHI, Fumie, NAKAMURA, Minoru, DAINI, Masaki, YAMASHITA, Toru, IMAEDA, Toshihiro, MIKAMI, Satoshi, KAKEI, Hiroyuki, WANG, Chunxiang, HASHIZUME, Shogo, MORIMOTO, Shinji
Year of Publication 29.03.2023
Get full text
Year of Publication 29.03.2023
Patent
INHIBITORS OF CGAS FOR TREATING AUTOINFLAMMATORY DISEASES AND CANCER METASTASIS
OKAMOTO, Rei, PATEL, Dinshaw, LAMA, Lodoe, AIDA, Jumpei, TUSCHL, Thomas, GLICKMAN, J.Fraser, ASANO, Yasutomi, IMAEDA, Toshihiro, MILLER, Michael, KAMEL, Taku, HASHIZUME, Shogo, KUROITA, Takanobu, TOMITA, Daisuke, MICHINO, Mayako
Year of Publication 16.11.2022
Get full text
Year of Publication 16.11.2022
Patent
1-((1H-PYRAZOL-4-YL)METHYL)-3-(PHENYL)-1,3-DIHYDRO-2H-IMIDAZOL-2-ONE DERIVATIVES AND RELATED COMPOUNDS AS GPR139 ANTAGONISTS FOR THE TREATMENT OF E.G. DEPRESSION
HASUI, Tomoaki, NAKAMURA, Shinji, TAKAMI, Kazuaki, TAKASHIMA, Sachie, YAMAGUCHI, Fumie, NAKAMURA, Minoru, DAINI, Masaki, YAMASHITA, Toru, IMAEDA, Toshihiro, MIKAMI, Satoshi, KAKEI, Hiroyuki, WANG, Chunxiang, HASHIZUME, Shogo, MORIMOTO, Shinji
Year of Publication 25.11.2021
Get full text
Year of Publication 25.11.2021
Patent
Substituted pyrido[4,3-b]indoles and azepino[4,5-b]indoles as inhibitors of cGAS
Okamoto, Rei, Kuroita, Takanobu, Tuschl, Thomas, Glickman, J. Fraser, Michino, Mayako, Lama, Lodoe, Kamei, Taku, Miller, Michael, Asano, Yasutomi, Tomita, Daisuke, Patel, Dinshaw, Aida, Jumpei, Imaeda, Toshihiro, Hashizume, Shogo
Year of Publication 16.08.2022
Get full text
Year of Publication 16.08.2022
Patent
INHIBITORS OF cGAS FOR TREATING AUTOINFLAMMATORY DISEASES AND CANCER METASTASIS
OKAMOTO, Rei, PATEL, Dinshaw, LAMA, Lodoe, KAMEI, Taku, AIDA, Jumpei, TUSCHL, Thomas, GLICKMAN, J. Fraser, ASANO, Yasutomi, IMAEDA, Toshihiro, MILLER, Michael, HASHIZUME, Shogo, KUROITA, Takanobu, TOMITA, Daisuke, MICHINO, Mayako
Year of Publication 16.06.2022
Get full text
Year of Publication 16.06.2022
Patent
2,3,4,5-TETRAHYDRO-1H-PYRIDO[4, 3-B]INDOLE INHIBITORS OF CGAS FOR TREATING AUTOINFLAMMATORY DISEASES
OKAMOTO, Rei, PATEL, Dinshaw, LAMA, Lodoe, KAMEI, Taku, AIDA, Jumpei, TUSCHL, Thomas, GLICKMAN, J. Fraser, ASANO, Yasutomi, IMAEDA, Toshihiro, MILLER, Michael, HASHIZUME, Shogo, KUROITA, Takanobu, TOMITA, Daisuke, MICHINO, Mayako
Year of Publication 30.03.2022
Get full text
Year of Publication 30.03.2022
Patent
INHIBITORS OF CGAS FOR TREATING AUTOINFLAMMATORY DISEASES AND CANCER METASTASIS
