Optimization of N'-(arylsulfonyl)pyrazoline-1-carboxamidines by exploiting a novel interaction site in the 5-HT sub(6) antagonistic binding pocket
Loevezijn, Arnold van, Venhorst, Jennifer, Bakker, Wouter IIwema, Lange, Jos HM, Looff, Wouter de, Henzen, Remco, Vries, Jelle de, Woestijne, Rob Pvan de, Hartog, Arnold Pden, Verhoog, Stefan, van der Neut, Martina AW, Bruin, Natasja MWJde, Kruse, Chris G
Published in Bioorganic & medicinal chemistry letters (15.03.2016)
Published in Bioorganic & medicinal chemistry letters (15.03.2016)
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Synthesis, SAR and intramolecular hydrogen bonding pattern of 1,3,5-trisubstituted 4,5-dihydropyrazoles as potent cannabinoid CB sub(1) receptor antagonists
Lange, Jos HM, Van der Neut, Martina AW, Hartog, Arnold Pden, Wals, Henri C, Hoogendoorn, Jan, Van Stuivenberg, Herman H, Van Vliet, Bernard J, Kruse, Chris G
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
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Synthesis and SAR of novel imidazoles as potent and selective cannabinoid CB sub(2) receptor antagonists with high binding efficiencies
Lange, Jos HM, Van der Neut, Martina AW, Wals, Henri C, Kuil, Gijs D, Borst, Alice JM, Mulder, Arie, Hartog, Arnold Pden, Zilaout, Hicham, Goutier, Wouter, Van Stuivenberg, Herman H, Van Vliet, Bernard J
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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7-Azaindole derivatives as potential partial nicotinic agonists
Stoit, Axel R., den Hartog, Arnold P., Mons, Harry, van Schaik, Sjoerd, Barkhuijsen, Nynke, Stroomer, Cees, Coolen, Hein K.A.C., Reinders, Jan Hendrik, Adolfs, Tiny J.P., van der Neut, Martina, Keizer, Hiskias, Kruse, Chris G.
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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