Phase I and pharmacokinetic study of an oral platinum complex given daily for 5 days in patients with cancer
McKeage, M J, Raynaud, F, Ward, J, Berry, C, O'Dell, D, Kelland, L R, Murrer, B, Santabárabara, P, Harrap, K R, Judson, I R
Published in Journal of clinical oncology (01.07.1997)
Published in Journal of clinical oncology (01.07.1997)
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Reduced drug accumulation as a major mechanism of acquired resistance to cisplatin in a human ovarian carcinoma cell line: circumvention studies using novel platinum (II) and (IV) ammine/amine complexes
LOH, S. Y, MISTRY, P, KELLAND, L. R, ABEL, G, HARRAP, K. R
Published in British journal of cancer (01.12.1992)
Published in British journal of cancer (01.12.1992)
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Phase I trial of ZD1694, a new folate-based thymidylate synthase inhibitor, in patients with solid tumors
Clarke, S J, Hanwell, J, de Boer, M, Planting, A, Verweij, J, Walker, M, Smith, R, Jackman, A L, Hughes, L R, Harrap, K R, Kennealey, G T, Judson, I R
Published in Journal of clinical oncology (01.05.1996)
Published in Journal of clinical oncology (01.05.1996)
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Preclinical antitumor evaluation of bis-acetato-ammine-dichloro-cyclohexylamine platinum(IV) : an orally active platinum drug
KELLAND, L. R, ABEL, G, MCKEAGE, M. J, JONES, M, GODDARD, P. M, VALENTI, M, MURRER, B. A, HARRAP, K. R
Published in Cancer research (Chicago, Ill.) (01.06.1993)
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Published in Cancer research (Chicago, Ill.) (01.06.1993)
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A novel trans-platinum coordination complex possessing in vitro and in vivo antitumor activity
KELLAND, L. R, BARNARD, C. F. J, MELLISH, K. J, JONES, M, GODDARD, P. M, VALENTI, M, BRYANT, A, MURRER, B. A, HARRAP, K. R
Published in Cancer research (Chicago, Ill.) (01.11.1994)
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Published in Cancer research (Chicago, Ill.) (01.11.1994)
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Ammine/amine platinum(IV) dicarboxylates : a novel class of platinum complex exhibiting selective cytotoxicity to intrinsically cisplatin-resistant human ovarian carcinoma cell lines
KELLAND, L. R, MURRER, B. A, ABEL, G, GIANDOMENICO, C. M, MISTRY, P, HARRAP, K. R
Published in Cancer research (Chicago, Ill.) (15.02.1992)
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Published in Cancer research (Chicago, Ill.) (15.02.1992)
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ZD1694 (Tomudex): A new thymidylate synthase inhibitor with activity in colorectal cancer
Jackman, A.L, Farrugia, D.C, Gibson, W, Kimbell, R, Harrap, K.R, Stephens, T.C, Azab, M, Boyle, F.T
Published in European journal of cancer (1990) (01.07.1995)
Published in European journal of cancer (1990) (01.07.1995)
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Genomic Imbalances Associated with Acquired Resistance to Platinum Analogues
Leyland-Jones, Brian, Kelland, Lloyd R., Harrap, Kenneth R., Hiorns, Lynne R.
Published in The American journal of pathology (01.07.1999)
Published in The American journal of pathology (01.07.1999)
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Lack of nephrotoxicity of oral ammine/amine platinum (IV) dicarboxylate complexes in rodents
MCKEAGE, M. J, MORGAN, S. E, BOXALL, F. E, MURRER, B. A, HARD, G. C, HARRAP, K. R
Published in British journal of cancer (01.05.1993)
Published in British journal of cancer (01.05.1993)
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Metabolic studies of an orally active platinum anticancer drug by liquid chromatography-electrospray ionization mass spectrometry
Poon, G.K., Raynaud, F.I., Mistry, P., Odell, D.E., Kelland, L.R., Harrap, K.R., Barnard, C.F.J., Murrer, B.A.
Published in Journal of Chromatography A (29.09.1995)
Published in Journal of Chromatography A (29.09.1995)
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The cytotoxic action of four ammine/amine platinum(IV) dicarboxylates: a flow cytometric study
ORMEROD, M. G, ORR, R. M, O'NEILL, C. F, CHWALINSKI, T, TITLEY, J. C, KELLAND, L. R, HARRAP, K. R
Published in British journal of cancer (01.12.1996)
Published in British journal of cancer (01.12.1996)
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