Okamoto, Rei, Kuroita, Takanobu, Tuschl, Thomas, Glickman, J. Fraser, Michino, Mayako, Lama, Lodoe, Kamei, Taku, Miller, Michael, Asano, Yasutomi, Tomita, Daisuke, Patel, Dinshaw, Aida, Jumpei, Imaeda, Toshihiro, Hashizume, Shogo
Year of Publication 19.01.2022
Get full text
Year of Publication 19.01.2022
Patent
2,3,4,5-TETRAHYDRO-1H-PYRIDO[4, 3-B]INDOLE INHIBITORS OF CGAS FOR TREATING AUTOINFLAMMATORY DISEASES
OKAMOTO, Rei, PATEL, Dinshaw, LAMA, Lodoe, KAMEI, Taku, AIDA, Jumpei, TUSCHL, Thomas, GLICKMAN, J. Fraser, ASANO, Yasutomi, IMAEDA, Toshihiro, MILLER, Michael, HASHIZUME, Shogo, KUROITA, Takanobu, TOMITA, Daisuke, MICHINO, Mayako
Year of Publication 01.09.2021
Get full text
Year of Publication 01.09.2021
Patent
2,3,4,5-TETRAHYDRO-1H-PYRIDO[4, 3-b]INDOLE INHIBITORS OF cGAS FOR TREATING AUTOINFLAMMATORY DISEASES
OKAMOTO, Rei, PATEL, Dinshaw, LAMA, Lodoe, KAMEI, Taku, AIDA, Jumpei, TUSCHL, Thomas, GLICKMAN, J. Fraser, ASANO, Yasutomi, IMAEDA, Toshihiro, MILLER, Michael, HASHIZUME, Shogo, KUROITA, Takanobu, TOMITA, Daisuke, MICHINO, Mayako
Year of Publication 27.05.2021
Get full text
Year of Publication 27.05.2021
Patent
2,3,4,5-TETRAHYDRO-1H-PYRIDO[4, 3-B]INDOLE INHIBITORS OF CGAS FOR TREATING AUTOINFLAMMATORY DISEASES
OKAMOTO, Rei, PATEL, Dinshaw, LAMA, Lodoe, KAMEI, Taku, AIDA, Jumpei, TUSCHL, Thomas, GLICKMAN, J. Fraser, ASANO, Yasutomi, IMAEDA, Toshihiro, MILLER, Michael, HASHIZUME, Shogo, KUROITA, Takanobu, TOMITA, Daisuke, MICHINO, Mayako
Year of Publication 16.12.2020
Get full text
Year of Publication 16.12.2020
Patent
INHIBITORS OF CGAS FOR TREATING AUTOINFLAMMATORY DISEASES AND CANCER METASTASIS
KUROITA, TAKANOBU, ASANO, YASUTOMI, GLICKMAN, J. FRASER, HASHIZUME, SHOGO, MICHINO, MAYAKO, IMAEDA, TOSHIHIRO, LAMA, LODOE, MILLER, MICHAEL, PATEL, DINSHAW, OKAMOTO, REI, TOMITA, DAISUKE, TUSCHL, THOMAS, AIDA, JUMPEI, KAMEI, TAKU
Year of Publication 17.09.2020
Get full text
Year of Publication 17.09.2020
Patent
INHIBITORS OF CGAS FOR TREATING AUTOINFLAMMATORY DISEASES AND CANCER METASTASIS
OKAMOTO, Rei, PATEL, Dinshaw, LAMA, Lodoe, KAMEI, Taku, AIDA, Jumpei, TUSCHL, Thomas, GLICKMAN, J. Fraser, ASANO, Yasutomi, IMAEDA, Toshihiro, MILLER, Michael, HASHIZUME, Shogo, KUROITA, Takanobu, TOMITA, Daisuke, MICHINO, Mayako
Year of Publication 17.09.2020
Get full text
Year of Publication 17.09.2020
Patent