Development of Potent Thrombin Receptor Antagonist Peptides
Bernatowicz, Michael S, Klimas, Clifford E, Hartl, Karen S, Peluso, Marianne, Allegretto, Nick J, Seiler, Steven M
Published in Journal of medicinal chemistry (06.12.1996)
Published in Journal of medicinal chemistry (06.12.1996)
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Pharmacological characterization of potent, long-acting thromboxane receptor antagonists, SQ 33,261 and SQ 33,552
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Published in The Journal of pharmacology and experimental therapeutics (01.04.1992)
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Published in The Journal of pharmacology and experimental therapeutics (01.04.1992)
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Prostacyclin agonists reduce early atherosclerosis in hyperlipidemic hamsters. Octimibate and BMY 42393 suppress monocyte chemotaxis, macrophage cholesteryl ester accumulation, scavenger receptor activity, and tumor necrosis factor production
Kowala, M C, Mazzucco, C E, Hartl, K S, Seiler, S M, Warr, G A, Abid, S, Grove, R I
Published in Arteriosclerosis and thrombosis (01.03.1993)
Published in Arteriosclerosis and thrombosis (01.03.1993)
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Isolation and identification of lysophosphatidylcholines as endogenous modulators of thromboxane receptors
Phillipson, D W, Tymiak, A A, Tuttle, J G, Hartl, K S, Harper, T W, Bolgar, M S, Allen, G T, Ogletree, M L
Published in Journal of lipid mediators (01.06.1993)
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Published in Journal of lipid mediators (01.06.1993)
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Nonprostanoid prostacyclin mimetics. 4. Derivatives of 2-[3-[2-(4,5-diphenyl-2-oxazolyl)ethyl]phenoxy]acetic acid substituted .alpha. to the oxazole ring
Meanwell, Nicholas A, Rosenfeld, Michael J, Wright, J. J. Kim, Brassard, Catherine L, Buchanan, John O, Federici, Marianne E, Fleming, J. Stuart, Gamberdella, Marianne, Hartl, Karen S
Published in Journal of medicinal chemistry (26.11.1993)
Published in Journal of medicinal chemistry (26.11.1993)
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Nonprostanoid prostacyclin mimetics. 5. Structure-activity relationships associated with [3-[4-(4,5-diphenyl-2-oxazolyl)-5-oxazolyl]phenoxy]acetic acid
Meanwell, Nicholas A, Romine, Jeffrey L, Rosenfeld, Michael J, Martin, Scott W, Trehan, Ashok K, Wright, J. J. Kim, Malley, Mary F, Gougoutas, Jack Z, Brassard, Catherine L
Published in Journal of medicinal chemistry (26.11.1993)
Published in Journal of medicinal chemistry (26.11.1993)
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Non-prostanoid prostacyclin mimetics. 6. Derivatives of 2-[3-[2-(4,5-Diphenyl-2-oxazolyl)ethyl]phenoxy]acetic acid modified beta-to the oxazole ring
Meanwell, N A, Rosenfeld, M J, Trehan, A K, Wright, J J, Brassard, C L, Buchanan, J O, Federici, M E, Fleming, J S, Gamberdella, M, Hartl, K S
Published in Drug design and discovery (01.01.1994)
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Published in Drug design and discovery (01.01.1994)
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Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors
SUTTON, James C, BOLTON, Scott A, BISACCHI, Gregory S, DAVIS, Malcolm E, HARTL, Karen S, JACOBSON, Bruce, MATHUR, Arvind, OGLETREE, Martin L, SLUSARCHYK, William A, ZAHLER, Robert, SEILER, Steven M
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors
Sutton, James C, Bolton, Scott A, Hartl, Karen S, Huang, Ming-Hsing, Jacobs, Glenn, Meng, Wei, Ogletree, Martin L, Pi, Zulan, Schumacher, William A, Seiler, Steven M, Slusarchyk, William A, Treuner, Uwe, Zahler, Robert, Zhao, Guohua, Bisacchi, Gregory S
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
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Synthesis of potent and highly selective inhibitors of human tryptase
Slusarchyk, William A., Bolton, Scott A., Hartl, Karen S., Huang, Ming-Hsing, Jacobs, Glenn, Meng, Wei, Ogletree, Martin L., Pi, Zulan, Schumacher, William A., Seiler, Steven M., Sutton, James C., Treuner, Uwe, Zahler, Robert, Zhao, Guohua, Bisacchi, Gregory S.
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
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Synthesis of potent and highly selective nonguanidine azetidinone inhibitors of human tryptase
BISACCHI, Gregory S, SLUSARCHYK, William A, TREUNER, Uwe, ZAHLER, Robert, GUOHUA ZHAO, SEILER, Steven M, BOLTON, Scott A, HARTL, Karen S, JACOBS, Glenn, MATHUR, Arvind, WEI MENG, OGLETREE, Martin L, ZULAN PI, SUTTON, James C
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Synthesis of potent and selective 2-azepanone inhibitors of human tryptase
Zhao, Guohua, Bolton, Scott A., Kwon, Chet, Hartl, Karen S., Seiler, Steven M., Slusarchyk, William A., Sutton, James C., Bisacchi, Gregory S.
Published in Bioorganic & medicinal chemistry letters (19.01.2004)
Published in Bioorganic & medicinal chemistry letters (19.01.2004)
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Nonprostanoid prostacyclin mimetics. IV: Derivatives of 2-[3-[2-(4,5-diphenyl-2-oxazolyl)ethyl]phenoxy]acetic acid substituted α to the oxazole ring
MEANWELL, N. A, ROSENFELD, M. J, SEILER, S. M, WRIGHT, J. J. K, BRASSARD, C. L, BUCHANAN, J. O, FEDERICI, M. E, FLEMING, J. S, GAMBERDELLA, M, HARTL, K. S, ZAVOICO, G. B
Published in Journal of medicinal chemistry (1993)
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Published in Journal of medicinal chemistry (1993)
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Nonprostanoid prostacyclin mimetics. V: Structure-activity relationships associated with [3-[4-(4,5-diphenyl-2-oxazolyl)-5-oxazolyl]phenoxy]acetic acid
MEANWELL, N. A, ROMINE, J. L, FEDERICI, M. E, FLEMING, J. S, GAMBERDELLA, M, HARTL, K. S, ZAVOICO, G. B, SEILER, S. M, ROSENFELD, M. J, MARTIN, S. W, TREHAN, A. K, WRIGHT, J. J. K, MALLEY, M. F, GOUGOUTAS, J. Z, BRASSARD, C. L, BUCHANAN, J. O
Published in Journal of medicinal chemistry (1993)
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Published in Journal of medicinal chemistry (1993)
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